NL8500485A - Voorlopers van antiinflammatoire oxicamen. - Google Patents

Voorlopers van antiinflammatoire oxicamen. Download PDF

Info

Publication number
NL8500485A
NL8500485A NL8500485A NL8500485A NL8500485A NL 8500485 A NL8500485 A NL 8500485A NL 8500485 A NL8500485 A NL 8500485A NL 8500485 A NL8500485 A NL 8500485A NL 8500485 A NL8500485 A NL 8500485A
Authority
NL
Netherlands
Prior art keywords
dioxide
methyl
benzothiazine
compound according
carboxamide
Prior art date
Application number
NL8500485A
Other languages
English (en)
Dutch (nl)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NL8500485A publication Critical patent/NL8500485A/nl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NL8500485A 1984-02-23 1985-02-21 Voorlopers van antiinflammatoire oxicamen. NL8500485A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23
US58268484 1984-02-23

Publications (1)

Publication Number Publication Date
NL8500485A true NL8500485A (nl) 1985-09-16

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8500485A NL8500485A (nl) 1984-02-23 1985-02-21 Voorlopers van antiinflammatoire oxicamen.

Country Status (22)

Country Link
JP (1) JPS60184077A (fr)
KR (1) KR850006198A (fr)
AU (1) AU552478B2 (fr)
BE (1) BE901783A (fr)
DD (1) DD232045A5 (fr)
DE (1) DE3505576A1 (fr)
DK (1) DK81185A (fr)
ES (1) ES8606312A1 (fr)
FI (1) FI850742L (fr)
FR (1) FR2565980A1 (fr)
GB (1) GB2154585A (fr)
GR (1) GR850442B (fr)
HU (1) HUT37616A (fr)
IL (1) IL74407A0 (fr)
IT (1) IT1185514B (fr)
LU (1) LU85780A1 (fr)
NL (1) NL8500485A (fr)
NO (1) NO850725L (fr)
PL (1) PL252023A1 (fr)
PT (1) PT79988B (fr)
SE (1) SE8500889L (fr)
ZA (1) ZA851317B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
WO2008044095A1 (fr) * 2006-10-11 2008-04-17 Techfields Biochem Co. Ltd Pro-médicaments d'oxicams solubles dans l'eau et chargés positivement et composés apparentés avec une vitesse de pénétration de la peau très élevée
AU2007354632B2 (en) 2007-06-04 2014-06-26 Techfields Inc Pro-drugs of NSAIAs with very high skin and membranes penetration rates and their new medicinal uses
MX362949B (es) 2008-12-04 2019-02-27 Yu Chongxi Composiciones de alta penetracion y sus aplicaciones.

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (it) * 1982-02-05 1982-02-05 Chiesi Farma Spa Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.
IT1206525B (it) * 1982-12-10 1989-04-27 Zionale S R L A Roma Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione

Also Published As

Publication number Publication date
SE8500889D0 (sv) 1985-02-22
IT1185514B (it) 1987-11-12
FI850742A0 (fi) 1985-02-22
DK81185D0 (da) 1985-02-22
GB8504355D0 (en) 1985-03-20
BE901783A (fr) 1985-08-21
FI850742L (fi) 1985-08-24
DD232045A5 (de) 1986-01-15
ZA851317B (en) 1986-10-29
ES540590A0 (es) 1986-04-16
AU552478B2 (en) 1986-06-05
ES8606312A1 (es) 1986-04-16
PL252023A1 (en) 1985-11-05
LU85780A1 (fr) 1985-12-11
NO850725L (no) 1985-08-26
PT79988B (en) 1987-02-02
KR850006198A (ko) 1985-10-02
AU3906685A (en) 1985-09-05
GR850442B (fr) 1985-06-19
SE8500889L (sv) 1985-08-24
DE3505576A1 (de) 1985-09-05
DK81185A (da) 1985-09-10
IT8519585A0 (it) 1985-02-21
HUT37616A (en) 1986-01-23
JPS60184077A (ja) 1985-09-19
FR2565980A1 (fr) 1985-12-20
PT79988A (en) 1985-03-01
GB2154585A (en) 1985-09-11
IL74407A0 (en) 1985-05-31

Similar Documents

Publication Publication Date Title
FI63587B (fi) Foerfarande foer framstaellning av anti-inflammatoriska halogenerade 4-hydroxi-2-alkyl-3-karbamoyl-2h-tieno-1,2-tiazin-1,1-dioxidderivat
US5707992A (en) Antiproliferative quinazolines
AU634553B2 (en) Heteroarylamino- and heteroaryloxy-pyridinamines and related compounds, a process for their preparation and their use as medicaments
JPS63135384A (ja) N9−シクロペンチル−置換アデニン誘導体及びその製造方法
US20220194942A1 (en) 3,6-METHANO-1H-PYRROLO[3,2-b]PYRIDINE AND 3,6-METHANO-1H-PYRROLO[3,2-c]PYRIDINE COMPOUNDS AND MEDICAMENTS USING SAME
FI59253B (fi) Foerfarande foer framstaellning av terapeutiskt anvaendbara 4-hydroxi-2h-tieno(2,3-e) och (3,4-e)-1,2-tiazin-3-karboxamid-1,1-dioxid-derivat
WO2023144450A1 (fr) Composés destinés à être utilisés dans le traitement du cancer et d'états inflammatoires
NZ215805A (en) Heterocyclic thioesters
PL192783B1 (pl) Nowe pochodne chromenu, sposób ich otrzymywania, kompozycja farmaceutyczna zawierająca te związki oraz ich zastosowanie
NL8500485A (nl) Voorlopers van antiinflammatoire oxicamen.
AU672675B2 (en) Thiazolopyrimidine derivatives
EP0303172A2 (fr) Oxyimino-céphalosporines
FI89267C (fi) Foerfarande foer framstaellning av terapeutiskt aktiva 4,5-dihydro-oxazoler
CA2091688A1 (fr) Composes naphtaleniques a substituant, a proprietes antiproliferatives
PT87660B (pt) Processo para a preparacao de derivados de labdano polioxigenados e de composicoes farmaceuticas que os contem
JP2008515777A (ja) 疾患治療用のヒストンデアセチラーゼ阻害剤としての新規スルホンアミド
EP0685466A1 (fr) Dérivés de 3-hétéroaliphatyle- et 3-(hétéro)-(aryle)-aliphatyle-2(1H)-quinolone
NZ231044A (en) 3-acyl-2-oxindole-1-carboxamide derivatives
NL193192C (nl) Oxicamderivaat, farmaceutisch preparaat dat het derivaat bevat en werkwijze voor het bereiden van oxicamderivaten.
EP0365194B1 (fr) Prodrogues de 3-aryl-2-oxindole-1-carboxamide antiinflammatoires
EP0207651A2 (fr) Dérivés de la 7-phénylpyrazolo-[1,5-a]-1,3,5-triazine à activité anti-inflammatoire
EP1555264A1 (fr) Hétérocycles à cinq chaínons comme inhibiteurs de la famille des SRC proteines kinases
US4767858A (en) Anti-arthritic pyrazolo-triazine derivatives
EP0284069B1 (fr) Composés ester d'acide benzopyranopyridineacétique et leurs applications pharmaceutiques
KR850001548B1 (ko) N-(3-메르캅토-2-알킬-1-옥소프로필)-2,3-디하이드로-1h-인돌-2-카복실산 유도체의 제조방법

Legal Events

Date Code Title Description
BV The patent application has lapsed