MXPA03010596A - Preparaciones granuladas de gaboxadol. - Google Patents

Preparaciones granuladas de gaboxadol.

Info

Publication number
MXPA03010596A
MXPA03010596A MXPA03010596A MXPA03010596A MXPA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A
Authority
MX
Mexico
Prior art keywords
gaboxadol
granular preparations
preparation
granular
dosage forms
Prior art date
Application number
MXPA03010596A
Other languages
English (en)
Inventor
Holm Per
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of MXPA03010596A publication Critical patent/MXPA03010596A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

La presente invencion se relaciona con un producto granulado que contiene gaboxadol como sal de adicion de acido, con un proceso de granulacion en fusion para la preparacion del mismo y con formas de dosificacion unitaria farmaceuticas macizas preparadas con dicha preparacion granulada de gaboxadol.
MXPA03010596A 2001-05-21 2002-05-17 Preparaciones granuladas de gaboxadol. MXPA03010596A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200100817 2001-05-21
PCT/DK2002/000332 WO2002094225A1 (en) 2001-05-21 2002-05-17 Granular preparations of gaboxadol

Publications (1)

Publication Number Publication Date
MXPA03010596A true MXPA03010596A (es) 2004-03-09

Family

ID=8160520

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03010596A MXPA03010596A (es) 2001-05-21 2002-05-17 Preparaciones granuladas de gaboxadol.

Country Status (26)

Country Link
US (1) US20040157876A1 (es)
EP (1) EP1389091A1 (es)
JP (1) JP2004530695A (es)
KR (1) KR20030097890A (es)
CN (1) CN1511026A (es)
AR (1) AR033896A1 (es)
AU (1) AU2002338855B2 (es)
BG (1) BG108441A (es)
BR (1) BR0209834A (es)
CA (1) CA2447603A1 (es)
CZ (1) CZ20033269A3 (es)
EA (2) EA009731B1 (es)
HR (1) HRP20030950A2 (es)
HU (1) HUP0400051A2 (es)
IL (1) IL158733A0 (es)
IS (1) IS7020A (es)
ME (1) MEP6308A (es)
MX (1) MXPA03010596A (es)
NO (1) NO20035146D0 (es)
NZ (1) NZ547636A (es)
PL (1) PL366541A1 (es)
SK (1) SK15542003A3 (es)
UA (1) UA80092C2 (es)
WO (1) WO2002094225A1 (es)
YU (1) YU92103A (es)
ZA (1) ZA200308594B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001022941A1 (en) * 1999-09-28 2001-04-05 H. Lundbeck A/S Melt granulated composition and modified release dosage form prepared from said composition
PT1641456E (pt) 2003-06-25 2010-06-01 Lundbeck & Co As H Gaboxadol para o tratamento de depressão e outros distúrbios afectivos
TW200528098A (en) * 2003-12-18 2005-09-01 Lundbeck & Co As H Treatment of insomnia in human patients
GB0402118D0 (en) 2004-01-30 2004-03-03 Merck Sharp & Dohme Polymorphic forms of a GABAA agonist
EP1848420A4 (en) 2005-01-28 2008-01-23 Merck & Co Inc POLYMORPHIC FORMS OF A GABAA AGONIST
EP1906953A4 (en) * 2005-04-29 2009-05-20 Lundbeck & Co As H FORMS OF ACID SALTS AND BASIC SALTS OF GABOXADOL
CA2725356C (en) * 2008-05-30 2018-10-16 Psychogenics, Inc. Use of eltoprazine for improving symptoms of cognitive impairment associated with non-adhd neurological and mental disorders
EP2334299A1 (en) * 2008-09-01 2011-06-22 H. Lundbeck A/S Pharmaceutical composition comprising gaboxadol and an inhibitor of patl or oat
CA2859174C (en) 2011-12-12 2019-03-05 Orbis Biosciences, Inc. Sustained release particle formulations

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4315934A (en) * 1979-09-24 1982-02-16 Sandoz Ltd. Organic compounds
DE19525598C2 (de) * 1995-07-13 1997-09-25 Max Planck Gesellschaft Schlafmittel
US6649186B1 (en) * 1996-09-20 2003-11-18 Ethypharm Effervescent granules and methods for their preparation
WO2001022941A1 (en) * 1999-09-28 2001-04-05 H. Lundbeck A/S Melt granulated composition and modified release dosage form prepared from said composition
US6375982B1 (en) * 2000-07-05 2002-04-23 Capricorn Pharma, Inc. Rapid-melt semi-solid compositions, methods of making same and method of using same

Also Published As

Publication number Publication date
HRP20030950A2 (en) 2005-08-31
HUP0400051A2 (hu) 2004-04-28
EA200301282A1 (ru) 2004-04-29
NO20035146L (no) 2003-11-19
CZ20033269A3 (en) 2004-03-17
IS7020A (is) 2003-11-10
NZ547636A (en) 2008-03-28
WO2002094225A1 (en) 2002-11-28
SK15542003A3 (sk) 2004-05-04
CN1511026A (zh) 2004-07-07
CA2447603A1 (en) 2002-11-28
UA80092C2 (en) 2007-08-27
EP1389091A1 (en) 2004-02-18
ZA200308594B (en) 2004-11-04
JP2004530695A (ja) 2004-10-07
IL158733A0 (en) 2004-05-12
BG108441A (en) 2005-02-28
NO20035146D0 (no) 2003-11-19
EA200700703A1 (ru) 2007-08-31
MEP6308A (xx) 2010-02-10
EA009731B1 (ru) 2008-02-28
BR0209834A (pt) 2004-06-15
AR033896A1 (es) 2004-01-07
PL366541A1 (en) 2005-02-07
YU92103A (sh) 2006-05-25
KR20030097890A (ko) 2003-12-31
US20040157876A1 (en) 2004-08-12
AU2002338855B2 (en) 2007-08-16

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Legal Events

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FA Abandonment or withdrawal