ZA200110470B - Aspartate deribative of amlodipine. - Google Patents

Aspartate deribative of amlodipine.

Info

Publication number
ZA200110470B
ZA200110470B ZA200110470A ZA200110470A ZA200110470B ZA 200110470 B ZA200110470 B ZA 200110470B ZA 200110470 A ZA200110470 A ZA 200110470A ZA 200110470 A ZA200110470 A ZA 200110470A ZA 200110470 B ZA200110470 B ZA 200110470B
Authority
ZA
South Africa
Prior art keywords
deribative
amlodipine
aspartate
aspartate deribative
Prior art date
Application number
ZA200110470A
Other languages
English (en)
Inventor
Jacobus Maria Lemmens
Theodorus Hendricus Ant Peters
Franciscus Bernardus Benneker
Original Assignee
Bioorg Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29740328&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200110470(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bioorg Bv filed Critical Bioorg Bv
Publication of ZA200110470B publication Critical patent/ZA200110470B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/90—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having more than three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ZA200110470A 2000-12-29 2001-12-20 Aspartate deribative of amlodipine. ZA200110470B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25860200P 2000-12-29 2000-12-29
US80934901A 2001-03-16 2001-03-16
BE2001/0712A BE1014455A6 (nl) 2000-12-29 2001-11-05 Aspartaatderivaat van amlodipine.

Publications (1)

Publication Number Publication Date
ZA200110470B true ZA200110470B (en) 2002-07-11

Family

ID=29740328

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200110470A ZA200110470B (en) 2000-12-29 2001-12-20 Aspartate deribative of amlodipine.

Country Status (14)

Country Link
US (1) US6479525B2 (fr)
EP (1) EP1309558A1 (fr)
BE (1) BE1014455A6 (fr)
BR (1) BR0116553A (fr)
CA (2) CA2433191A1 (fr)
CR (1) CR7011A (fr)
DE (1) DE20116170U1 (fr)
GB (1) GB2372036B (fr)
GR (1) GR1004124B (fr)
HU (1) HUP0105456A3 (fr)
IE (1) IES20011105A2 (fr)
MX (1) MXPA03005886A (fr)
WO (1) WO2002053540A1 (fr)
ZA (1) ZA200110470B (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2287110T3 (es) * 2000-04-11 2007-12-16 Sankyo Company, Limited Composicion farmaceutica estabilizada que contiene un bloqueador de calcio consistente en azelnidipina.
MXPA03005882A (es) * 2000-12-29 2005-04-19 Pfizer Ltd Derivado amida de amlodipina.
EP1309554A1 (fr) * 2000-12-29 2003-05-14 Synthon Licensing, Ltd. Derive d'amide d'amlodipine
US6653481B2 (en) * 2000-12-29 2003-11-25 Synthon Bv Process for making amlodipine
BR0116557A (pt) * 2000-12-29 2003-10-28 Pfizer Ltd Processo, processo para fabricação de um sal de maleato de amlodipina substancialmente livre de aspartato de amlodipina, processo para purificação, maleato de amlodipina, composição farmacêutica para tratar ou prevenir angina ou hipertenção, método para tratar hipertenção, angina ou ataque cardìaco, benzeno sulfonato de amlodipina, hidrocloreto de amlodipina e uso de maleato de amlodipina substancialmente livre de aspartato de amlodipina
KR100467669B1 (ko) * 2002-08-21 2005-01-24 씨제이 주식회사 암로디핀의 유기산염
TW200736245A (en) * 2005-11-29 2007-10-01 Sankyo Co Acid addition salts of optically active dihydropyridine derivatives
TW200806648A (en) * 2005-11-29 2008-02-01 Sankyo Co Acid addition salts of dihydropyridine derivatives
ES2886067T3 (es) 2016-10-07 2021-12-16 Silvergate Pharmaceuticals Inc Formulaciones de amlodipina
EP3773574A4 (fr) 2018-04-11 2022-03-02 Silvergate Pharmaceuticals, Inc. Formulations d'amlodipine

