DE3505576A1 - Vorwirkstoffe entzuendungshemmender oxicame und solche vorwirkstoffe enthaltende pharmazeutische zusammensetzungen - Google Patents
Vorwirkstoffe entzuendungshemmender oxicame und solche vorwirkstoffe enthaltende pharmazeutische zusammensetzungenInfo
- Publication number
- DE3505576A1 DE3505576A1 DE19853505576 DE3505576A DE3505576A1 DE 3505576 A1 DE3505576 A1 DE 3505576A1 DE 19853505576 DE19853505576 DE 19853505576 DE 3505576 A DE3505576 A DE 3505576A DE 3505576 A1 DE3505576 A1 DE 3505576A1
- Authority
- DE
- Germany
- Prior art keywords
- methyl
- dioxide
- carboxamide
- benzothiazine
- pyridyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58268484A | 1984-02-23 | 1984-02-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
DE3505576A1 true DE3505576A1 (de) | 1985-09-05 |
Family
ID=24330094
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE19853505576 Ceased DE3505576A1 (de) | 1984-02-23 | 1985-02-18 | Vorwirkstoffe entzuendungshemmender oxicame und solche vorwirkstoffe enthaltende pharmazeutische zusammensetzungen |
Country Status (22)
Country | Link |
---|---|
JP (1) | JPS60184077A (fr) |
KR (1) | KR850006198A (fr) |
AU (1) | AU552478B2 (fr) |
BE (1) | BE901783A (fr) |
DD (1) | DD232045A5 (fr) |
DE (1) | DE3505576A1 (fr) |
DK (1) | DK81185A (fr) |
ES (1) | ES8606312A1 (fr) |
FI (1) | FI850742L (fr) |
FR (1) | FR2565980A1 (fr) |
GB (1) | GB2154585A (fr) |
GR (1) | GR850442B (fr) |
HU (1) | HUT37616A (fr) |
IL (1) | IL74407A0 (fr) |
IT (1) | IT1185514B (fr) |
LU (1) | LU85780A1 (fr) |
NL (1) | NL8500485A (fr) |
NO (1) | NO850725L (fr) |
PL (1) | PL252023A1 (fr) |
PT (1) | PT79988B (fr) |
SE (1) | SE8500889L (fr) |
ZA (1) | ZA851317B (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4623486A (en) * | 1985-05-29 | 1986-11-18 | Pfizer Inc. | [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity |
US4610982A (en) * | 1985-06-03 | 1986-09-09 | Pfizer Inc. | Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor |
US20090238763A1 (en) | 2006-07-09 | 2009-09-24 | Chongxi Yu | High penetration compositions and uses thereof |
US20090221703A1 (en) | 2006-07-09 | 2009-09-03 | Chongxi Yu | High penetration composition and uses thereof |
WO2008044095A1 (fr) * | 2006-10-11 | 2008-04-17 | Techfields Biochem Co. Ltd | Pro-médicaments d'oxicams solubles dans l'eau et chargés positivement et composés apparentés avec une vitesse de pénétration de la peau très élevée |
AU2007354632B2 (en) | 2007-06-04 | 2014-06-26 | Techfields Inc | Pro-drugs of NSAIAs with very high skin and membranes penetration rates and their new medicinal uses |
MX362949B (es) | 2008-12-04 | 2019-02-27 | Yu Chongxi | Composiciones de alta penetracion y sus aplicaciones. |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3704298A (en) * | 1971-06-22 | 1972-11-28 | Warner Lambert Co | 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides |
US4309427A (en) * | 1981-01-15 | 1982-01-05 | Pfizer Inc. | Benzothiazine dioxide derivatives |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3591574A (en) * | 1968-05-29 | 1971-07-06 | American Home Prod | Tri-n-phenylglycyl derivatives of insulin |
US3787324A (en) * | 1971-03-01 | 1974-01-22 | Warner Lambert Co | 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production |
AU518216B2 (en) * | 1977-09-06 | 1981-09-17 | Hafslund Nycomed Pharma Aktiengesellschaft | Thienothiazine derivatives |
