ZA200603601B - 1-(quinoline amino) and 1-(isoquinoline amino)-substituted pentan-2-ols, method for their production and their use as anti-inflammatories - Google Patents
1-(quinoline amino) and 1-(isoquinoline amino)-substituted pentan-2-ols, method for their production and their use as anti-inflammatories Download PDFInfo
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- ZA200603601B ZA200603601B ZA200603601A ZA200603601A ZA200603601B ZA 200603601 B ZA200603601 B ZA 200603601B ZA 200603601 A ZA200603601 A ZA 200603601A ZA 200603601 A ZA200603601 A ZA 200603601A ZA 200603601 B ZA200603601 B ZA 200603601B
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- alkyl
- group
- cycloalkyl
- aryl
- compounds
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- 238000004519 manufacturing process Methods 0.000 title claims description 11
- 238000000034 method Methods 0.000 title description 25
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P31/04—Antibacterial agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
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- A—HUMAN NECESSITIES
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- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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- A—HUMAN NECESSITIES
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- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Diabetes (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Rheumatology (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Communicable Diseases (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Transplantation (AREA)
- Gastroenterology & Hepatology (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10346940A DE10346940B3 (de) | 2003-10-06 | 2003-10-06 | Substituierte Pentanole, ihre Verwendung zur Herstellung von Arzneimitteln speziell Entzündungshemmer sowie diese enthaltende pharmazeutische Präparate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200603601B true ZA200603601B (en) | 2007-07-25 |
Family
ID=34428261
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200603601A ZA200603601B (en) | 2003-10-06 | 2006-05-05 | 1-(quinoline amino) and 1-(isoquinoline amino)-substituted pentan-2-ols, method for their production and their use as anti-inflammatories |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP1673344A1 (fr) |
| JP (1) | JP2007507450A (fr) |
| KR (1) | KR20060121894A (fr) |
| CN (1) | CN1863775A (fr) |
| AU (1) | AU2004279544A1 (fr) |
| BR (1) | BRPI0415084A (fr) |
| CA (1) | CA2539572A1 (fr) |
| DE (1) | DE10346940B3 (fr) |
| IL (1) | IL174433A0 (fr) |
| MX (1) | MXPA06003895A (fr) |
| NO (1) | NO20062022L (fr) |
| WO (1) | WO2005035502A1 (fr) |
| ZA (1) | ZA200603601B (fr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2009246870B2 (en) | 2008-05-14 | 2013-08-01 | Otonomy, Inc. | Controlled release corticosteroid compositions and methods for the treatment of otic disorders |
| US8236786B2 (en) | 2008-08-07 | 2012-08-07 | Pulmagen Therapeutics (Inflammation) Limited | Respiratory disease treatment |
| ES2442343T3 (es) | 2008-12-30 | 2014-02-11 | Pulmagen Therapeutics (Inflammation) Limited | Compuestos de sulfonamida para el tratamiento de trastornos respiratorios |
| WO2010150014A1 (fr) | 2009-06-24 | 2010-12-29 | Pulmagen Therapeutics (Inflammation) Limited | Glitazones 5r-5–deutérés pour le traitement de maladies respiratoires |
| WO2011098746A1 (fr) | 2010-02-09 | 2011-08-18 | Pulmagen Therapeutics (Inflammation) Limited | Sels d'addition acide cristallins de l'énantiomère (5r) de la pioglitazone |
| GB201002243D0 (en) | 2010-02-10 | 2010-03-31 | Argenta Therapeutics Ltd | Respiratory disease treatment |
| GB201002224D0 (en) | 2010-02-10 | 2010-03-31 | Argenta Therapeutics Ltd | Respiratory disease treatment |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19723722A1 (de) * | 1997-05-30 | 1998-12-10 | Schering Ag | Nichtsteroidale Gestagene |
| DE19856475A1 (de) * | 1998-11-27 | 2000-05-31 | Schering Ag | Nichtsteroidale Entzündungshemmer |
| DE10038639A1 (de) * | 2000-07-28 | 2002-02-21 | Schering Ag | Nichtsteroidale Entzündungshemmer |
| DE10215316C1 (de) * | 2002-04-02 | 2003-12-18 | Schering Ag | Chinolin- und Isochinolin-Derivate, ein pharmazeutisches Mittel und ihre Verwendung als Entzündungshemmer |
-
2003
- 2003-10-06 DE DE10346940A patent/DE10346940B3/de not_active Withdrawn - After Issue
-
2004
- 2004-09-24 EP EP04787047A patent/EP1673344A1/fr not_active Withdrawn
- 2004-09-24 AU AU2004279544A patent/AU2004279544A1/en not_active Abandoned
- 2004-09-24 KR KR1020067006547A patent/KR20060121894A/ko not_active Application Discontinuation
- 2004-09-24 JP JP2006530041A patent/JP2007507450A/ja active Pending
- 2004-09-24 CA CA002539572A patent/CA2539572A1/fr not_active Abandoned
- 2004-09-24 WO PCT/EP2004/010880 patent/WO2005035502A1/fr active Application Filing
- 2004-09-24 BR BRPI0415084-8A patent/BRPI0415084A/pt not_active Application Discontinuation
- 2004-09-24 CN CNA2004800292061A patent/CN1863775A/zh active Pending
- 2004-09-24 MX MXPA06003895A patent/MXPA06003895A/es not_active Application Discontinuation
-
2006
- 2006-03-21 IL IL174433A patent/IL174433A0/en unknown
- 2006-05-05 NO NO20062022A patent/NO20062022L/no unknown
- 2006-05-05 ZA ZA200603601A patent/ZA200603601B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL174433A0 (en) | 2006-08-01 |
| NO20062022L (no) | 2006-05-05 |
| CA2539572A1 (fr) | 2005-04-21 |
| EP1673344A1 (fr) | 2006-06-28 |
| DE10346940B3 (de) | 2005-06-16 |
| MXPA06003895A (es) | 2006-07-03 |
| BRPI0415084A (pt) | 2006-12-12 |
| WO2005035502A1 (fr) | 2005-04-21 |
| AU2004279544A1 (en) | 2005-04-21 |
| CN1863775A (zh) | 2006-11-15 |
| JP2007507450A (ja) | 2007-03-29 |
| KR20060121894A (ko) | 2006-11-29 |
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