ZA95636B - Protease inhibitor conjugates - Google Patents
Protease inhibitor conjugatesInfo
- Publication number
- ZA95636B ZA95636B ZA95636A ZA95636A ZA95636B ZA 95636 B ZA95636 B ZA 95636B ZA 95636 A ZA95636 A ZA 95636A ZA 95636 A ZA95636 A ZA 95636A ZA 95636 B ZA95636 B ZA 95636B
- Authority
- ZA
- South Africa
- Prior art keywords
- protease inhibitor
- inhibitor conjugates
- conjugates
- protease
- inhibitor
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/08—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
- A61K51/088—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Epidemiology (AREA)
- Optics & Photonics (AREA)
- Pharmacology & Pharmacy (AREA)
- Physics & Mathematics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9401483A GB9401483D0 (en) | 1994-01-26 | 1994-01-26 | Organic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA95636B true ZA95636B (en) | 1996-07-26 |
Family
ID=10749357
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA95636A ZA95636B (en) | 1994-01-26 | 1995-01-26 | Protease inhibitor conjugates |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP0741747A1 (en) |
| JP (1) | JPH09509653A (en) |
| AU (1) | AU1576495A (en) |
| CA (1) | CA2179889A1 (en) |
| GB (1) | GB9401483D0 (en) |
| IL (1) | IL112423A0 (en) |
| PE (1) | PE45295A1 (en) |
| SG (1) | SG47079A1 (en) |
| WO (1) | WO1995020603A1 (en) |
| ZA (1) | ZA95636B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9515489D0 (en) * | 1995-07-28 | 1995-09-27 | Sandoz Ltd | Organic compounds |
| DE10046514A1 (en) | 2000-09-15 | 2002-04-25 | Diagnostikforschung Inst | Process for imaging and diagnosis of thrombi using magnetic resonance imaging using particulate contrast media |
| EP1466916B1 (en) | 2002-09-09 | 2007-10-24 | Trigen Limited | Peptide boronic acids useful in making salts thereof |
| US7576206B2 (en) | 2003-08-14 | 2009-08-18 | Cephalon, Inc. | Proteasome inhibitors and methods of using the same |
| US7223745B2 (en) | 2003-08-14 | 2007-05-29 | Cephalon, Inc. | Proteasome inhibitors and methods of using the same |
| US7468383B2 (en) | 2005-02-11 | 2008-12-23 | Cephalon, Inc. | Proteasome inhibitors and methods of using the same |
| AU2010341530B2 (en) | 2009-12-22 | 2016-03-10 | Cephalon, Inc. | Proteasome inhibitors and processes for their preparation, purification and use |
| CN114685453A (en) | 2016-06-21 | 2022-07-01 | 奥瑞恩眼科有限责任公司 | Heterocyclic prolinamide derivatives |
| JP7164521B2 (en) | 2016-06-21 | 2022-11-01 | オリオン・オフサルモロジー・エルエルシー | carbocyclic prolinamide derivatives |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4668503A (en) * | 1982-07-26 | 1987-05-26 | Trustees Of University Of Massachusetts | Process for labeling amines with 99m Tc |
| US5187157A (en) * | 1987-06-05 | 1993-02-16 | Du Pont Merck Pharmaceutical Company | Peptide boronic acid inhibitors of trypsin-like proteases |
| DE69023394T2 (en) * | 1989-06-16 | 1996-07-04 | Merck Frosst Canada Inc | Chelate derivatives of atrial-natriurethic factor (ANF). |
| GB9017694D0 (en) * | 1990-08-13 | 1990-09-26 | Sandoz Ltd | Improvements in or relating to organic chemistry |
| US5252721A (en) * | 1990-09-28 | 1993-10-12 | Neorx Corporation | S3 N chelating compounds |
| ATE186550T1 (en) * | 1991-04-22 | 1999-11-15 | Mallinckrodt Medical Inc | COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR DETECTING AND LOCALIZING TISSUES HAVING NEUROKININ-1 RECEPTORS |
-
1994
- 1994-01-26 GB GB9401483A patent/GB9401483D0/en active Pending
-
1995
- 1995-01-24 PE PE1995260194A patent/PE45295A1/en not_active Application Discontinuation
- 1995-01-24 IL IL11242395A patent/IL112423A0/en unknown
- 1995-01-25 WO PCT/EP1995/000269 patent/WO1995020603A1/en not_active Application Discontinuation
- 1995-01-25 AU AU15764/95A patent/AU1576495A/en not_active Abandoned
- 1995-01-25 SG SG1996005775A patent/SG47079A1/en unknown
- 1995-01-25 JP JP7519884A patent/JPH09509653A/en active Pending
- 1995-01-25 CA CA002179889A patent/CA2179889A1/en not_active Abandoned
- 1995-01-25 EP EP95907611A patent/EP0741747A1/en not_active Ceased
- 1995-01-26 ZA ZA95636A patent/ZA95636B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB9401483D0 (en) | 1994-03-23 |
| CA2179889A1 (en) | 1995-08-03 |
| PE45295A1 (en) | 1995-12-29 |
| IL112423A0 (en) | 1995-03-30 |
| JPH09509653A (en) | 1997-09-30 |
| WO1995020603A1 (en) | 1995-08-03 |
| AU1576495A (en) | 1995-08-15 |
| SG47079A1 (en) | 1998-03-20 |
| EP0741747A1 (en) | 1996-11-13 |
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