IL112423A0 - Inhibitors of serine proteases, their preparation and pharmaceutical compositions containing them - Google Patents
Inhibitors of serine proteases, their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL112423A0 IL112423A0 IL11242395A IL11242395A IL112423A0 IL 112423 A0 IL112423 A0 IL 112423A0 IL 11242395 A IL11242395 A IL 11242395A IL 11242395 A IL11242395 A IL 11242395A IL 112423 A0 IL112423 A0 IL 112423A0
- Authority
- IL
- Israel
- Prior art keywords
- inhibitors
- preparation
- pharmaceutical compositions
- compositions containing
- serine proteases
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/08—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
- A61K51/088—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Epidemiology (AREA)
- Optics & Photonics (AREA)
- Pharmacology & Pharmacy (AREA)
- Physics & Mathematics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Peptides Or Proteins (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9401483A GB9401483D0 (en) | 1994-01-26 | 1994-01-26 | Organic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL112423A0 true IL112423A0 (en) | 1995-03-30 |
Family
ID=10749357
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL11242395A IL112423A0 (en) | 1994-01-26 | 1995-01-24 | Inhibitors of serine proteases, their preparation and pharmaceutical compositions containing them |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP0741747A1 (en) |
| JP (1) | JPH09509653A (en) |
| AU (1) | AU1576495A (en) |
| CA (1) | CA2179889A1 (en) |
| GB (1) | GB9401483D0 (en) |
| IL (1) | IL112423A0 (en) |
| PE (1) | PE45295A1 (en) |
| SG (1) | SG47079A1 (en) |
| WO (1) | WO1995020603A1 (en) |
| ZA (1) | ZA95636B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9515489D0 (en) * | 1995-07-28 | 1995-09-27 | Sandoz Ltd | Organic compounds |
| DE10046514A1 (en) | 2000-09-15 | 2002-04-25 | Diagnostikforschung Inst | Process for imaging and diagnosis of thrombi using magnetic resonance imaging using particulate contrast media |
| MXPA05002661A (en) | 2002-09-09 | 2005-08-19 | Trigen Ltd | Boronic acid salts ant their use in the treatment of thrombosis. |
| US7223745B2 (en) | 2003-08-14 | 2007-05-29 | Cephalon, Inc. | Proteasome inhibitors and methods of using the same |
| US7576206B2 (en) | 2003-08-14 | 2009-08-18 | Cephalon, Inc. | Proteasome inhibitors and methods of using the same |
| US7468383B2 (en) | 2005-02-11 | 2008-12-23 | Cephalon, Inc. | Proteasome inhibitors and methods of using the same |
| EP2516449A1 (en) | 2009-12-22 | 2012-10-31 | Cephalon, Inc. | Proteasome inhibitors and processes for their preparation, purification and use |
| EP4257191A3 (en) | 2016-06-21 | 2023-11-22 | Orion Ophthalmology LLC | Heterocyclic prolinamide derivatives |
| JP7164521B2 (en) | 2016-06-21 | 2022-11-01 | オリオン・オフサルモロジー・エルエルシー | carbocyclic prolinamide derivatives |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4668503A (en) * | 1982-07-26 | 1987-05-26 | Trustees Of University Of Massachusetts | Process for labeling amines with 99m Tc |
| US5187157A (en) * | 1987-06-05 | 1993-02-16 | Du Pont Merck Pharmaceutical Company | Peptide boronic acid inhibitors of trypsin-like proteases |
| EP0403243B1 (en) * | 1989-06-16 | 1995-11-08 | Merck Frosst Canada Inc. | Chelate derivatives of atrial natriuretic factor (ANF) |
| GB9017694D0 (en) * | 1990-08-13 | 1990-09-26 | Sandoz Ltd | Improvements in or relating to organic chemistry |
| US5252721A (en) * | 1990-09-28 | 1993-10-12 | Neorx Corporation | S3 N chelating compounds |
| WO1992018536A2 (en) * | 1991-04-22 | 1992-10-29 | Mallinckrodt Medical, Inc. | Method for detecting an localizing tissues having neurokinine 1 receptors |
-
1994
- 1994-01-26 GB GB9401483A patent/GB9401483D0/en active Pending
-
1995
- 1995-01-24 IL IL11242395A patent/IL112423A0/en unknown
- 1995-01-24 PE PE1995260194A patent/PE45295A1/en not_active Application Discontinuation
