ZA200804732B - Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivatives - Google Patents
Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivativesInfo
- Publication number
- ZA200804732B ZA200804732B ZA200804732A ZA200804732A ZA200804732B ZA 200804732 B ZA200804732 B ZA 200804732B ZA 200804732 A ZA200804732 A ZA 200804732A ZA 200804732 A ZA200804732 A ZA 200804732A ZA 200804732 B ZA200804732 B ZA 200804732B
- Authority
- ZA
- South Africa
- Prior art keywords
- diazapanyl
- piperazinyl
- preparation
- novel processes
- benzamide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/06—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with radicals, containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US73194105P | 2005-10-31 | 2005-10-31 |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA200804732B true ZA200804732B (en) | 2009-11-25 |
Family
ID=37766699
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200804732A ZA200804732B (en) | 2005-10-31 | 2008-05-30 | Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivatives |
Country Status (19)
Country | Link |
---|---|
US (2) | US7728129B2 (zh) |
EP (2) | EP1951700A2 (zh) |
JP (1) | JP2009513702A (zh) |
KR (1) | KR20080067365A (zh) |
CN (1) | CN101389617A (zh) |
AR (1) | AR056750A1 (zh) |
AU (1) | AU2006309077A1 (zh) |
BR (1) | BRPI0617947A2 (zh) |
CA (1) | CA2628210A1 (zh) |
CR (1) | CR10037A (zh) |
EA (2) | EA014905B1 (zh) |
EC (1) | ECSP088416A (zh) |
IL (1) | IL190963A0 (zh) |
NO (1) | NO20082459L (zh) |
NZ (1) | NZ567357A (zh) |
SV (1) | SV2009002893A (zh) |
TW (1) | TW200736239A (zh) |
WO (1) | WO2007053427A2 (zh) |
ZA (1) | ZA200804732B (zh) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0324159D0 (en) | 2003-10-15 | 2003-11-19 | Glaxo Group Ltd | Novel compounds |
CA2672661C (en) * | 2006-12-14 | 2015-04-28 | Janssen Pharmaceutica N.V. | Process for the preparation of piperazinyl and diazepanyl benzamide derivatives |
CA2697941A1 (en) | 2007-09-06 | 2009-03-12 | Glaxo Group Limited | Piperazine derivative having affinity for the histamine h3 receptor |
CN111610246B (zh) * | 2019-02-25 | 2023-05-12 | 中国科学院上海有机化学研究所 | 用于质谱检测的羧基衍生化试剂组合物及其用途 |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9807354D0 (en) * | 1998-04-07 | 1998-06-03 | Glaxo Group Ltd | Antiviral compound |
US7141593B1 (en) * | 1999-06-04 | 2006-11-28 | Abbott Laboratories | Pharmaceutical formulations |
SK5202000A3 (en) | 2000-04-07 | 2001-12-03 | Slovakofarma As | Method for the preparation of (e)-n-(6,6-dimethyl-2-hepten-4- inyl)-n-methyl-1-naphthalenemethylamine (terbinaphin) |
DK1296939T3 (da) * | 2000-07-05 | 2006-01-30 | Basf Ag | Fremgangsmåde til fremstilling af trioximderivater |
ATE404575T1 (de) * | 2001-05-22 | 2008-08-15 | Pfizer Prod Inc | Neue kristallforme von azithromycin |
US6548670B1 (en) | 2001-07-19 | 2003-04-15 | Air Products And Chemicals, Inc. | Methods for preparing 5- and 6-benzyl-functionalized quinoxalines |
US6821502B2 (en) * | 2002-06-12 | 2004-11-23 | Chevron U.S.A. Inc. | Method of making aluminum-containing zeolite with IFR structure |
UA80573C2 (en) | 2002-10-23 | 2007-10-10 | Janssen Pharmaceutica Nv | Piperazinyl and diazapanyl benzamides and benzthioamides |
WO2005021525A1 (en) * | 2003-08-27 | 2005-03-10 | Janssen Pharmaceutica, N.V. | Aryl piperidine amides |
AR047541A1 (es) * | 2004-02-13 | 2006-01-25 | Sandoz Ag | Fosfato de 5-[[4-[2-metil-2-piridinil-amino-etoxi]fenil]metil]-2,4 tiazolidinadiona (rosiglitazona) y sus formas polimorficas |
US7351833B2 (en) * | 2004-07-23 | 2008-04-01 | Abbott Laboratories | (1S,5S)-3-(5,6-dichloropyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane benzenesulfonate |
US8436176B2 (en) * | 2004-12-30 | 2013-05-07 | Medicis Pharmaceutical Corporation | Process for preparing 2-methyl-1-(2-methylpropyl)-1H-imidazo[4,5-c][1,5]naphthyridin-4-amine |
