ECSP099461A - Compuesto heteromonocíclico y uso del mismo - Google Patents

Compuesto heteromonocíclico y uso del mismo

Info

Publication number
ECSP099461A
ECSP099461A EC2009009461A ECSP099461A ECSP099461A EC SP099461 A ECSP099461 A EC SP099461A EC 2009009461 A EC2009009461 A EC 2009009461A EC SP099461 A ECSP099461 A EC SP099461A EC SP099461 A ECSP099461 A EC SP099461A
Authority
EC
Ecuador
Prior art keywords
formula
compound
same
group
diseases
Prior art date
Application number
EC2009009461A
Other languages
English (en)
Spanish (es)
Inventor
Takanobu Kuroita
Hiroki Sakamoto
Hideyuki Igawa
Minoru Sasaki
Kouhei Asano
Tsuyoshi Maekawa
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of ECSP099461A publication Critical patent/ECSP099461A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
EC2009009461A 2006-11-24 2009-06-23 Compuesto heteromonocíclico y uso del mismo ECSP099461A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006317839 2006-11-24
JP2007232106 2007-09-06

Publications (1)

Publication Number Publication Date
ECSP099461A true ECSP099461A (es) 2009-11-30

Family

ID=39205144

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2009009461A ECSP099461A (es) 2006-11-24 2009-06-23 Compuesto heteromonocíclico y uso del mismo

Country Status (21)

