ZA200308859B - Pyrimidine, triazine and pyrazine derivatives as glutamate receptors. - Google Patents

Pyrimidine, triazine and pyrazine derivatives as glutamate receptors. Download PDF

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Publication number
ZA200308859B
ZA200308859B ZA200308859A ZA200308859A ZA200308859B ZA 200308859 B ZA200308859 B ZA 200308859B ZA 200308859 A ZA200308859 A ZA 200308859A ZA 200308859 A ZA200308859 A ZA 200308859A ZA 200308859 B ZA200308859 B ZA 200308859B
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South Africa
Prior art keywords
phenyl
carbonitrile
pyrimidine
formula
fluoro
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ZA200308859A
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English (en)
Inventor
Alfred Binggeli
Thierry Masquelin
Maurice Wilhelm
Hans-Peter Maerki
Vincent Mutel
Wolfgang Wostl
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Hoffmann La Roche
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Publication of ZA200308859B publication Critical patent/ZA200308859B/en

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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
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    • C07D253/06—1,2,4-Triazines
    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
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ZA200308859A 2001-06-01 2003-11-13 Pyrimidine, triazine and pyrazine derivatives as glutamate receptors. ZA200308859B (en)

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Application Number Priority Date Filing Date Title
EP01113379 2001-06-01

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ZA200308859B true ZA200308859B (en) 2005-02-14

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ZA200308859A ZA200308859B (en) 2001-06-01 2003-11-13 Pyrimidine, triazine and pyrazine derivatives as glutamate receptors.

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EP (1) EP1397351B1 (enExample)
JP (1) JP4049742B2 (enExample)
KR (1) KR100602927B1 (enExample)
CN (1) CN1245391C (enExample)
AR (1) AR036075A1 (enExample)
AT (1) ATE448210T1 (enExample)
AU (1) AU2002319183B2 (enExample)
BR (1) BR0210102A (enExample)
CA (1) CA2448602C (enExample)
DE (1) DE60234338D1 (enExample)
DK (1) DK1397351T3 (enExample)
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PT (1) PT1397351E (enExample)
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JP4049742B2 (ja) 2008-02-20
KR100602927B1 (ko) 2006-07-20
US20030060466A1 (en) 2003-03-27
CA2448602A1 (en) 2002-12-12
KR20040003039A (ko) 2004-01-07
DK1397351T3 (da) 2010-01-18
WO2002098864A1 (en) 2002-12-12
MXPA03010822A (es) 2004-02-17
JP2004536814A (ja) 2004-12-09
BR0210102A (pt) 2004-06-08
CN1245391C (zh) 2006-03-15
CA2448602C (en) 2009-03-31
ATE448210T1 (de) 2009-11-15
EP1397351B1 (en) 2009-11-11
CN1512988A (zh) 2004-07-14
PT1397351E (pt) 2010-01-04
EP1397351A1 (en) 2004-03-17
ES2332505T3 (es) 2010-02-08
DE60234338D1 (de) 2009-12-24
US6673795B2 (en) 2004-01-06
AR036075A1 (es) 2004-08-11
AU2002319183B2 (en) 2007-05-10

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