ZA200508568B - Cannabinoid receptor ligands and uses thereof - Google Patents
Cannabinoid receptor ligands and uses thereof Download PDFInfo
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- ZA200508568B ZA200508568B ZA200508568A ZA200508568A ZA200508568B ZA 200508568 B ZA200508568 B ZA 200508568B ZA 200508568 A ZA200508568 A ZA 200508568A ZA 200508568 A ZA200508568 A ZA 200508568A ZA 200508568 B ZA200508568 B ZA 200508568B
- Authority
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- South Africa
- Prior art keywords
- compound
- alkyl
- composition
- pharmaceutically acceptable
- salt
- Prior art date
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- 150000003335 secondary amines Chemical class 0.000 description 1
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- KDYFGRWQOYBRFD-UHFFFAOYSA-L succinate(2-) Chemical compound [O-]C(=O)CCC([O-])=O KDYFGRWQOYBRFD-UHFFFAOYSA-L 0.000 description 1
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- YBBRCQOCSYXUOC-UHFFFAOYSA-N sulfuryl dichloride Chemical class ClS(Cl)(=O)=O YBBRCQOCSYXUOC-UHFFFAOYSA-N 0.000 description 1
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- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 description 1
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- AVCVDUDESCZFHJ-UHFFFAOYSA-N triphenylphosphane;hydrochloride Chemical compound [Cl-].C1=CC=CC=C1[PH+](C=1C=CC=CC=1)C1=CC=CC=C1 AVCVDUDESCZFHJ-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
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- Pyrane Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
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US46490803P | 2003-04-23 | 2003-04-23 |
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Country Status (31)
Country | Link |
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US (1) | US20040214856A1 (xx) |
EP (1) | EP1622903B1 (xx) |
JP (1) | JP2006524225A (xx) |
KR (1) | KR20060006048A (xx) |
CN (1) | CN1809566A (xx) |
AP (1) | AP2005003427A0 (xx) |
AR (1) | AR044037A1 (xx) |
AT (1) | ATE409700T1 (xx) |
AU (1) | AU2004232552A1 (xx) |
BR (1) | BRPI0409791A (xx) |
CA (1) | CA2521538A1 (xx) |
CL (1) | CL2004000827A1 (xx) |
CO (1) | CO5640084A2 (xx) |
DE (1) | DE602004016839D1 (xx) |
EA (1) | EA200501504A1 (xx) |
EC (1) | ECSP056117A (xx) |
ES (1) | ES2309517T3 (xx) |
GT (1) | GT200400076A (xx) |
IS (1) | IS8054A (xx) |
MA (1) | MA27766A1 (xx) |
MX (1) | MXPA05011454A (xx) |
NL (1) | NL1026027C2 (xx) |
NO (1) | NO20055516L (xx) |
OA (1) | OA13047A (xx) |
PA (1) | PA8600601A1 (xx) |
PE (1) | PE20050419A1 (xx) |
TN (1) | TNSN05272A1 (xx) |
TW (1) | TW200510419A (xx) |
UY (1) | UY28276A1 (xx) |
WO (1) | WO2004094421A1 (xx) |
ZA (1) | ZA200508568B (xx) |
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EP1546115A4 (en) | 2002-09-27 | 2010-08-04 | Merck Sharp & Dohme | SUBSTITUTED PYRIMIDINES |
US7094572B2 (en) * | 2003-03-14 | 2006-08-22 | Bristol-Myers Squibb | Polynucleotide encoding a novel human G-protein coupled receptor variant of HM74, HGPRBMY74 |
US7141669B2 (en) * | 2003-04-23 | 2006-11-28 | Pfizer Inc. | Cannabiniod receptor ligands and uses thereof |
US7268133B2 (en) | 2003-04-23 | 2007-09-11 | Pfizer, Inc. Patent Department | Cannabinoid receptor ligands and uses thereof |
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-
2004
- 2004-04-12 US US10/823,152 patent/US20040214856A1/en not_active Abandoned