Country Link
US (2) US20100056526A1 (fr)
EP (2) EP2256115A1 (fr)
JP (1) JP2010510962A (fr)
KR (1) KR20090085117A (fr)
AR (1) AR063912A1 (fr)
AU (1) AU2007322608A1 (fr)
BR (1) BRPI0719060A2 (fr)
CA (1) CA2670404A1 (fr)
CL (1) CL2007003352A1 (fr)
CO (1) CO6231035A2 (fr)
CR (1) CR10847A (fr)
EA (1) EA200970510A1 (fr)
EC (1) ECSP099461A (fr)
IL (1) IL198819A0 (fr)
MA (1) MA30985B1 (fr)
MX (1) MX2009005449A (fr)
NO (1) NO20092415L (fr)
PE (1) PE20081228A1 (fr)
TN (1) TN2009000199A1 (fr)
TW (1) TW200829581A (fr)
WO (1) WO2008062905A2 (fr)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7103906B1 (en) 2000-09-29 2006-09-05 International Business Machines Corporation User controlled multi-device media-on-demand system
MX336193B (es) 2000-10-11 2016-01-11 Rovi Guides Inc Sistemas y metodos para proporcionar almacenamiento de datos en servidores, mediante un sistema de entrega de medios a peticion.
US8086575B2 (en) 2004-09-23 2011-12-27 Rovi Solutions Corporation Methods and apparatus for integrating disparate media formats in a networked media system
US9681105B2 (en) 2005-12-29 2017-06-13 Rovi Guides, Inc. Interactive media guidance system having multiple devices
US8607287B2 (en) 2005-12-29 2013-12-10 United Video Properties, Inc. Interactive media guidance system having multiple devices
US7803940B2 (en) 2006-11-24 2010-09-28 Takeda Pharmaceutical Company Limited Heteromonocyclic compound or a salt thereof having strong antihypertensive action, insulin sensitizing activity and the like production thereof and use thereof for prophylaxis or treatment of cardiovascular diseases, metabolic diseases and/or central nervous system diseases
KR20090085117A (ko) * 2006-11-24 2009-08-06 다케다 야쿠힌 고교 가부시키가이샤 헤테로모노시클릭 화합물 및 이의 용도
US20090019492A1 (en) 2007-07-11 2009-01-15 United Video Properties, Inc. Systems and methods for mirroring and transcoding media content
ES2433225T3 (es) * 2009-01-30 2013-12-10 Takeda Pharmaceutical Company Limited Compuesto con anillos condensados y uso del mismo
JPWO2010095462A1 (ja) 2009-02-23 2012-08-23 興和株式会社 新規な3−(5−アルコキシピリミジン−2−イル)ピリミジン−4(3h)−オン構造を有する化合物及びこれを含有する医薬
US8664226B2 (en) 2009-04-17 2014-03-04 Kowa Company, Ltd. Compound having 3-heteroarylpyrimidin-4-(3H)-one structure and pharmaceutical preparation containing same
EP2436675A1 (fr) 2009-05-29 2012-04-04 Kowa Company, Ltd. Nouveau dérivé d'acide -phénoxybenzèneacétique et préparation pharmaceutique le contenant
JPWO2011024468A1 (ja) 2009-08-27 2013-01-24 興和株式会社 新規なスルホンアミド誘導体及びこれを含有する医薬
US9014546B2 (en) 2009-09-23 2015-04-21 Rovi Guides, Inc. Systems and methods for automatically detecting users within detection regions of media devices
TWI500611B (zh) * 2009-09-29 2015-09-21 Kowa Co 新穎苯基吡啶衍生物及含有該衍生物之醫藥
WO2011077711A1 (fr) * 2009-12-22 2011-06-30 興和株式会社 Nouveau dérivé de 2-pyridone et produit pharmaceutique le contenant
JPWO2011105099A1 (ja) * 2010-02-25 2013-06-20 興和株式会社 新規な4−アルコキシピリミジン構造を有する化合物及びこれを含有する医薬
WO2011142381A1 (fr) * 2010-05-11 2011-11-17 Fujita Takashi Dérivé benzo- ou pyrido-imidazole
WO2012011592A1 (fr) * 2010-07-23 2012-01-26 武田薬品工業株式会社 Composé hétérocyclique et application de celui-ci
UY33650A (es) 2010-10-07 2012-04-30 Takeda Pharmaceutical Compuestos heterocíclicos
WO2012078674A1 (fr) 2010-12-06 2012-06-14 Confluence Life Sciences, Inc. Composés indole/indazole-pyrimidinyle substitués
WO2012078673A1 (fr) 2010-12-06 2012-06-14 Confluence Life Sciences, Inc. Composés urée-pyridine substitués
US9359300B2 (en) 2010-12-06 2016-06-07 Confluence Life Sciences, Inc. Methyl/difluorophenyl-methoxy substituted pyridinone-pyridinyl compounds, methyl-pyridinyl-methoxy substituted pyridinone-pyridinyl compounds, and methyl-pyrimidinyl-methoxy substituted pyridinone-pyridinyl compounds
EP2648516B1 (fr) 2010-12-06 2018-09-05 Aclaris Therapeutics, Inc. Composés pyridinone-pyridinyle substitués
PL2687523T3 (pl) * 2011-03-14 2016-06-30 Kowa Co Nowa pochodna fenylopirydyny i lek zawierający ją
EP2567959B1 (fr) 2011-09-12 2014-04-16 Sanofi Dérivés d'amide d'acide 6-(4-hydroxy-phényl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique en tant qu'inhibiteurs de kinase
WO2013086208A1 (fr) 2011-12-06 2013-06-13 Confluence Life Sciences, Inc. Composés de pyrimidinone-phényl-pyrimidinyle substitués
KR102011534B1 (ko) * 2011-12-21 2019-08-16 오노 야꾸힝 고교 가부시키가이샤 인자 XIa 억제제로서 피리디논 및 피리미디논 유도체
JO3470B1 (ar) 2012-10-08 2020-07-05 Merck Sharp & Dohme مشتقات 5- فينوكسي-3h-بيريميدين-4-أون واستخدامها كمثبطات ناسخ عكسي ل hiv
ES2869048T3 (es) 2013-06-07 2021-10-22 Aclaris Therapeutics Inc Compuestos de piridinona-piridinilo sustituidos con metil/fluoro-piridinil-metoxi y compuestos de piridinona-piridinilo sustituidos con fluoro-pirimidinil-metoxi
CN105473558B (zh) 2013-06-20 2019-04-19 拜耳作物科学股份公司 作为杀螨剂和杀昆虫剂的芳基硫化物衍生物和芳基硫氧化物衍生物
BR112015031155A2 (pt) 2013-06-20 2017-07-25 Bayer Cropscience Ag derivados de sulfureto de arila e derivados de aril sulfóxido como acaricidas e inseticidas
US9674563B2 (en) 2013-11-04 2017-06-06 Rovi Guides, Inc. Systems and methods for recommending content
RU2694254C1 (ru) 2013-12-19 2019-07-11 Саншайн Лейк Фарма Ко., Лтд. Азотсодержащие гетероциклические производные и их применение в лекарственных препаратах
EP3785714A1 (fr) 2014-04-01 2021-03-03 Merck Sharp & Dohme Corp. Promédicaments d'inhibiteurs de la transcriptase inverse du vih
PT3231803T (pt) 2014-12-10 2020-09-03 Ono Pharmaceutical Co Derivado de di-hidroindolizinona
US20190297887A1 (en) 2016-07-12 2019-10-03 Bayer Cropscience Aktiengesellschaft Bicyclic compounds as pesticides
KR101984121B1 (ko) * 2017-08-21 2019-05-30 보령제약 주식회사 피리미디논 유도체 화합물 및 이의 용도
CN115666566A (zh) 2020-03-27 2023-01-31 阿克拉瑞斯治疗股份有限公司 用于免疫病况的治疗的mk2途径抑制剂的口服组合物
US11116737B1 (en) 2020-04-10 2021-09-14 University Of Georgia Research Foundation, Inc. Methods of using probenecid for treatment of coronavirus infections

