AP2005003376A0 - Triazole compounds useful in therapy. - Google Patents

Triazole compounds useful in therapy.

Info

Publication number
AP2005003376A0
AP2005003376A0 AP2005003376A AP2005003376A AP2005003376A0 AP 2005003376 A0 AP2005003376 A0 AP 2005003376A0 AP 2005003376 A AP2005003376 A AP 2005003376A AP 2005003376 A AP2005003376 A AP 2005003376A AP 2005003376 A0 AP2005003376 A0 AP 2005003376A0
Authority
AP
ARIPO
Prior art keywords
therapy
compounds useful
triazole compounds
triazole
useful
Prior art date
Application number
AP2005003376A
Other languages
English (en)
Inventor
Stephen Bryans Justin
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0303852.8A external-priority patent/GB0303852D0/en
Priority claimed from GBGB0317227.7A external-priority patent/GB0317227D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of AP2005003376A0 publication Critical patent/AP2005003376A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2333/00—Assays involving biological materials from specific organisms or of a specific nature
    • G01N2333/435—Assays involving biological materials from specific organisms or of a specific nature from animals; from humans
    • G01N2333/705—Assays involving receptors, cell surface antigens or cell surface determinants
    • G01N2333/72—Assays involving receptors, cell surface antigens or cell surface determinants for hormones
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2500/00—Screening for compounds of potential therapeutic value
    • G01N2500/04—Screening involving studying the effect of compounds C directly on molecule A (e.g. C are potential ligands for a receptor A, or potential substrates for an enzyme A)

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Child & Adolescent Psychology (AREA)
  • Oncology (AREA)
AP2005003376A 2003-02-19 2004-02-09 Triazole compounds useful in therapy. AP2005003376A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0303852.8A GB0303852D0 (en) 2003-02-19 2003-02-19 Triazole compounds useful in therapy
GBGB0317227.7A GB0317227D0 (en) 2003-07-23 2003-07-23 Treatment of male sexual dysfunction
PCT/IB2004/000432 WO2004074291A1 (en) 2003-02-19 2004-02-09 Triazole compounds useful in therapy

Publications (1)

Publication Number Publication Date
AP2005003376A0 true AP2005003376A0 (en) 2005-09-30

Family

ID=34889119

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2005003376A AP2005003376A0 (en) 2003-02-19 2004-02-09 Triazole compounds useful in therapy.

Country Status (25)

Country Link
EP (1) EP1597260B1 (ja)
JP (2) JP4033886B2 (ja)
KR (1) KR100750028B1 (ja)
AP (1) AP2005003376A0 (ja)
AT (1) ATE349449T1 (ja)
AU (1) AU2004213242B2 (ja)
BR (1) BRPI0407676A (ja)
CA (1) CA2516557C (ja)
DE (1) DE602004003914T2 (ja)
DK (1) DK1597260T3 (ja)
EA (1) EA009460B1 (ja)
EC (1) ECSP055973A (ja)
ES (1) ES2277237T3 (ja)
GE (1) GEP20074089B (ja)
HR (1) HRP20050681A2 (ja)
IS (1) IS2450B (ja)
MA (1) MA27712A1 (ja)
MX (1) MXPA05008923A (ja)
NO (1) NO20054053L (ja)
OA (1) OA13029A (ja)
PL (1) PL378747A1 (ja)
PT (1) PT1597260E (ja)
RS (1) RS20050638A (ja)
SI (1) SI1597260T1 (ja)
TN (1) TNSN05200A1 (ja)