JPS5714589A (en) * | 1980-06-27 | 1982-01-25 | Mitsui Toatsu Chem Inc | Benzothiazine derivative, its preparation and drug composition |
IT8219486A0 (it) * | 1982-02-05 | 1982-02-05 | Chiesi Farma Spa | Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche. |
IT1206525B (it) * | 1982-12-10 | 1989-04-27 | Zionale S R L A Roma | Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione |
-
1985
- 1985-01-23 JP JP60010722A patent/JPS60184077A/ja active Pending
- 1985-02-18 DE DE19853505576 patent/DE3505576A1/de not_active Ceased
- 1985-02-19 PL PL25202385A patent/PL252023A1/xx unknown
- 1985-02-20 PT PT79988A patent/PT79988B/pt unknown
- 1985-02-20 GR GR850442A patent/GR850442B/el unknown
- 1985-02-20 GB GB08504355A patent/GB2154585A/en not_active Withdrawn
- 1985-02-20 LU LU85780A patent/LU85780A1/fr unknown
- 1985-02-21 DD DD85273451A patent/DD232045A5/de unknown
- 1985-02-21 NL NL8500485A patent/NL8500485A/nl not_active Application Discontinuation
- 1985-02-21 ES ES540590A patent/ES8606312A1/es not_active Expired
- 1985-02-21 IL IL74407A patent/IL74407A0/xx unknown
- 1985-02-21 ZA ZA851317A patent/ZA851317B/xx unknown
- 1985-02-21 IT IT8519585A patent/IT1185514B/it active
- 1985-02-21 BE BE0/214544A patent/BE901783A/fr not_active IP Right Cessation
- 1985-02-22 NO NO850725A patent/NO850725L/no unknown
- 1985-02-22 KR KR1019850001106A patent/KR850006198A/ko not_active Application Discontinuation
- 1985-02-22 FR FR8502586A patent/FR2565980A1/fr active Pending
- 1985-02-22 AU AU39066/85A patent/AU552478B2/en not_active Ceased
- 1985-02-22 FI FI850742A patent/FI850742L/fi not_active Application Discontinuation
- 1985-02-22 DK DK81185A patent/DK81185A/da not_active Application Discontinuation
- 1985-02-22 SE SE8500889A patent/SE8500889L/xx not_active Application Discontinuation
- 1985-02-22 HU HU85678A patent/HUT37616A/hu unknown
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3704298A (en) * | 1971-06-22 | 1972-11-28 | Warner Lambert Co | 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides |
US4309427A (en) * | 1981-01-15 | 1982-01-05 | Pfizer Inc. | Benzothiazine dioxide derivatives |
Non-Patent Citations (2)
Title |
---|
Derwent-Referat CPJ 48714 E/24-B02 der JP 82-70 888 * |
J. Med. Chem. 25, 1982, 12-18 * |
Also Published As
Publication number | Publication date |
---|---|
SE8500889D0 (sv) | 1985-02-22 |
IT1185514B (it) | 1987-11-12 |
FI850742A0 (fi) | 1985-02-22 |
DK81185D0 (da) | 1985-02-22 |
GB8504355D0 (en) | 1985-03-20 |
BE901783A (fr) | 1985-08-21 |
FI850742L (fi) | 1985-08-24 |
DD232045A5 (de) | 1986-01-15 |
ZA851317B (en) | 1986-10-29 |
ES540590A0 (es) | 1986-04-16 |
AU552478B2 (en) | 1986-06-05 |
ES8606312A1 (es) | 1986-04-16 |
PL252023A1 (en) | 1985-11-05 |
LU85780A1 (fr) | 1985-12-11 |
NO850725L (no) | 1985-08-26 |
PT79988B (en) | 1987-02-02 |
KR850006198A (ko) | 1985-10-02 |
AU3906685A (en) | 1985-09-05 |
GR850442B (fr) | 1985-06-19 |
SE8500889L (sv) | 1985-08-24 |
NL8500485A (nl) | 1985-09-16 |
DK81185A (da) | 1985-09-10 |
IT8519585A0 (it) | 1985-02-21 |
HUT37616A (en) | 1986-01-23 |
JPS60184077A (ja) | 1985-09-19 |
FR2565980A1 (fr) | 1985-12-20 |
PT79988A (en) | 1985-03-01 |
GB2154585A (en) | 1985-09-11 |
IL74407A0 (en) | 1985-05-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
OP8 | Request for examination as to paragraph 44 patent law | ||
8131 | Rejection |