Family Cites Families (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5411980A (en) * 1989-07-28 1995-05-02 Merck & Co., Inc. Substituted triazolinones, triazolinethiones, and triazolinimines as angiotensin II antagonists
DE69013607T2 (de) 1989-08-02 1995-03-02 Takeda Chemical Industries Ltd Pyrazol-Derivate, Verfahren zu deren Herstellung und Anwendung.
JPH03218371A (ja) 1989-08-02 1991-09-25 Takeda Chem Ind Ltd ピラゾール誘導体
JP3032844B2 (ja) 1990-02-15 2000-04-17 武田薬品工業株式会社 ピリミジンジオン誘導体
DE69129998T2 (de) 1990-02-15 1998-12-24 Takeda Chemical Industries Ltd Pyrimidindionderivate, deren Herstellung und Verwendung
JP3114073B2 (ja) 1990-03-07 2000-12-04 武田薬品工業株式会社 アンジオテンシンii拮抗薬−含窒素異項環化合物
CA2037630C (fr) * 1990-03-07 2001-07-03 Akira Morimoto Composes heterocycliques renfermant de l'azote, methode de production et applications correspondantes
US5166206A (en) * 1990-03-30 1992-11-24 Merck & Co., Inc. Substituted pyrimidines, pyrimidinones and pyridopyrimidines
US5472967A (en) * 1991-02-20 1995-12-05 Synthelabo 4-pyrimidinone derivatives their preparation and their application in therapy
IL102183A (en) 1991-06-27 1999-11-30 Takeda Chemical Industries Ltd The heterocyclic compounds are converted into biphenyl groups, their production and the pharmaceutical compositions containing them
IT1250749B (it) * 1991-08-02 1995-04-21 Luso Farmaco Inst Composti eterociclici ad attivita' a ii antagonista
EP0829479B1 (fr) 1992-09-14 2004-04-14 Takeda Chemical Industries, Ltd. Composés hétérocycliques et leur utilisation comme antagonistes d'angiotensine II
JPH06239859A (ja) 1992-09-14 1994-08-30 Takeda Chem Ind Ltd アンギオテンシンii拮抗作用を有する環状化合物およびその用途
ATE204276T1 (de) 1992-12-22 2001-09-15 Takeda Chemical Industries Ltd Heterocyclische verbindungen mit angiotensin-ii- antagonistischer wirkung und ihre anwendung
JP3412887B2 (ja) 1992-12-22 2003-06-03 武田薬品工業株式会社 アンギオテンシンii拮抗作用を有する複素環化合物およびその用途
US20010020100A1 (en) * 1994-06-14 2001-09-06 G.D. Searle & Co. N-substituted-1, 2, 4-triazolone compounds for treatment of cardiovascular disorders
US6025372A (en) 1997-04-04 2000-02-15 Merck & Co., Inc. Somatostatin agonists
US6057338A (en) 1997-04-04 2000-05-02 Merck & Co., Inc. Somatostatin agonists
AU1285499A (en) 1997-10-30 1999-05-24 Merck & Co., Inc. Somatostatin agonists
AR035016A1 (es) 1999-08-25 2004-04-14 Takeda Chemical Industries Ltd Composicion de azol promotor de produccion/secrecion de neurotrofina, compuesto prodroga del mismo, composicion farmaceutica que lo comprende y uso del mismo para preparar esta ultima.
EP1227090A4 (fr) 1999-10-07 2002-11-20 Tadeka Chemical Ind Ltd Derives d'amines
ES2225252T3 (es) 1999-11-10 2005-03-16 Takeda Chemical Industries, Ltd. Compuestos n-heterociclicos de 5 miembros con actividad hipoglucemica e hipolipidemica.
CA2407149C (fr) 2000-04-28 2010-10-12 Takeda Chemical Industries, Ltd. Antagonistes de l'hormone concentrant la melanine
US7229986B2 (en) 2000-05-16 2007-06-12 Takeda Pharmaceutical Company Ltd. Melanin-concentrating hormone antagonist
US6974806B2 (en) 2000-07-13 2005-12-13 Takeda Pharmaceutical Company Limited Lipid-rich plaque inhibitors
WO2003042204A1 (fr) 2001-10-19 2003-05-22 Takeda Chemical Industries, Ltd. Derive d'amine
PL371319A1 (en) 2002-01-11 2005-06-13 Takeda Pharmaceutical Company Limited Coumarin derivatives, process for their production and use thereof
WO2004048363A1 (fr) 2002-11-22 2004-06-10 Takeda Pharmaceutical Company Limited Derives d'imidazole, leur procede de production et d'utilisation
KR20090085117A (ko) * 2006-11-24 2009-08-06 다케다 야쿠힌 고교 가부시키가이샤 헤테로모노시클릭 화합물 및 이의 용도
US7803940B2 (en) * 2006-11-24 2010-09-28 Takeda Pharmaceutical Company Limited Heteromonocyclic compound or a salt thereof having strong antihypertensive action, insulin sensitizing activity and the like production thereof and use thereof for prophylaxis or treatment of cardiovascular diseases, metabolic diseases and/or central nervous system diseases

