AR027537A1 - Un nuevo procedimiento para la preparacion de isoindolina - Google Patents
Un nuevo procedimiento para la preparacion de isoindolinaInfo
- Publication number
- AR027537A1 AR027537A1 ARP010100820A ARP010100820A AR027537A1 AR 027537 A1 AR027537 A1 AR 027537A1 AR P010100820 A ARP010100820 A AR P010100820A AR P010100820 A ARP010100820 A AR P010100820A AR 027537 A1 AR027537 A1 AR 027537A1
- Authority
- AR
- Argentina
- Prior art keywords
- isoindolin
- preparation
- new procedure
- synthesis
- procedure
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Endocrinology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Indole Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Procedimiento para la síntesis industrial de isoindolina por hidrogenacion catalítica de ftalonitrilo. Aplicacion en la síntesis del ácido2-(S)-bencil-4-oxo-4-(cis-perhidroisoindol-2-il)-butírico, sus sales farmacéuticamente aceptables y sus hidratos
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0002383A FR2805535B1 (fr) | 2000-02-25 | 2000-02-25 | Nouveau procede de preparation de l'isoindoline |
Publications (1)
Publication Number | Publication Date |
---|---|
AR027537A1 true AR027537A1 (es) | 2003-04-02 |
Family
ID=8847398
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP010100820A AR027537A1 (es) | 2000-02-25 | 2001-02-23 | Un nuevo procedimiento para la preparacion de isoindolina |
Country Status (23)
Country | Link |
---|---|
US (1) | US6320058B2 (es) |
EP (1) | EP1127876B1 (es) |
JP (1) | JP3545351B2 (es) |
KR (1) | KR100464183B1 (es) |
CN (1) | CN1197848C (es) |
AR (1) | AR027537A1 (es) |
AT (1) | ATE227707T1 (es) |
AU (1) | AU774807B2 (es) |
BR (1) | BR0100757A (es) |
CA (1) | CA2338899C (es) |
DE (1) | DE60100044T2 (es) |
DK (1) | DK1127876T3 (es) |
EA (1) | EA003515B1 (es) |
ES (1) | ES2187492T3 (es) |
FR (1) | FR2805535B1 (es) |
HK (1) | HK1040248B (es) |
HU (1) | HUP0100881A3 (es) |
NO (1) | NO318881B1 (es) |
NZ (1) | NZ510205A (es) |
PL (1) | PL346035A1 (es) |
PT (1) | PT1127876E (es) |
SI (1) | SI1127876T1 (es) |
ZA (1) | ZA200101529B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1787983B1 (en) * | 2004-08-16 | 2011-03-09 | Eisai R&D Management Co., Ltd. | Methods for producing isoindole derivatives |
CN1324010C (zh) * | 2005-01-12 | 2007-07-04 | 江苏省药物研究所 | 一种米格列奈的制备方法 |
CN100441570C (zh) * | 2006-05-24 | 2008-12-10 | 严洁 | 一种米格列奈钙的制备及质量控制方法 |
FR2967673B1 (fr) * | 2010-11-24 | 2012-12-28 | Minakem | Synthese de n-heterocycles par alkylation reductrice de derives cyanes |
EP2800739B1 (en) | 2012-01-06 | 2015-12-23 | Lonza Ltd | Method for preparation of octahydrocyclopenta[c]pyrrole |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2773902A (en) * | 1954-05-10 | 1956-12-11 | California Research Corp | Hydrogenation of phthalonitriles |
US4254059A (en) * | 1979-08-01 | 1981-03-03 | Allied Chemical Corporation | Process for hydrogenation of nitriles |
-
2000
- 2000-02-25 FR FR0002383A patent/FR2805535B1/fr not_active Expired - Fee Related
-
2001
- 2001-02-16 CA CA002338899A patent/CA2338899C/fr not_active Expired - Fee Related
- 2001-02-16 US US09/785,956 patent/US6320058B2/en not_active Expired - Fee Related
- 2001-02-19 JP JP2001041119A patent/JP3545351B2/ja not_active Expired - Fee Related
- 2001-02-22 PL PL01346035A patent/PL346035A1/xx not_active IP Right Cessation
- 2001-02-23 DK DK01400484T patent/DK1127876T3/da active
- 2001-02-23 EP EP01400484A patent/EP1127876B1/fr not_active Expired - Lifetime
- 2001-02-23 ZA ZA200101529A patent/ZA200101529B/xx unknown