- 2004-04-13 AT AT04727076T patent/ATE409700T1/de not_active IP Right Cessation
- 2004-04-13 AU AU2004232552A patent/AU2004232552A1/en not_active Abandoned
- 2004-04-13 WO PCT/IB2004/001357 patent/WO2004094421A1/en active IP Right Grant
- 2004-04-13 CN CNA2004800175674A patent/CN1809566A/zh active Pending
- 2004-04-13 MX MXPA05011454A patent/MXPA05011454A/es unknown
- 2004-04-13 JP JP2006506562A patent/JP2006524225A/ja not_active Abandoned
- 2004-04-13 ES ES04727076T patent/ES2309517T3/es not_active Expired - Lifetime
- 2004-04-13 DE DE602004016839T patent/DE602004016839D1/de not_active Expired - Fee Related
- 2004-04-13 CA CA002521538A patent/CA2521538A1/en not_active Abandoned
- 2004-04-13 OA OA1200500291A patent/OA13047A/en unknown
- 2004-04-13 KR KR1020057020010A patent/KR20060006048A/ko not_active Application Discontinuation
- 2004-04-13 AP AP2005003427A patent/AP2005003427A0/xx unknown
- 2004-04-13 BR BRPI0409791-2A patent/BRPI0409791A/pt not_active IP Right Cessation
- 2004-04-13 EP EP04727076A patent/EP1622903B1/en not_active Expired - Lifetime
- 2004-04-13 EA EA200501504A patent/EA200501504A1/ru unknown
- 2004-04-16 CL CL200400827A patent/CL2004000827A1/es unknown
- 2004-04-20 GT GT200400076A patent/GT200400076A/es unknown
- 2004-04-20 PA PA20048600601A patent/PA8600601A1/es unknown
- 2004-04-20 PE PE2004000389A patent/PE20050419A1/es not_active Application Discontinuation
- 2004-04-21 AR ARP040101339A patent/AR044037A1/es unknown
- 2004-04-21 UY UY28276A patent/UY28276A1/es not_active Application Discontinuation
- 2004-04-22 TW TW093111297A patent/TW200510419A/zh unknown
- 2004-04-23 NL NL1026027A patent/NL1026027C2/nl not_active IP Right Cessation
-
2005
- 2005-09-29 IS IS8054A patent/IS8054A/is unknown
- 2005-10-21 TN TNP2005000272A patent/TNSN05272A1/fr unknown
- 2005-10-21 EC EC2005006117A patent/ECSP056117A/es unknown
- 2005-10-21 CO CO05106974A patent/CO5640084A2/es not_active Application Discontinuation
- 2005-10-21 ZA ZA200508568A patent/ZA200508568B/en unknown
- 2005-10-21 MA MA28565A patent/MA27766A1/fr unknown
- 2005-11-22 NO NO20055516A patent/NO20055516L/no not_active Application Discontinuation
Also Published As
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AR044037A1 (es) | 2005-08-24 |
ECSP056117A (es) | 2006-03-01 |
ES2309517T3 (es) | 2008-12-16 |
PA8600601A1 (es) | 2005-05-24 |
KR20060006048A (ko) | 2006-01-18 |
CO5640084A2 (es) | 2006-05-31 |
WO2004094421A1 (en) | 2004-11-04 |
TNSN05272A1 (fr) | 2007-07-10 |
AP2005003427A0 (en) | 2005-12-31 |
TW200510419A (en) | 2005-03-16 |
OA13047A (en) | 2006-11-10 |
DE602004016839D1 (de) | 2008-11-13 |
MXPA05011454A (es) | 2005-12-12 |
NO20055516L (no) | 2005-11-22 |
IS8054A (is) | 2005-09-29 |
GT200400076A (es) | 2004-12-16 |
EP1622903A1 (en) | 2006-02-08 |
MA27766A1 (fr) | 2006-02-01 |
AU2004232552A1 (en) | 2004-11-04 |
CA2521538A1 (en) | 2004-11-04 |
UY28276A1 (es) | 2004-11-30 |
NL1026027A1 (nl) | 2004-10-27 |
JP2006524225A (ja) | 2006-10-26 |
EP1622903B1 (en) | 2008-10-01 |
NL1026027C2 (nl) | 2005-07-05 |
EA200501504A1 (ru) | 2006-04-28 |
BRPI0409791A (pt) | 2006-05-30 |
PE20050419A1 (es) | 2005-06-18 |
ATE409700T1 (de) | 2008-10-15 |
CN1809566A (zh) | 2006-07-26 |
CL2004000827A1 (es) | 2005-03-04 |
US20040214856A1 (en) | 2004-10-28 |
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