ZA827063B - Pharmaceutical compositions having a peripheral antagonistic action with respect to opiates - Google Patents
Pharmaceutical compositions having a peripheral antagonistic action with respect to opiatesInfo
- Publication number
- ZA827063B ZA827063B ZA827063A ZA827063A ZA827063B ZA 827063 B ZA827063 B ZA 827063B ZA 827063 A ZA827063 A ZA 827063A ZA 827063 A ZA827063 A ZA 827063A ZA 827063 B ZA827063 B ZA 827063B
- Authority
- ZA
- South Africa
- Prior art keywords
- opiates
- respect
- antagonistic action
- pharmaceutical compositions
- peripheral antagonistic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/22—Bridged ring systems
- C07D221/28—Morphinans
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8119607A FR2514644A1 (fr) | 1981-10-19 | 1981-10-19 | Composition pharmaceutique a action antagoniste peripherique des opiaces |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA827063B true ZA827063B (en) | 1983-07-27 |
Family
ID=9263165
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA827063A ZA827063B (en) | 1981-10-19 | 1982-09-27 | Pharmaceutical compositions having a peripheral antagonistic action with respect to opiates |
Country Status (10)
Country | Link |
---|---|
US (1) | US4489079A (xx) |
EP (1) | EP0077723B1 (xx) |
JP (1) | JPS5874608A (xx) |
AT (1) | ATE17942T1 (xx) |
AU (1) | AU559451B2 (xx) |
DE (1) | DE3269082D1 (xx) |
FR (1) | FR2514644A1 (xx) |
IL (1) | IL66853A (xx) |
NZ (1) | NZ202210A (xx) |
ZA (1) | ZA827063B (xx) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2547820B1 (fr) * | 1983-06-24 | 1986-04-18 | Midy Spa | Antagonistes peripheriques des opiaces |
US5624958A (en) * | 1987-12-31 | 1997-04-29 | Isaacs; Charles E. | Disinfecting contact lenses |
US5552406A (en) * | 1994-06-17 | 1996-09-03 | The Mclean Hospital Corporation | Method for treating pain and brain perfusion abnormalities using mixed opioid agonist-antagonists |
DE19752080A1 (de) * | 1997-11-25 | 1999-07-29 | Karlsruhe Forschzent | Verfahren zur Herstellung eines mehrkomponentigen, oxidischen Keramikpulvers |
NZ518684A (en) * | 1999-11-29 | 2003-11-28 | Adolor Corp | Use of a peripheral mu opioid antagonist to treat or prevent ileus |
US6469030B2 (en) * | 1999-11-29 | 2002-10-22 | Adolor Corporation | Methods for the treatment and prevention of ileus |
ES2569262T3 (es) * | 2001-10-18 | 2016-05-09 | Nektar Therapeutics | Conjugados poliméricos de antagonistas de opioides |
US20050191340A1 (en) * | 2002-08-09 | 2005-09-01 | Gruenenthal Gmbh | Opioid-receptor antagonists in transdermal systems having buprenorphine |
EP2604282B1 (en) * | 2003-12-16 | 2019-06-19 | Nektar Therapeutics | Method for preparing of monodisperse oligo ethylene glycol |
ES2586245T3 (es) * | 2007-08-09 | 2016-10-13 | Rensselaer Polytechnic Institute | Carboxamidas cuaternarias opioides |
NZ600379A (en) | 2009-12-04 | 2014-05-30 | Alkermes Pharma Ireland Ltd | Morphinan derivatives for the treatment of drug overdose |
JP5964809B2 (ja) | 2010-03-22 | 2016-08-03 | レンセラール ポリテクニック インスティチュート | オピオイド受容体リガンドとしてのカルボキサミド基を含有するモルヒネ誘導体 |
CA2807965C (en) | 2010-08-23 | 2016-03-15 | Alkermes Pharma Ireland Limited | Methods for treating antipsychotic-induced weight gain |
LT2725908T (lt) | 2011-06-29 | 2017-09-11 | Alkermes, Inc. | Periferinio poveikio opioidų junginiai |
US9211293B2 (en) | 2011-12-15 | 2015-12-15 | Alkermes Pharma Ireland Limited | Opioid agonist antagonist combinations |
US9656961B2 (en) | 2013-05-24 | 2017-05-23 | Alkermes Pharma Ireland Limited | Methods for treating depressive symptoms |
CA2911231C (en) | 2013-05-24 | 2021-12-07 | Alkermes Pharma Ireland Limited | Morphan and morphinan analogues, and methods of use |
EP4243768A1 (en) | 2020-11-12 | 2023-09-20 | Alkermes Pharma Ireland Limited | Immediate release multilayer tablet |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4176186A (en) * | 1978-07-28 | 1979-11-27 | Boehringer Ingelheim Gmbh | Quaternary derivatives of noroxymorphone which relieve intestinal immobility |
-
1981
- 1981-10-19 FR FR8119607A patent/FR2514644A1/fr active Granted
-
1982
- 1982-09-22 IL IL66853A patent/IL66853A/xx unknown
- 1982-09-24 US US06/422,568 patent/US4489079A/en not_active Expired - Fee Related
- 1982-09-27 ZA ZA827063A patent/ZA827063B/xx unknown
- 1982-09-30 AU AU88922/82A patent/AU559451B2/en not_active Expired - Fee Related
- 1982-10-12 JP JP57177719A patent/JPS5874608A/ja active Pending
- 1982-10-13 AT AT82401876T patent/ATE17942T1/de not_active IP Right Cessation
- 1982-10-13 DE DE8282401876T patent/DE3269082D1/de not_active Expired
- 1982-10-13 EP EP82401876A patent/EP0077723B1/fr not_active Expired
- 1982-10-18 NZ NZ202210A patent/NZ202210A/en unknown
Also Published As
Publication number | Publication date |
---|---|
NZ202210A (en) | 1985-03-20 |
DE3269082D1 (en) | 1986-03-27 |
AU559451B2 (en) | 1987-03-12 |
IL66853A (en) | 1985-08-30 |
JPS5874608A (ja) | 1983-05-06 |
AU8892282A (en) | 1983-04-28 |
IL66853A0 (en) | 1982-12-31 |
EP0077723A1 (fr) | 1983-04-27 |
FR2514644B1 (xx) | 1984-04-20 |
ATE17942T1 (de) | 1986-02-15 |
EP0077723B1 (fr) | 1986-02-12 |
US4489079A (en) | 1984-12-18 |
FR2514644A1 (fr) | 1983-04-22 |
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