AU649876B2 - 13 beta-O-methoxymethyl-22,23-dihydro avermectin B1a/B1b aglycone as a superior antiparasitic agents - Google Patents

13 beta-O-methoxymethyl-22,23-dihydro avermectin B1a/B1b aglycone as a superior antiparasitic agents Download PDF

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Publication number
AU649876B2
AU649876B2 AU22140/92A AU2214092A AU649876B2 AU 649876 B2 AU649876 B2 AU 649876B2 AU 22140/92 A AU22140/92 A AU 22140/92A AU 2214092 A AU2214092 A AU 2214092A AU 649876 B2 AU649876 B2 AU 649876B2
Authority
AU
Australia
Prior art keywords
compounds
avermectin
compound
methoxymethyl
aglycone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU22140/92A
Other languages
English (en)
Other versions
AU2214092A (en
Inventor
Bruce O. Linn
Helmut Mrozik
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of AU2214092A publication Critical patent/AU2214092A/en
Application granted granted Critical
Publication of AU649876B2 publication Critical patent/AU649876B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agronomy & Crop Science (AREA)
  • Biochemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AU22140/92A 1991-09-04 1992-09-03 13 beta-O-methoxymethyl-22,23-dihydro avermectin B1a/B1b aglycone as a superior antiparasitic agents Ceased AU649876B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75483891A 1991-09-04 1991-09-04
US754838 1991-09-04

Publications (2)

Publication Number Publication Date
AU2214092A AU2214092A (en) 1993-03-11
AU649876B2 true AU649876B2 (en) 1994-06-02

Family

ID=25036577

Family Applications (1)

Application Number Title Priority Date Filing Date
AU22140/92A Ceased AU649876B2 (en) 1991-09-04 1992-09-03 13 beta-O-methoxymethyl-22,23-dihydro avermectin B1a/B1b aglycone as a superior antiparasitic agents

Country Status (5)

Country Link
EP (1) EP0530901A1 (de)
JP (1) JPH05213958A (de)
AU (1) AU649876B2 (de)
CA (1) CA2077131A1 (de)
ZA (1) ZA926677B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US7919522B2 (en) 2007-05-03 2011-04-05 Merial Limited Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds
CN101679451A (zh) * 2007-05-03 2010-03-24 梅瑞尔有限公司 包含c-13烷氧基醚大环内酯类化合物和苯基吡唑类化合物的组合物
JP5740676B2 (ja) * 2013-10-17 2015-06-24 メリアル リミテッド Ｃ−１３アルコキシエーテルマクロライド化合物及びフェニルピラゾール化合物を含む組成物
CN115403644B (zh) * 2022-09-01 2024-04-05 石家庄学院 一种烟碱甲氨基或氨基阿维菌素B1a化合物及其制备方法和应用

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU5071985A (en) * 1984-12-04 1986-06-12 Sankyo Company Limited 13`` -milbemycin derivatives for controlling ecto-and endoparasites of plants and animals
AU5400486A (en) * 1985-02-25 1986-08-28 Merck & Co., Inc. 13-akoxymethoxy avermectin aglycone derivatives

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU5071985A (en) * 1984-12-04 1986-06-12 Sankyo Company Limited 13`` -milbemycin derivatives for controlling ecto-and endoparasites of plants and animals
AU5400486A (en) * 1985-02-25 1986-08-28 Merck & Co., Inc. 13-akoxymethoxy avermectin aglycone derivatives

Also Published As

Publication number Publication date
CA2077131A1 (en) 1993-03-05
JPH05213958A (ja) 1993-08-24
ZA926677B (en) 1993-04-28
EP0530901A1 (de) 1993-03-10
AU2214092A (en) 1993-03-11

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