ZA200301865B - New treatments for restless legs syndrome. - Google Patents
New treatments for restless legs syndrome. Download PDFInfo
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- ZA200301865B ZA200301865B ZA200301865A ZA200301865A ZA200301865B ZA 200301865 B ZA200301865 B ZA 200301865B ZA 200301865 A ZA200301865 A ZA 200301865A ZA 200301865 A ZA200301865 A ZA 200301865A ZA 200301865 B ZA200301865 B ZA 200301865B
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- South Africa
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
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- Animal Behavior & Ethology (AREA)
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- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Hydrogenated Pyridines (AREA)
- Fats And Perfumes (AREA)
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| US24466600P | 2000-10-31 | 2000-10-31 |
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| EP (1) | EP1330248A2 (fr) |
| JP (1) | JP2004512367A (fr) |
| KR (1) | KR20030042037A (fr) |
| CN (1) | CN1606442A (fr) |
| AR (1) | AR031152A1 (fr) |
| AU (1) | AU2002211226A1 (fr) |
| BR (1) | BR0115071A (fr) |
| CA (1) | CA2421705A1 (fr) |
| EA (1) | EA200300527A1 (fr) |
| IL (1) | IL155591A0 (fr) |
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| PE (1) | PE20020514A1 (fr) |
| PL (1) | PL360904A1 (fr) |
| WO (1) | WO2002036123A2 (fr) |
| ZA (1) | ZA200301865B (fr) |
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| CA2314893C (fr) | 1997-12-22 | 2005-09-13 | Euro-Celtique, S.A. | Combinaison d'agonistes et d'antagonistes d'opioides |
| US6375957B1 (en) | 1997-12-22 | 2002-04-23 | Euro-Celtique, S.A. | Opioid agonist/opioid antagonist/acetaminophen combinations |
| USRE46117E1 (en) | 1999-12-22 | 2016-08-23 | Teva Pharmaceuticals International Gmbh | Modulators of dopamine neurotransmission |
| DE10053397A1 (de) * | 2000-10-20 | 2002-05-02 | Schering Ag | Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen |
| DE10066158B4 (de) * | 2000-08-24 | 2007-08-09 | Neurobiotec Gmbh | Verwendung eines transdermalen therapeutischen Systems zur Behandlung des Restless-Legs-Syndroms |
| DE10064453A1 (de) * | 2000-12-16 | 2002-07-04 | Schering Ag | Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen |
| DE60238756D1 (de) | 2001-05-11 | 2011-02-10 | Endo Pharmaceuticals Inc | Opioid enthaltende arzneiform gegen missbrauch |
| EP1492506B2 (fr) * | 2002-04-05 | 2016-06-29 | Euro-Celtique S.A. | Matrice pour liberation prolongee, constante et independante de composes actifs |
| US20050079217A1 (en) * | 2002-07-25 | 2005-04-14 | Ganorkar Loksidh D. | Sustained-release tablet composition comprising a dopamine receptor agonist |
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| ES2579853T3 (es) * | 2010-09-20 | 2016-08-17 | A.Carlsson Research Ab | Compuestos de fenilpiperidina para el tratamiento de demencia |
| EP2950799B1 (fr) | 2013-01-30 | 2019-12-04 | Pharmorx Therapeutics, Inc. | Traitement de la dépression et autres maladies avec un agent à faible dose |
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| EP3337564A4 (fr) | 2015-08-21 | 2019-01-23 | Portola Pharmaceuticals, Inc. | Composition et procédés d'utilisation de petites molécules de type tétrahydroisoquinoline pour se lier à pcsk9 et moduler l'activité protéique de pcsk9 |
| EP3337788A4 (fr) | 2015-08-21 | 2019-03-27 | Portola Pharmaceuticals, Inc. | Modulateurs phénylpipérazine proprotéine convertase subtilisine/kexine de type 9 (pcsk9) et leur utilisation |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5273975A (en) | 1989-06-09 | 1993-12-28 | The Upjohn Company | Heterocyclic amines having central nervous system activity |