- 2001-02-23 ES ES01400484T patent/ES2187492T3/es not_active Expired - Lifetime
- 2001-02-23 PT PT01400484T patent/PT1127876E/pt unknown
- 2001-02-23 SI SI200130006T patent/SI1127876T1/xx unknown
- 2001-02-23 AR ARP010100820A patent/AR027537A1/es active IP Right Grant
- 2001-02-23 BR BR0100757-2A patent/BR0100757A/pt not_active Application Discontinuation
- 2001-02-23 DE DE60100044T patent/DE60100044T2/de not_active Expired - Fee Related
- 2001-02-23 NZ NZ510205A patent/NZ510205A/xx unknown
- 2001-02-23 CN CNB011168773A patent/CN1197848C/zh not_active Expired - Fee Related
- 2001-02-23 AU AU23237/01A patent/AU774807B2/en not_active Ceased
- 2001-02-23 KR KR10-2001-0009248A patent/KR100464183B1/ko not_active IP Right Cessation
- 2001-02-23 AT AT01400484T patent/ATE227707T1/de not_active IP Right Cessation
- 2001-02-23 NO NO20010936A patent/NO318881B1/no not_active IP Right Cessation
- 2001-02-23 HU HU0100881A patent/HUP0100881A3/hu unknown
- 2001-02-26 EA EA200100179A patent/EA003515B1/ru unknown
-
2002
- 2002-03-14 HK HK02101967.5A patent/HK1040248B/zh not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CR11780A (es) | Nuevo proceso para la sintesis de ivabradina y sales de adicion resultantes con un acido farmaceuticamente aceptable (solicitud divisonal) | |
UY28360A1 (es) | Nuevos compuestos | |
PA8518801A1 (es) | Derivados de 2-aminocarbonil-9h-purina | |
ES2187261B2 (es) | Compuestos de eteres y amidas y su preparacion, como agentes anti-diabeticos. | |
CY1108101T1 (el) | Ενωσεις πυριμιδινης και η χρηση τους στην παρασκευη ενος τριαζολο-πυριμιδιν καρβα νουκλεοζιτη | |
BRPI0820474B8 (pt) | uso do composto 1-[2-(2,4-dimetil-fenil-sulfanil)-fenil]-piperazina ou de sais farmaceuticamente aceitáveis do mesmo | |
UY32649A (es) | "sales de 4-(dimetilamino)butil 2-(4-((2-amino-4-metil-6-(pentilamino)pirimidin-5-il)metil)fenil)acetato" | |
UY28348A1 (es) | Compuestos novedosos | |
BR0114903A (pt) | 7-azaindóis, sua aplicação como inibidores da fosfodiesterase 4 e processos para a sua preparação | |
AP2003002856A0 (en) | Broadspectrum 2-(substitutted-amino)-benzothiazolesulphonamide HIV protease inhibitors. | |
AR027537A1 (es) | Un nuevo procedimiento para la preparacion de isoindolina | |
HN1998000167A (es) | Nuevo procedimiento para preparar una cetoimina | |
BRPI0414107B8 (pt) | produtos intermediários para a preparação de híbridos de oxazolidinon-quinolona | |
UY25357A1 (es) | Nuevos pentasacáridos, procedimiento para su preparación y composiciones farmacéuticas que los contienen. | |
BR0115301A (pt) | Uso de um inibidor seletivo da recaptação de norepinefrina | |
UY26556A1 (es) | Compuestos calcilíticos | |
DE50101838D1 (de) | Verbessertes Verfahren zur Herstellung von 2-(4-Trifluormethoxyphenyl)ethylamin | |
AR023788A1 (es) | Modificacion amorfa de torasemida | |
HN1999000043A (es) | Procedimiento para alquilar sulfonamidas impedidas estericamente. | |
HN2001000172A (es) | Proceso para preparar 2 - (4 - piridil)amino - 6 - dialquiloxifenil pirido [2,3 - d]pirimidin - 7 - onas. | |
AR031972A1 (es) | Composicion farmaceutica solida termoformable para la liberacion controlada de perindopril | |
AR032049A1 (es) | Una composicion farmaceutica solida termoformable para la liberacion controlada de trimetazidina | |
ATE232525T1 (de) | Enanthioauswählende synthese | |
BR0105939A (pt) | Método para a produção de derivados de citidina | |
ECSP993045A (es) | Derivados de acridina, procedimiento para su preparacion y su utilizacion como analgesico |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant, registration |