AP3225A - New combination between 4-{3-[CIS-hexahydrocyclopenta[C]pyrrol-2(1H)-yl]propoxy}benzamide and an NMDA receptor antagonist, and pharmaceutical compositions containing it - Google Patents
New combination between 4-{3-[CIS-hexahydrocyclopenta[C]pyrrol-2(1H)-yl]propoxy}benzamide and an NMDA receptor antagonist, and pharmaceutical compositions containing itInfo
- Publication number
- AP3225A AP3225A AP2012006607A AP2012006607A AP3225A AP 3225 A AP3225 A AP 3225A AP 2012006607 A AP2012006607 A AP 2012006607A AP 2012006607 A AP2012006607 A AP 2012006607A AP 3225 A AP3225 A AP 3225A
- Authority
- AP
- ARIPO
- Prior art keywords
- hexahydrocyclopenta
- pyrrol
- benzamide
- propoxy
- cis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1103777A FR2983732B1 (fr) | 2011-12-09 | 2011-12-09 | Nouvelle association entre le 4-{3-[cis-hexahydrocyclopenta[c]pyrrol-2(1h)-yl]propoxy}pharmaceutiques qui la contiennent |
Publications (2)
Publication Number | Publication Date |
---|---|
AP2012006607A0 AP2012006607A0 (en) | 2012-12-31 |
AP3225A true AP3225A (en) | 2015-04-30 |
Family
ID=47682151
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2012006607A AP3225A (en) | 2011-12-09 | 2012-12-05 | New combination between 4-{3-[CIS-hexahydrocyclopenta[C]pyrrol-2(1H)-yl]propoxy}benzamide and an NMDA receptor antagonist, and pharmaceutical compositions containing it |
Country Status (27)
Country | Link |
---|---|
US (2) | US8921409B2 (xx) |
EP (1) | EP2601942A1 (xx) |
JP (1) | JP5591310B2 (xx) |
KR (1) | KR101489670B1 (xx) |
CN (1) | CN103157111B (xx) |
AP (1) | AP3225A (xx) |
AR (1) | AR089112A1 (xx) |
AU (1) | AU2012258339A1 (xx) |
BR (1) | BR102012031031A2 (xx) |
CA (1) | CA2798549A1 (xx) |
CL (1) | CL2012003437A1 (xx) |
CO (2) | CO6660080A1 (xx) |
CR (1) | CR20120608A (xx) |
EA (1) | EA201201530A1 (xx) |
EC (1) | ECSP12012329A (xx) |
FR (1) | FR2983732B1 (xx) |
GT (1) | GT201200329A (xx) |
MA (1) | MA34867B1 (xx) |
MD (1) | MD4348B1 (xx) |
MX (1) | MX2012014184A (xx) |
NI (1) | NI201200178A (xx) |
PE (1) | PE20130813A1 (xx) |
SG (1) | SG191494A1 (xx) |
TN (1) | TN2012000563A1 (xx) |
TW (1) | TWI457123B (xx) |
UY (1) | UY34475A (xx) |
WO (1) | WO2013083887A1 (xx) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR3003466B1 (fr) * | 2013-03-22 | 2015-08-07 | Servier Lab | Utilisation du 4-{3-[cis-hexahydrocyclopenta[c]pyrrol-2(1h)-yl]propoxy}benzamide pour le traitement des douleurs neuropathiques |
KR101484405B1 (ko) * | 2013-08-14 | 2015-01-19 | 서울대학교산학협력단 | Ninjurin1 결핍 유래의 강박증 예방 또는 치료용 약학적 조성물 |
GB201509134D0 (en) * | 2015-05-28 | 2015-07-15 | Electrophoretics Ltd | Biomolecules involved in Alzheimer's disease |
JP7429942B2 (ja) * | 2015-07-22 | 2024-02-09 | アナベックス ライフ サイエンシズ コーポレイション | テトラヒドロ-n,n-ジメチル-2,2-ジフェニル-3-フランメタンアミン(anavex2-73)のエナンチオマーならびにシグマ1レセプターにより調節されるアルツハイマー型および他の傷害の処置におけるその使用 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE60324788D1 (de) * | 2002-05-31 | 2009-01-02 | Lundbeck & Co As H | Kombination aus einem nmda-antagonist und acetylcholinesterase-hemmern zur behandlung der alzheimer-krankheit |
KR20070104480A (ko) * | 2003-05-27 | 2007-10-25 | 포레스트 래보러토리즈, 인코포레이티드 | 우울증 및 그 밖의 기분장애의 치료를 위한 nmda수용체 길항제 및 선택적 세로토닌 재흡수 억제제의 배합물 |
US7432280B2 (en) * | 2003-06-20 | 2008-10-07 | Eli Lilly And Company | 3-aminopiperidines and 3-aminoquinuclidines as inhibitors of monoamine uptake |