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Publication number Priority date Publication date Assignee Title
TW200904403A (en) * 2007-04-25 2009-02-01 Daiichi Sankyo Co Ltd Tricyclic aryl compounds
CN102812011A (zh) * 2009-11-16 2012-12-05 梅利科技公司 [1,5]-二氮杂环辛间四烯衍生物
US8420633B2 (en) * 2010-03-31 2013-04-16 Hoffmann-La Roche Inc. Aryl-cyclohexyl-tetraazabenzo[e]azulenes
US8461151B2 (en) * 2010-04-13 2013-06-11 Hoffmann-La Roche Inc. Aryl-/heteroaryl-cyclohexenyl-tetraazabenzo[e]azulenes
US8492376B2 (en) * 2010-04-21 2013-07-23 Hoffmann-La Roche Inc. Heteroaryl-cyclohexyl-tetraazabenzo[e]azulenes
US8481528B2 (en) * 2010-04-26 2013-07-09 Hoffmann-La Roche Inc. Heterobiaryl-cyclohexyl-tetraazabenzo[e]azulenes
US9006450B2 (en) 2010-07-01 2015-04-14 Boehringer Ingelheim International Gmbh Compounds, pharmaceutical compositions and uses thereof
SI3077396T1 (sl) * 2013-12-05 2021-08-31 F. Hoffmann-La Roche Ag Sinteza trans-8-kloro-5-metil-1-(4-(piridin-2-iloksi)-cikloheksil)-5,6- dihidro-4H-2,3,5,10b-tetraaza-benzo(e)azulena in njegovih kristalnih oblik
HU231206B1 (hu) * 2017-12-15 2021-10-28 Richter Gedeon Nyrt. Triazolobenzazepinek

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GB8823475D0 (en) * 1988-10-06 1988-11-16 Merck Sharp & Dohme Chemical compounds
US5438035A (en) * 1994-06-24 1995-08-01 American Cyanamid Company Methods for controlling undesirable plant species with benzodiazepine compounds
US5753648A (en) * 1995-01-17 1998-05-19 American Cyanamid Company Tricyclic benzazepine vasopressin antagonists
DE69725182T2 (de) * 1996-11-01 2004-06-24 Wyeth 5H PYRROLO[2,1-c][1,4]BENZODIAZEPIN-3-CARBOXAMIDDERIVATE
TR200102069T2 (tr) * 1999-01-19 2001-11-21 Ortho-Mcneil Pharmaceutical, Inc. Vasopresin reseptörü antagonistleri olarak trisiklik benzodiazepinler.
US7109193B2 (en) * 2001-04-12 2006-09-19 Wyeth Tricyclic diazepines tocolytic oxytocin receptor antagonists
GB0224919D0 (en) * 2002-10-25 2002-12-04 Pfizer Ltd Triazole compounds useful in therapy

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ATE349449T1 (de) 2007-01-15
GEP20074089B (en) 2007-04-10
IS2450B (is) 2008-11-15
JP2007045838A (ja) 2007-02-22
TNSN05200A1 (fr) 2007-06-11
SI1597260T1 (sl) 2007-04-30
MXPA05008923A (es) 2006-03-09
EA200501136A1 (ru) 2006-06-30
EP1597260B1 (en) 2006-12-27
AU2004213242A1 (en) 2004-09-02
HRP20050681A2 (en) 2005-12-31
DK1597260T3 (da) 2007-04-02
MA27712A1 (fr) 2006-01-02
PT1597260E (pt) 2007-01-31
IS7957A (is) 2005-07-25
JP4033886B2 (ja) 2008-01-16
CA2516557A1 (en) 2004-09-02
AU2004213242B2 (en) 2007-04-19
NO20054053D0 (no) 2005-08-31
EP1597260A1 (en) 2005-11-23
OA13029A (en) 2006-11-10
PL378747A1 (pl) 2006-05-15
DE602004003914D1 (de) 2007-02-08
KR20050106443A (ko) 2005-11-09
EA009460B1 (ru) 2007-12-28
RS20050638A (en) 2007-12-31
BRPI0407676A (pt) 2006-03-01
KR100750028B1 (ko) 2007-08-16
ECSP055973A (es) 2006-01-16
NO20054053L (no) 2005-10-31
ES2277237T3 (es) 2007-07-01
DE602004003914T2 (de) 2007-05-31
JP2006517921A (ja) 2006-08-03
CA2516557C (en) 2008-11-18

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