- 1995-01-25 AU AU15764/95A patent/AU1576495A/en not_active Abandoned
- 1995-01-25 JP JP7519884A patent/JPH09509653A/en active Pending
- 1995-01-25 WO PCT/EP1995/000269 patent/WO1995020603A1/en not_active Application Discontinuation
- 1995-01-25 CA CA002179889A patent/CA2179889A1/en not_active Abandoned
- 1995-01-25 SG SG1996005775A patent/SG47079A1/en unknown
- 1995-01-25 EP EP95907611A patent/EP0741747A1/en not_active Ceased
- 1995-01-26 ZA ZA95636A patent/ZA95636B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO1995020603A1 (en) | 1995-08-03 |
| JPH09509653A (en) | 1997-09-30 |
| GB9401483D0 (en) | 1994-03-23 |
| EP0741747A1 (en) | 1996-11-13 |
| SG47079A1 (en) | 1998-03-20 |
| PE45295A1 (en) | 1995-12-29 |
| ZA95636B (en) | 1996-07-26 |
| CA2179889A1 (en) | 1995-08-03 |
| AU1576495A (en) | 1995-08-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL99163A0 (en) | Inhibitors for serine proteases,their preparation and pharmaceutical compositions containing them | |
| HUP9900964A3 (en) | Protease inhibitors and pharmaceutical compositions containing these compounds | |
| HUP9702035A3 (en) | Inhibitors of leukocita-adhesion- and vla-4-antagonists and pharmaceutical compositions containing them | |
| HUP9702036A3 (en) | Inhibitors of leucocita-adhesion and wla-4-antagonists and pharmaceutical compositions containing them | |
| HUP9702034A3 (en) | Inhibitors of leukocita-adhesion and vla-4-antagonists and pharmaceutical compositions containing them | |
| HUP0104768A3 (en) | 4-amino-3-oxo-azepanes as protease inhibitors and pharmaceutical compositions containing the same | |
| HUP0103806A3 (en) | Serine protease inhibitor and pharmaceutical compositions containing them | |
| IL109867A0 (en) | alpha-heteroaryloxymethyl ketones as interleukin -1beta protease inhibitors and pharmaceutical compositions containing them | |
| HUP0105077A3 (en) | Serine protease inhibitors and pharmaceutical compositions containing them | |
| HUP0100669A3 (en) | Peptide derivatives as serine protease inhibitors, their use and pharmaceutical compositions comprising thereof | |
| IL128664A (en) | Heterocyclic metalloprotease inhibitors and pharmaceutical compositions comprising them | |
| IL138028A0 (en) | Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical use | |
| HUP0201479A2 (en) | Novel macrocyclic compounds as metalloprotease inhibitors and pharmaceutical compositions containing them | |
| HUP0103283A3 (en) | Pyrazinone protease inhibitors, pharmaceutical compositions containing them and use of the compounds | |
| HU9700811D0 (en) | New inhibitors of metalloprotease, process for preparing them and pharmaceutical compositions containing them | |
| IL119466A0 (en) | Thrombin inhibitors their preparation and pharmaceutical compositions containing them | |
| HUP0100186A3 (en) | Compounds as lactam metalloprotease inhibitors and pharmaceutical compositions containing them | |
| IL120311A0 (en) | Serine protease inhibitors and pharmaceutical compositions containing them | |
| IL120310A0 (en) | Serine protease inhibitors and pharmaceutical compositions containing them | |
| HUP0002951A3 (en) | Bis-aminomethylcarbonyl compounds as protease inhibitors and pharmaceutical compositions containing them | |
| IL115771A (en) | Apolipoprotein-B synthesis inhibitors their preparation and pharmaceutical compositions containing them | |
| HUP9902256A3 (en) | Amidino protease inhibitors and pharmaceutical compositions containing them | |
| HUP0004644A3 (en) | Pyrrolopyrrolone derivatives as inhibitors of neutrophil elastase and pharmaceutical compositions containing them | |
| IL117247A (en) | Pharmaceutical compositions comprising protease inhibitors and quinoxalines | |
| IL112423A0 (en) | Inhibitors of serine proteases, their preparation and pharmaceutical compositions containing them |