ZA822083B - N-substituted-amido-amino acids - Google Patents

N-substituted-amido-amino acids

Info

Publication number
ZA822083B
ZA822083B ZA822083A ZA822083A ZA822083B ZA 822083 B ZA822083 B ZA 822083B ZA 822083 A ZA822083 A ZA 822083A ZA 822083 A ZA822083 A ZA 822083A ZA 822083 B ZA822083 B ZA 822083B
Authority
ZA
South Africa
Prior art keywords
alkyl
carbon atoms
lower alkoxy
amino
heterocyclic
Prior art date
Application number
ZA822083A
Other languages
English (en)
Inventor
J Skiles
R Youssefyeh
J Suh
H Jones
Original Assignee
Usv Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Usv Pharma Corp filed Critical Usv Pharma Corp
Publication of ZA822083B publication Critical patent/ZA822083B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
ZA822083A 1981-03-30 1982-03-26 N-substituted-amido-amino acids ZA822083B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24905381A 1981-03-30 1981-03-30

Publications (1)

Publication Number Publication Date
ZA822083B true ZA822083B (en) 1983-02-23

Family

ID=22941861

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA822083A ZA822083B (en) 1981-03-30 1982-03-26 N-substituted-amido-amino acids

Country Status (10)

Country Link
EP (1) EP0061768B1 (ja)
JP (1) JPS57175152A (ja)
KR (1) KR830008998A (ja)
AT (1) ATE19782T1 (ja)
AU (1) AU556932B2 (ja)
DE (1) DE3271116D1 (ja)
IL (1) IL65347A (ja)
NZ (1) NZ200162A (ja)
PH (3) PH20083A (ja)
ZA (1) ZA822083B (ja)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820729A (en) * 1981-03-30 1989-04-11 Rorer Pharmaceutical Corporation N-substituted-amido-amino acids
US4686295A (en) * 1982-03-10 1987-08-11 Usv Pharmaceutical Corporation N-carboxy anhydride intermediates
US4482544A (en) * 1982-11-29 1984-11-13 Usv Pharmaceutical Corporation Compounds for treating hypertension
JPS6248696A (ja) * 1985-08-27 1987-03-03 Kanegafuchi Chem Ind Co Ltd Ｎ−〔１（ｓ）−エトキシカルボニル−３−フエニルプロピル〕−ｌ−アラニル−ｌ−プロリンの製造法
US5079366A (en) * 1987-04-07 1992-01-07 University Of Florida Quarternary pyridinium salts
US4888427A (en) * 1987-04-07 1989-12-19 University Of Florida Amino acids containing dihydropyridine ring systems for site-specific delivery of peptides to the brain
FR2626279B1 (fr) * 1988-01-26 1990-07-13 Roussel Uclaf Nouveaux derives de l'indolo(3,2,1-de)(1,4)-oxazino(2,3,4-ij)(1,5) naphthyridine, leur procede de preparation et les nouveaux intermediaires ainsi obtenus, leur application comme medicaments et les compositions les renfermant
CA2614099A1 (en) 2005-07-05 2007-01-11 Cipla Limited Process for the synthesis of the ace inhibitor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL58849A (en) * 1978-12-11 1983-03-31 Merck & Co Inc Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them
US4256761A (en) * 1979-07-13 1981-03-17 Usv Pharmaceutical Corporation Antihypertensive amides

Also Published As

Publication number Publication date
JPH0448800B2 (ja) 1992-08-07
AU556932B2 (en) 1986-11-27
IL65347A0 (en) 1982-05-31
PH20083A (en) 1986-09-24
JPS57175152A (en) 1982-10-28
IL65347A (en) 1987-12-31
NZ200162A (en) 1985-08-16
DE3271116D1 (de) 1986-06-19
EP0061768A1 (en) 1982-10-06
EP0061768B1 (en) 1986-05-14
AU8170682A (en) 1982-10-07
PH21449A (en) 1987-10-28
KR830008998A (ko) 1983-12-16
PH21632A (en) 1988-01-13
ATE19782T1 (de) 1986-05-15

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