ZA926677B - 13beta-o-methoxymethyl-22,23-dihydro avermectin b1a/b1b aglycone as a superior antiparasitic agent - Google Patents

13beta-o-methoxymethyl-22,23-dihydro avermectin b1a/b1b aglycone as a superior antiparasitic agent

Info

Publication number
ZA926677B
ZA926677B ZA926677A ZA926677A ZA926677B ZA 926677 B ZA926677 B ZA 926677B ZA 926677 A ZA926677 A ZA 926677A ZA 926677 A ZA926677 A ZA 926677A ZA 926677 B ZA926677 B ZA 926677B
Authority
ZA
South Africa
Prior art keywords
13beta
aglycone
methoxymethyl
superior
antiparasitic agent
Prior art date
Application number
ZA926677A
Other languages
English (en)
Inventor
Bruce O Linn
O Linn Bruce
Helmut Mrozik
Mrozik Helmut
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of ZA926677B publication Critical patent/ZA926677B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agronomy & Crop Science (AREA)
  • Biochemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
ZA926677A 1991-09-04 1992-09-03 13beta-o-methoxymethyl-22,23-dihydro avermectin b1a/b1b aglycone as a superior antiparasitic agent ZA926677B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75483891A 1991-09-04 1991-09-04

Publications (1)

Publication Number Publication Date
ZA926677B true ZA926677B (en) 1993-04-28

Family

ID=25036577

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA926677A ZA926677B (en) 1991-09-04 1992-09-03 13beta-o-methoxymethyl-22,23-dihydro avermectin b1a/b1b aglycone as a superior antiparasitic agent

Country Status (5)

Country Link
EP (1) EP0530901A1 (de)
JP (1) JPH05213958A (de)
AU (1) AU649876B2 (de)
CA (1) CA2077131A1 (de)
ZA (1) ZA926677B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US7919522B2 (en) 2007-05-03 2011-04-05 Merial Limited Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds
CN101679451A (zh) * 2007-05-03 2010-03-24 梅瑞尔有限公司 包含c-13烷氧基醚大环内酯类化合物和苯基吡唑类化合物的组合物
JP5740676B2 (ja) * 2013-10-17 2015-06-24 メリアル リミテッド Ｃ−１３アルコキシエーテルマクロライド化合物及びフェニルピラゾール化合物を含む組成物
CN115403644B (zh) * 2022-09-01 2024-04-05 石家庄学院 一种烟碱甲氨基或氨基阿维菌素B1a化合物及其制备方法和应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT39739A (en) * 1984-12-04 1986-10-29 Ciba Geigy Ag Process for production of derivatives of 13,3-milbemycin and medical preparatives containing thereof
US4587247A (en) * 1985-02-25 1986-05-06 Merck & Co., Inc. Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use

Also Published As

Publication number Publication date
AU649876B2 (en) 1994-06-02
CA2077131A1 (en) 1993-03-05
JPH05213958A (ja) 1993-08-24
EP0530901A1 (de) 1993-03-10
AU2214092A (en) 1993-03-11

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