Also Published As

Publication number Publication date
MX2009005449A (es) 2009-06-02
NO20092415L (no) 2009-08-17
CO6231035A2 (es) 2010-12-20
PE20081228A1 (es) 2008-10-29
WO2008062905A3 (fr) 2008-12-04
EP2256115A1 (fr) 2010-12-01
AU2007322608A1 (en) 2008-05-29
US20100056526A1 (en) 2010-03-04
JP2010510962A (ja) 2010-04-08
EP2074117A2 (fr) 2009-07-01
CR10847A (es) 2009-07-13
AU2007322608A2 (en) 2009-07-16
KR20090085117A (ko) 2009-08-06
MA30985B1 (fr) 2009-12-01
WO2008062905A2 (fr) 2008-05-29
US20080207654A1 (en) 2008-08-28
TN2009000199A1 (en) 2010-10-18
CA2670404A1 (fr) 2008-05-29
CL2007003352A1 (es) 2008-07-04
TW200829581A (en) 2008-07-16
BRPI0719060A2 (pt) 2014-02-04
EA200970510A1 (ru) 2009-12-30
IL198819A0 (en) 2010-02-17
AR063912A1 (es) 2009-02-25

Similar Documents

Publication Publication Date Title
ECSP099461A (es) Compuesto heteromonocíclico y uso del mismo
AR071531A1 (es) Compuesto cristalino heteromonociclico
AR079327A1 (es) Derivados de 2-amino-5,5-difluor -5,6-dihidro-4h-(1,3) oxazin-4-il) fenil)-amida
AR085960A1 (es) 1,3-oxazinas como inhibidores de la bace1 y/o de la bace2
PE20201165A1 (es) Analogos de piridazina 1,4-disustituida y metodos para el tratamiento de condiciones relacionadas con la deficiencia de smn
AR053120A1 (es) Aminopiridinas como inhibidores de beta secretasa
CO6382126A2 (es) Compuestos heteroaromaticos fusionados y espirociclicos para el tratamiento de infecciones bacterianas
AR077935A1 (es) Derivados de 3-amino-5 fenil-5,6-dihidro-2h-(1,4)oxazina
CO5590957A2 (es) Amino-1,3,5-triazinas sustituidas en n con radicales biciclicos quirales, procedimiento para su preparacion, composiciones de las mismas y su uso como herbicidas y reguladores del crecimiento de las plantas
PE20171341A1 (es) Compuestos de pirazina para el tratamiento de enfermedades infecciosas
AR049388A1 (es) Heterociclos como inhibidores de aldosterona sintasa
AR061923A1 (es) Compuestos derivados de benzofuran-piperidina
CO2017001178A2 (es) Derivado de piridona que tiene un grupo tetrahidropiranil metilo
PE20160751A1 (es) Moduladores de tetrahidropiridopirazinas de gpr6
AR043434A1 (es) Derivados de piperizacina acilados como agonistas del receptor de melanocortina-4. composiciones farmaceuticas y usos
AR054560A1 (es) Espiropiperidina como inhibidores de beta-secretasa para el tratamiento de la enfermedad de alzheimer
AR058885A1 (es) Compuestos de piperidina 3,5-sustituidos
AR074608A1 (es) Derivados de 2-(piperidin-1-il)-4-heterociclil-tiazol-5-carboxilico para infecciones bacterianas
ES2530943T3 (es) Derivados de la cromenona con actividad antitumoral
PE20090648A1 (es) Compuestos para el tratamiento de la hepatitis c
ECSP11011318A (es) Derivados de benzofurano
AR059905A1 (es) Pirrolidina-3-ilaminas n-substituidas como antagonistas del receptor histamina-3, composicion farmaceutica y proceso para preparar el compuesto
PE20141553A1 (es) Compuestos de triazolopiridina como inhibidores de la ped10a
UY28333A1 (es) Inhibidores de caspasa y sus usos.
AR073043A1 (es) Compuestos de azetidinas polisustituidos, composiciones farmaceuticas que los contienen, metodo de preparacion y uso de los mismos en el tratamiento de enfermedades respiratorias, metabolicas y del sistema nervioso central, entre otras.