YU92103A - Granulirani preparati gaboksadola - Google Patents

Granulirani preparati gaboksadola

Info

Publication number
YU92103A
YU92103A YU92103A YUP92103A YU92103A YU 92103 A YU92103 A YU 92103A YU 92103 A YU92103 A YU 92103A YU P92103 A YUP92103 A YU P92103A YU 92103 A YU92103 A YU 92103A
Authority
YU
Yugoslavia
Prior art keywords
gaboxadol
granular preparations
preparation
granular
dosage forms
Prior art date
Application number
YU92103A
Other languages
English (en)
Inventor
Michiel Onne Elema
Lene Andresen
Per Holm
Original Assignee
H. Lundbeck A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S
Publication of YU92103A publication Critical patent/YU92103A/sh

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Sadašnji pronalazak se odnosi na granulirani proizvod koji sadrži gaboksadol kao kiselu adicionu so, postupak granulacije topljenjem za njegovo pripremanje, i na čvrste farmaceutski jedinične oblike doze pripremljene iz navedenog granuliranog preparata gaboksadola.[The present invention relates to a granulated product containing gaboxadol as an acid addition salt, a melt granulation process for the preparation thereof and to solid pharmaceutical unit dosage forms prepared from said granular preparation of gaboxadol.
YU92103A 2001-05-21 2002-05-17 Granulirani preparati gaboksadola YU92103A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DKPA200100817 2001-05-21

Publications (1)

Publication Number Publication Date
YU92103A true YU92103A (sh) 2006-05-25

Family

ID=8160520

Family Applications (1)

Application Number Title Priority Date Filing Date
YU92103A YU92103A (sh) 2001-05-21 2002-05-17 Granulirani preparati gaboksadola

Country Status (26)

Country Link
US (1) US20040157876A1 (sh)
EP (1) EP1389091A1 (sh)
JP (1) JP2004530695A (sh)
KR (1) KR20030097890A (sh)
CN (1) CN1511026A (sh)
AR (1) AR033896A1 (sh)
AU (1) AU2002338855B2 (sh)
BG (1) BG108441A (sh)
BR (1) BR0209834A (sh)
CA (1) CA2447603A1 (sh)
CZ (1) CZ20033269A3 (sh)
EA (2) EA200700703A1 (sh)
HR (1) HRP20030950A2 (sh)
HU (1) HUP0400051A2 (sh)
IL (1) IL158733A0 (sh)
IS (1) IS7020A (sh)
ME (1) MEP6308A (sh)
MX (1) MXPA03010596A (sh)
NO (1) NO20035146D0 (sh)
NZ (1) NZ547636A (sh)
PL (1) PL366541A1 (sh)
SK (1) SK15542003A3 (sh)
UA (1) UA80092C2 (sh)
WO (1) WO2002094225A1 (sh)
YU (1) YU92103A (sh)
ZA (1) ZA200308594B (sh)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2385749A1 (en) * 1999-09-28 2001-04-05 H. Lundbeck A/S Melt granulated composition and modified release dosage form prepared from said composition
PL1641456T3 (pl) 2003-06-25 2010-08-31 H Lundbeck As Gaboksadol do leczenia depresji i innych zaburzeń afektywnych
TW200528098A (en) * 2003-12-18 2005-09-01 Lundbeck & Co As H Treatment of insomnia in human patients
GB0402118D0 (en) 2004-01-30 2004-03-03 Merck Sharp & Dohme Polymorphic forms of a GABAA agonist
EP2292222A1 (en) 2005-01-28 2011-03-09 H. Lundbeck A/S Polymorphic Forms of a GABAA Agonist
EP1906953A4 (en) * 2005-04-29 2009-05-20 Lundbeck & Co As H FORMS OF ACID SALTS AND BASIC SALTS OF GABOXADOL
JP5792061B2 (ja) * 2008-05-30 2015-10-07 サイコジェニックス・インコーポレーテッドPsychogenics Inc. 神経及び精神障害の治療法
CA2732636A1 (en) * 2008-09-01 2009-05-07 H. Lundbeck A/S Pharmaceutical composition comprising gaboxadol and an inhibitor of pat1 or oat
WO2013090452A1 (en) 2011-12-12 2013-06-20 Orbis Biosciences, Inc. Sustained release particle formulations

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4315934A (en) * 1979-09-24 1982-02-16 Sandoz Ltd. Organic compounds
DE19525598C2 (de) * 1995-07-13 1997-09-25 Max Planck Gesellschaft Schlafmittel
US6649186B1 (en) * 1996-09-20 2003-11-18 Ethypharm Effervescent granules and methods for their preparation
CA2385749A1 (en) * 1999-09-28 2001-04-05 H. Lundbeck A/S Melt granulated composition and modified release dosage form prepared from said composition
US6375982B1 (en) * 2000-07-05 2002-04-23 Capricorn Pharma, Inc. Rapid-melt semi-solid compositions, methods of making same and method of using same

Also Published As

Publication number Publication date
WO2002094225A1 (en) 2002-11-28
NZ547636A (en) 2008-03-28
AR033896A1 (es) 2004-01-07
EA200301282A1 (ru) 2004-04-29
IL158733A0 (en) 2004-05-12
CA2447603A1 (en) 2002-11-28
BG108441A (en) 2005-02-28
AU2002338855B2 (en) 2007-08-16
UA80092C2 (en) 2007-08-27
PL366541A1 (en) 2005-02-07
NO20035146L (no) 2003-11-19
SK15542003A3 (sk) 2004-05-04
HUP0400051A2 (hu) 2004-04-28
CZ20033269A3 (en) 2004-03-17
US20040157876A1 (en) 2004-08-12
KR20030097890A (ko) 2003-12-31
EA009731B1 (ru) 2008-02-28
JP2004530695A (ja) 2004-10-07
CN1511026A (zh) 2004-07-07
HRP20030950A2 (en) 2005-08-31
BR0209834A (pt) 2004-06-15
EP1389091A1 (en) 2004-02-18
EA200700703A1 (ru) 2007-08-31
MEP6308A (xx) 2010-02-10
IS7020A (is) 2003-11-10
MXPA03010596A (es) 2004-03-09
ZA200308594B (en) 2004-11-04
NO20035146D0 (no) 2003-11-19

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