ZA200607981B - Azaindoles useful as inhibitors of jak and other protein kinases - Google Patents
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| SI (1) | SI2332940T1 (zh) |
| UA (1) | UA87494C2 (zh) |
| ZA (1) | ZA200607981B (zh) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI1012159B1 (pt) * | 2009-05-22 | 2022-01-25 | Incyte Holdings Corporation | Compostos derivados de n-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo[2,3-d] pirimidinas e pirrol-3-il-pirrolo[2,3-d] pirimidinas como inibidores de janus cinase, composições farmacêuticas compreendendo os referidos compostos e usos dos mesmos |
| EP2528917B1 (en) * | 2010-01-27 | 2016-10-19 | Vertex Pharmaceuticals Incorporated | Pyrazolopyridines useful for the treatment of autoimmune, inflammatory or (hyper)proliferative diseases |
| KR20130094693A (ko) * | 2010-04-30 | 2013-08-26 | 셀좀 리미티드 | Ｊａｋ 저해제로서의 피라졸 화합물 |
| CA2822057A1 (en) * | 2010-12-16 | 2012-06-21 | Vertex Pharmaceuticals Incorporated | Inhibitors of influenza viruses replication |
| CN103562205A (zh) * | 2010-12-16 | 2014-02-05 | 沃泰克斯药物股份有限公司 | 流感病毒复制的抑制剂 |
| JP2013545817A (ja) * | 2010-12-16 | 2013-12-26 | バーテックス ファーマシューティカルズ インコーポレイテッド | インフルエンザウイルス複製阻害物質 |
| DE102011009961A1 (de) * | 2011-02-01 | 2012-08-02 | Merck Patent Gmbh | 7-Azaindolderivate |
| EP2487159A1 (en) * | 2011-02-11 | 2012-08-15 | MSD Oss B.V. | RorgammaT inhibitors |
| PL3141548T3 (pl) * | 2011-07-05 | 2020-09-07 | Vertex Pharmaceuticals Incorporated | Sposoby i związki pośrednie do wytwarzania azaindoli |
| CN109641868B (zh) * | 2016-08-30 | 2021-12-03 | 广东东阳光药业有限公司 | 流感病毒复制抑制剂及其使用方法和用途 |
| CN110128421B (zh) * | 2018-02-09 | 2020-08-11 | 新发药业有限公司 | 一种5-卤代-7-氮杂吲哚的简便制备方法 |
| CN108299426B (zh) * | 2018-03-20 | 2020-09-04 | 宝鸡文理学院 | 一种[1,2,4]-三唑并[4,3-a]吡啶类化合物及其合成方法 |
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Also Published As
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| SI2332940T1 (sl) | 2013-03-29 |
| CN1938303A (zh) | 2007-03-28 |
| CN100569772C (zh) | 2009-12-16 |
| UA87494C2 (en) | 2009-07-27 |
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