| EP0641320B1 (fr) | 1991-04-17 | 2001-05-30 | PHARMACIA & UPJOHN COMPANY | Derives de (s)-3-phenylpiperidine substitues, leur preparation et leur utilisation comme dopamine autorecepteur antagonistes |
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| US6001861A (en) | 1998-01-16 | 1999-12-14 | Pharmacia & Upjohn Company | Use of pramipexole in the treatment of restless legs syndrome |
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| SE9802546D0 (sv) * | 1998-07-15 | 1998-07-15 | Ross Nicholas Waters | Medicinal product and method for treatment and prevention of dyskinesia |
| US6455564B1 (en) * | 1999-01-06 | 2002-09-24 | Pharmacia & Upjohn Company | Method of treating sexual disturbances |
| DE19938823A1 (de) * | 1999-08-19 | 2001-02-22 | Boehringer Ingelheim Pharma | Medikamentöse Behandlung des Restless Leg Syndroms |
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| AR033520A1 (es) * | 2000-04-27 | 2003-12-26 | Upjohn Co | (5r)-(metilamino) -5,6-dihidro-4h-imidazo[4,5,1-ij] quinolin-2(1h)-tiona |
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- 2001-10-24 PE PE2001001052A patent/PE20020514A1/es not_active Application Discontinuation
- 2001-10-29 CN CNA018156134A patent/CN1606442A/zh active Pending
- 2001-10-29 EP EP01979241A patent/EP1330248A2/fr not_active Withdrawn
- 2001-10-29 KR KR10-2003-7005874A patent/KR20030042037A/ko not_active Application Discontinuation
- 2001-10-29 NZ NZ52557401A patent/NZ525574A/xx unknown
- 2001-10-29 BR BR0115071-5A patent/BR0115071A/pt not_active IP Right Cessation
- 2001-10-29 JP JP2002538934A patent/JP2004512367A/ja not_active Withdrawn
- 2001-10-29 IL IL15559101A patent/IL155591A0/xx unknown
- 2001-10-29 US US10/039,446 patent/US6602868B2/en not_active Expired - Fee Related
- 2001-10-29 CA CA002421705A patent/CA2421705A1/fr not_active Abandoned
- 2001-10-29 AU AU2002211226A patent/AU2002211226A1/en not_active Abandoned
- 2001-10-29 EA EA200300527A patent/EA200300527A1/ru unknown
- 2001-10-29 PL PL36090401A patent/PL360904A1/xx not_active Application Discontinuation
- 2001-10-29 MX MXPA03003912A patent/MXPA03003912A/es not_active Application Discontinuation
- 2001-10-29 WO PCT/US2001/027785 patent/WO2002036123A2/fr not_active Application Discontinuation
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2003
- 2003-03-06 ZA ZA200301865A patent/ZA200301865B/en unknown
- 2003-04-25 US US10/423,078 patent/US6716854B2/en not_active Expired - Fee Related
- 2003-04-29 NO NO20031923A patent/NO20031923L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ525574A (en) | 2004-12-24 |
| BR0115071A (pt) | 2003-07-29 |
| PL360904A1 (en) | 2004-09-20 |
| KR20030042037A (ko) | 2003-05-27 |
| EP1330248A2 (fr) | 2003-07-30 |
| IL155591A0 (en) | 2003-11-23 |
| US6602868B2 (en) | 2003-08-05 |
| NO20031923L (no) | 2003-06-27 |
| JP2004512367A (ja) | 2004-04-22 |
| NO20031923D0 (no) | 2003-04-29 |
| PE20020514A1 (es) | 2002-06-12 |
| US20030212065A1 (en) | 2003-11-13 |
| AR031152A1 (es) | 2003-09-10 |
| AU2002211226A1 (en) | 2002-05-15 |
| MXPA03003912A (es) | 2004-09-10 |
| US20020107257A1 (en) | 2002-08-08 |
| WO2002036123A2 (fr) | 2002-05-10 |
| CA2421705A1 (fr) | 2002-05-10 |
| CN1606442A (zh) | 2005-04-13 |
| US6716854B2 (en) | 2004-04-06 |
| WO2002036123A3 (fr) | 2002-09-19 |
| EA200300527A1 (ru) | 2003-08-28 |
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