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK161312C (da) * 1982-03-11 1991-12-09 Pfizer Analogifremgangsmaade til fremstilling af 2-aminoalkoxymethyl-4-phenyl-6-methyl-1,4-dihydropyridin-3,5-dicarboxylsyreestere eller syreadditionssalte deraf samt phthalimidoderivater til anvendelse som udgangsmateriale ved fremgangsmaaden
GB8608335D0 (en) 1986-04-04 1986-05-08 Pfizer Ltd Pharmaceutically acceptable salts
US4983740A (en) 1986-08-04 1991-01-08 Adir Et Compagnie Process for 1,4-dihydropyridine compounds
GB8710493D0 (en) 1987-05-02 1987-06-03 Pfizer Ltd Dihydropyridines
US5155120A (en) 1991-01-14 1992-10-13 Pfizer Inc Method for treating congestive heart failure
WO1993006082A1 (fr) 1991-09-13 1993-04-01 Merck & Co., Inc. Procede de preparation de 1,4-dihyropyridines-4-substitues
US5389654A (en) 1992-11-26 1995-02-14 Lek, Tovarna, Farmacevtskih In Kemicnih . . . 3-ethyl 5-methyl(±)2-[2-(N-tritylamino)ethoxymethyl]-4-(2-chlorophenyl)-1,4-dihydro-6-methyl-6-methyl-3,5-pyridinedicarboxylate
HU221810B1 (hu) 1997-08-12 2003-01-28 EGIS Gyógyszergyár Rt. Eljárás amlodipin-bezilát előállítására és az eljárás intermedierjei
ZA9810320B (en) 1997-11-14 2000-05-11 Gea Farmaceutisk Fabrik As Process for the preparation of 1,4-dihydropyridines and novel compounds of use for such purpose.
PL189666B1 (pl) 1998-04-09 2005-09-30 Adamed Sp Z Oo Sposób otrzymywania benzenosulfonianu amlodypiny
GB9812413D0 (en) 1998-06-10 1998-08-05 Glaxo Group Ltd Compound and its use
ES2151850B1 (es) 1998-10-26 2001-08-16 Esteve Quimica Sa Intermedio para la sintesis de amlodipino para su obtencion y utilizacion correspondiente.
GB9827387D0 (en) 1998-12-11 1999-02-03 Smithkline Beecham Plc Novel process
GB9827431D0 (en) 1998-12-11 1999-02-03 Smithkline Beecham Plc Novel compound
GB2371862B (en) 2000-12-29 2004-07-14 Bioorg Bv Reference standards for determining the purity or stability of amlodipine maleate and processes therefor
AT5874U1 (de) * 2000-12-29 2003-01-27 Bioorg Bv Pharmazeutische zubereitungen enthaltend amlodipinmaleat
BR0116557A (pt) * 2000-12-29 2003-10-28 Pfizer Ltd Processo, processo para fabricação de um sal de maleato de amlodipina substancialmente livre de aspartato de amlodipina, processo para purificação, maleato de amlodipina, composição farmacêutica para tratar ou prevenir angina ou hipertenção, método para tratar hipertenção, angina ou ataque cardìaco, benzeno sulfonato de amlodipina, hidrocloreto de amlodipina e uso de maleato de amlodipina substancialmente livre de aspartato de amlodipina
GB0114709D0 (en) 2001-06-15 2001-08-08 Pfizer Ltd Stabilised formulations of amlodipine maleate

Also Published As

Publication number Publication date
DE20116170U1 (de) 2002-04-04
GR20010100602A (el) 2002-10-09
BR0116553A (pt) 2004-02-03
GB2372036B (en) 2004-05-19
WO2002053540A1 (fr) 2002-07-11
HUP0105456A2 (en) 2002-10-28
CA2433191A1 (fr) 2002-07-11
GR1004124B (el) 2003-01-24
CA2366391C (fr) 2005-10-18
MXPA03005886A (es) 2005-04-19
CA2366391A1 (fr) 2002-06-29
GB2372036A (en) 2002-08-14
BE1014455A6 (nl) 2003-10-07
US6479525B2 (en) 2002-11-12
CR7011A (es) 2004-03-10
GB0131064D0 (en) 2002-02-13
HU0105456D0 (en) 2002-02-28
EP1309558A1 (fr) 2003-05-14
IES20011105A2 (en) 2002-12-30
HUP0105456A3 (en) 2004-01-28
US20020128296A1 (en) 2002-09-12

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