UA91546C2 (uk) * | 2005-05-03 | 2010-08-10 | Бьорінгер Інгельхайм Інтернаціональ Гмбх | КРИСТАЛІЧНА ФОРМА 1-ХЛОР-4-(β-D-ГЛЮКОПІРАНОЗ-1-ИЛ)-2-[4-((S)-ТЕТРАГІДРОФУРАН-3-ІЛОКСИ)-БЕНЗИЛ]-БЕНЗОЛУ, СПОСІБ ЇЇ ОДЕРЖАННЯ ТА ЇЇ ЗАСТОСУВАННЯ ПРИ ПРИГОТУВАННІ ЛІКАРСЬКИХ ЗАСОБІВ |
MY152185A (en) * | 2005-06-10 | 2014-08-29 | Novartis Ag | Modified release 1-[(3-hydroxy-adamant-1-ylamino)-acetyl]-pyrrolidine-2(s)-carbonitrile formulation |
WO2007027525A1 (en) * | 2005-08-29 | 2007-03-08 | Sanofi-Aventis U.S. Llc | Novel crystalline form of a pyridazino [4 , 5-b] indole derivative |
JP2008522983A (ja) * | 2005-09-13 | 2008-07-03 | シコール インコーポレイティド | ロクロニウムブロミドの合成方法 |
CA2663569A1 (en) * | 2006-09-28 | 2008-04-03 | Merck & Co., Inc. | Pharmaceutical compositions of hdac inhibitors and chelatable metal compounds, and metal-hdac inhibitor chelate complexes |
US7837978B2 (en) * | 2006-10-13 | 2010-11-23 | Chevron U.S.A. Inc. | Process for preparing aluminum-containing molecular sieve SSZ-26 |
PE20081506A1 (es) * | 2006-12-12 | 2008-12-09 | Infinity Discovery Inc | Formulaciones de ansamicina |
CN101778855A (zh) * | 2007-05-22 | 2010-07-14 | 阿尔迪默菲克斯技术有限责任公司 | 替诺福韦酯半富马酸共晶体 |
TW200944520A (en) * | 2008-01-29 | 2009-11-01 | Glaxo Group Ltd | Spiro compounds as NPY Y5 receptor antagonists |
-
2006
- 2006-10-26 NZ NZ567357A patent/NZ567357A/en not_active IP Right Cessation
- 2006-10-26 KR KR1020087013062A patent/KR20080067365A/ko not_active Application Discontinuation
- 2006-10-26 EA EA200801239A patent/EA014905B1/ru unknown
- 2006-10-26 JP JP2008538930A patent/JP2009513702A/ja active Pending
- 2006-10-26 EP EP06826786A patent/EP1951700A2/en not_active Withdrawn
- 2006-10-26 US US11/553,158 patent/US7728129B2/en active Active
- 2006-10-26 WO PCT/US2006/041859 patent/WO2007053427A2/en active Application Filing
- 2006-10-26 EA EA201001799A patent/EA201001799A1/ru unknown
- 2006-10-26 CA CA002628210A patent/CA2628210A1/en not_active Abandoned
- 2006-10-26 CN CNA2006800406803A patent/CN101389617A/zh active Pending
- 2006-10-26 BR BRPI0617947-9A patent/BRPI0617947A2/pt not_active IP Right Cessation
- 2006-10-26 AU AU2006309077A patent/AU2006309077A1/en not_active Abandoned
- 2006-10-26 EP EP11183817A patent/EP2404911A1/en not_active Withdrawn
- 2006-10-30 TW TW095139961A patent/TW200736239A/zh unknown
- 2006-10-31 AR ARP060104773A patent/AR056750A1/es not_active Application Discontinuation
-
2008
- 2008-04-17 IL IL190963A patent/IL190963A0/en unknown
- 2008-04-30 EC EC2008008416A patent/ECSP088416A/es unknown
- 2008-04-30 SV SV2008002893A patent/SV2009002893A/es not_active Application Discontinuation
- 2008-05-30 ZA ZA200804732A patent/ZA200804732B/xx unknown
- 2008-05-30 CR CR10037A patent/CR10037A/es not_active Application Discontinuation
- 2008-05-30 NO NO20082459A patent/NO20082459L/no not_active Application Discontinuation
-
2010
- 2010-04-19 US US12/762,912 patent/US20100197689A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN101389617A (zh) | 2009-03-18 |
WO2007053427A3 (en) | 2007-07-12 |
NO20082459L (no) | 2008-07-22 |
AU2006309077A1 (en) | 2007-05-10 |
CA2628210A1 (en) | 2007-05-10 |
SV2009002893A (es) | 2009-06-18 |
EA200801239A1 (ru) | 2008-08-29 |
US20100197689A1 (en) | 2010-08-05 |
EA014905B1 (ru) | 2011-02-28 |
JP2009513702A (ja) | 2009-04-02 |
WO2007053427A2 (en) | 2007-05-10 |
EP1951700A2 (en) | 2008-08-06 |
KR20080067365A (ko) | 2008-07-18 |
CR10037A (es) | 2008-11-24 |
NZ567357A (en) | 2011-05-27 |
EP2404911A1 (en) | 2012-01-11 |
BRPI0617947A2 (pt) | 2011-08-09 |
TW200736239A (en) | 2007-10-01 |
EA201001799A1 (ru) | 2011-06-30 |
IL190963A0 (en) | 2008-12-29 |
AR056750A1 (es) | 2007-10-24 |
US7728129B2 (en) | 2010-06-01 |
ECSP088416A (es) | 2008-05-30 |
US20070197508A1 (en) | 2007-08-23 |
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