SE8500889D0 - Prodrugs of antiinflammatory oxicams - Google Patents

Prodrugs of antiinflammatory oxicams

Info

Publication number
SE8500889D0
SE8500889D0 SE8500889A SE8500889A SE8500889D0 SE 8500889 D0 SE8500889 D0 SE 8500889D0 SE 8500889 A SE8500889 A SE 8500889A SE 8500889 A SE8500889 A SE 8500889A SE 8500889 D0 SE8500889 D0 SE 8500889D0
Authority
SE
Sweden
Prior art keywords
antiinflammatory
oxicams
prodrugs
toluoyl
benzoyl
Prior art date
Application number
SE8500889A
Other languages
English (en)
Other versions
SE8500889L (sv
Inventor
J G Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SE8500889D0 publication Critical patent/SE8500889D0/sv
Publication of SE8500889L publication Critical patent/SE8500889L/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
SE8500889A 1984-02-23 1985-02-22 Antiinflammatoriska oxicanforlekemedel SE8500889L (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23

Publications (2)

Publication Number Publication Date
SE8500889D0 true SE8500889D0 (sv) 1985-02-22
SE8500889L SE8500889L (sv) 1985-08-24

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8500889A SE8500889L (sv) 1984-02-23 1985-02-22 Antiinflammatoriska oxicanforlekemedel

Country Status (22)

Country Link
JP (1) JPS60184077A (sv)
KR (1) KR850006198A (sv)
AU (1) AU552478B2 (sv)
BE (1) BE901783A (sv)
DD (1) DD232045A5 (sv)
DE (1) DE3505576A1 (sv)
DK (1) DK81185A (sv)
ES (1) ES8606312A1 (sv)
FI (1) FI850742L (sv)
FR (1) FR2565980A1 (sv)
GB (1) GB2154585A (sv)
GR (1) GR850442B (sv)
HU (1) HUT37616A (sv)
IL (1) IL74407A0 (sv)
IT (1) IT1185514B (sv)
LU (1) LU85780A1 (sv)
NL (1) NL8500485A (sv)
NO (1) NO850725L (sv)
PL (1) PL252023A1 (sv)
PT (1) PT79988B (sv)
SE (1) SE8500889L (sv)
ZA (1) ZA851317B (sv)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
WO2008044095A1 (en) * 2006-10-11 2008-04-17 Techfields Biochem Co. Ltd Positively charged water-soluble prodrugs of oxicams and related compounds with very high skin penetration rate
AU2007354632B2 (en) 2007-06-04 2014-06-26 Techfields Inc Pro-drugs of NSAIAs with very high skin and membranes penetration rates and their new medicinal uses
MX362949B (es) 2008-12-04 2019-02-27 Yu Chongxi Composiciones de alta penetracion y sus aplicaciones.

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (it) * 1982-02-05 1982-02-05 Chiesi Farma Spa Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.
IT1206525B (it) * 1982-12-10 1989-04-27 Zionale S R L A Roma Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione

Also Published As

Publication number Publication date
IT1185514B (it) 1987-11-12
FI850742A0 (fi) 1985-02-22
DK81185D0 (da) 1985-02-22
GB8504355D0 (en) 1985-03-20
BE901783A (fr) 1985-08-21
FI850742L (fi) 1985-08-24
DD232045A5 (de) 1986-01-15
ZA851317B (en) 1986-10-29
ES540590A0 (es) 1986-04-16
AU552478B2 (en) 1986-06-05
ES8606312A1 (es) 1986-04-16
PL252023A1 (en) 1985-11-05
LU85780A1 (fr) 1985-12-11
NO850725L (no) 1985-08-26
PT79988B (en) 1987-02-02
KR850006198A (ko) 1985-10-02
AU3906685A (en) 1985-09-05
GR850442B (sv) 1985-06-19
SE8500889L (sv) 1985-08-24
DE3505576A1 (de) 1985-09-05
NL8500485A (nl) 1985-09-16
DK81185A (da) 1985-09-10
IT8519585A0 (it) 1985-02-21
HUT37616A (en) 1986-01-23
JPS60184077A (ja) 1985-09-19
FR2565980A1 (fr) 1985-12-20
PT79988A (en) 1985-03-01
GB2154585A (en) 1985-09-11
IL74407A0 (en) 1985-05-31

Similar Documents

Publication Publication Date Title
FI932104A0 (fi) Nya 4-arylpiperaziner och 4-arylpiperidiner
DK324286D0 (da) 1-substituerede oxindol-3-carboxamider og deres anvendelse som antiinflammatoriske og analgetiske midler
DE3881073T2 (de) Naphthalenverbindungen und antiallergische und antiinflammatorische pharmazeutische mittel.
SE8500889D0 (sv) Prodrugs of antiinflammatory oxicams
FI822203L (fi) Nya 2-aryl-3,4-diaza-bicyklo/4,n,0/-alken-(2)-oner-(5), foerfarande foer deras framstaellning och dessa innehaollande laekemedel
FI852806L (fi) 2-substituerade -1,3-propylidendifosfonatderivat och deras framstaellning.
SE8207302D0 (sv) Nya 2-pyrrolidonforeningar och forfarande for framstellning av desamma
ATE49120T1 (de) Entzuendungshemmende zusammensetzung.
AU574204B2 (en) 5-amino-1-phenylpyrazole derivatives
DE3362735D1 (de) 3-(1h-tetrazol-5-yl)-4(3h)-quinazolinones
GB2005247A (en) Perhydro naphthalene derivatives
AR245439A1 (es) Preparacion de acidos (2-cloro, bromo o nitro)-4-(alquil sulfonil) benzoico e intermediarios.
FR2348206A1 (fr) 2-cyclopropane carboxamido-5-halothiazoles et leur emploi en tant qu'agents anti-inflammatoires
DK0740657T3 (da) 4-Arylisoindoler med analgetisk virkning
ES2053686T3 (es) Nuevos di(met)acrilatos, procedimiento para su fabricacion y su empleo.
ES460807A1 (es) Procedimiento para la produccion de compuestos de isoindoli-nona.
SE8402361L (sv) Nya acylaminofenolderivat
SE8700566D0 (sv) Tetracyclic quinazolinones
ES8404358A1 (es) Un procedimiento para obtener derivados de isoxazolopirimidina.
FI880384A (fi) Nya imidazo- och triazolotiadiaziner, foerfarande foer deras framstaellning, dessa innehaollande laekemedel och deras anvaendning, samt naogra vid framstaellningen av naemnda foereningar bildade mellanprodukter.
FI873483A (fi) Oxiranpseudooligosackarider, foerfarande foer deras framstaellning, deras anvaendning och farmaceutiska preparat.
FR2361364A1 (fr) Nouveaux derives d'azetidine
FI934252A (fi) 1,5,6,7-tetrahydro-4H-indazol-4-oner innehaollande laekemedel, nya 1,5,6,7-tetrahydro-4H-indazol-4-oner och foerfarande foer deras framstaellning
IT1250751B (it) (3h,7h)selenazolo(3,4-a|piridine con attivita' antiasmatica ed antiinfiammatoria delle vie aereea
FI875626A (fi) Foerfarande foer framstaellning av dibenzo/be/ixepinaettiksyraderivat.

Legal Events

Date Code Title Description
NAV Patent application has lapsed

Ref document number: 8500889-4

Effective date: 19870123

Format of ref document f/p: F