WO2005067908A2 (en) * | 2004-01-05 | 2005-07-28 | Merz Pharma Gmbh & Co. Kgaa | Memantine for the treatment of mild and mild-to-moderate alzheimer’s disease |
FR2866647B1 (fr) * | 2004-02-20 | 2006-10-27 | Servier Lab | Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
TW200531680A (en) * | 2004-03-03 | 2005-10-01 | Merz Pharma Gmbh & Co Kgaa | Therapy using 1-aminocyclohexane derivatives for the treatment of behavioral disorders associated with alzheimer's disease |
JP2007529556A (ja) * | 2004-03-19 | 2007-10-25 | アクソニクス インコーポレイテッド | 認知障害の処置に有用なアセチルコリンエステラーゼ阻害剤およびn−メチル−d−アスパラギン酸拮抗剤 |
FR2937119B1 (fr) | 2008-10-15 | 2010-12-17 | Air Liquide | Procede de production d'energie et capture de co2 |
FR2937251B1 (fr) * | 2008-10-16 | 2011-03-18 | Servier Lab | Utilisation du 4-{3-°hexahydrocyclopenta°c!pyrrol-2(1h)-yl! propoxy}benzamide pour l'obtention de medicaments destines au traitement des troubles du sommeil |
FR2953515B1 (fr) * | 2009-12-09 | 2011-12-23 | Servier Lab | Nouveaux derives du type hexahydrocyclopenta[b]pyrrole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2011
- 2011-12-09 FR FR1103777A patent/FR2983732B1/fr not_active Expired - Fee Related
-
2012
- 2012-04-27 CO CO12069442A patent/CO6660080A1/es unknown
- 2012-11-28 AU AU2012258339A patent/AU2012258339A1/en not_active Abandoned
- 2012-11-28 UY UY0001034475A patent/UY34475A/es unknown
- 2012-11-28 PE PE2012002234A patent/PE20130813A1/es not_active Application Discontinuation
- 2012-11-29 TN TNP2012000563A patent/TN2012000563A1/fr unknown
- 2012-11-29 SG SG2012087771A patent/SG191494A1/en unknown
- 2012-12-03 CR CR20120608A patent/CR20120608A/es unknown
- 2012-12-03 NI NI201200178A patent/NI201200178A/es unknown
- 2012-12-03 MA MA35425A patent/MA34867B1/fr unknown
- 2012-12-03 MD MDA20120119A patent/MD4348B1/ro not_active IP Right Cessation
- 2012-12-05 MX MX2012014184A patent/MX2012014184A/es not_active Application Discontinuation
- 2012-12-05 BR BR102012031031-7A patent/BR102012031031A2/pt not_active Application Discontinuation
- 2012-12-05 AP AP2012006607A patent/AP3225A/xx active
- 2012-12-06 JP JP2012267342A patent/JP5591310B2/ja not_active Expired - Fee Related
- 2012-12-06 CL CL2012003437A patent/CL2012003437A1/es unknown
- 2012-12-06 KR KR20120141338A patent/KR101489670B1/ko not_active IP Right Cessation
- 2012-12-06 CO CO12221472A patent/CO6690116A1/es unknown
- 2012-12-06 US US13/706,828 patent/US8921409B2/en not_active Expired - Fee Related
- 2012-12-06 CA CA2798549A patent/CA2798549A1/fr not_active Abandoned
- 2012-12-06 TW TW101145875A patent/TWI457123B/zh not_active IP Right Cessation
- 2012-12-07 WO PCT/FR2012/000505 patent/WO2013083887A1/fr active Application Filing
- 2012-12-07 EA EA201201530A patent/EA201201530A1/ru unknown
- 2012-12-07 EP EP12195997.7A patent/EP2601942A1/fr not_active Withdrawn
- 2012-12-07 AR ARP120104595A patent/AR089112A1/es unknown
- 2012-12-07 EC ECSP12012329 patent/ECSP12012329A/es unknown
- 2012-12-07 GT GT201200329A patent/GT201200329A/es unknown
- 2012-12-10 CN CN201210530112.9A patent/CN103157111B/zh not_active Expired - Fee Related
-
2014
- 2014-11-25 US US14/553,206 patent/US20150080448A1/en not_active Abandoned
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