YU60790A - Postupak za dobijanje 5-fenilpirimidin jedinjenja i njihovih soli - Google Patents

Postupak za dobijanje 5-fenilpirimidin jedinjenja i njihovih soli

Info

Publication number
YU60790A
YU60790A YU60790A YU60790A YU60790A YU 60790 A YU60790 A YU 60790A YU 60790 A YU60790 A YU 60790A YU 60790 A YU60790 A YU 60790A YU 60790 A YU60790 A YU 60790A
Authority
YU
Yugoslavia
Prior art keywords
formula
preparation
compound
salts
phenylpyrimidine
Prior art date
Application number
YU60790A
Other languages
English (en)
Other versions
YU47557B (sh
Inventor
A.A Miller
M.S. Nobbs
R.M. Hyde
M.J. Leach
Original Assignee
The Wellcome Foundation Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by The Wellcome Foundation Ltd. filed Critical The Wellcome Foundation Ltd.
Priority to SI9010607A priority Critical patent/SI9010607B/sl
Publication of YU60790A publication Critical patent/YU60790A/sh
Priority to HR940540A priority patent/HRP940540B1/xx
Publication of YU47557B publication Critical patent/YU47557B/sh

Links

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

POSTUPAK ZA DOBIJANJE 5-FENILPIRIMIDIN JEDINJENJA I NJIHOVIH SOLI U prijavi je opisan postupak za pravljenje novih 5-fenilpirimidin derivata formule I: u kojoj radikali R1-R8 imaju značenja data u Zahtevu 1. U novom postupku intermedijer formule II: u kojoj su R3 do R8 kao što je definisano ranije, L je odlazeća grupa i Y je cijano ili karboksi, karbonil ili alkoksikarbonil reaguje sa jedinjenjem formule III: H2N - C - R1 gde je R1 kao što je definisano ranije. Jedinjenje formule I može se izolovati kao slobodna baza ili u obliku njene adicione soli sa kiselinom. Takodje je opisan i postupak za pravljenje preparata u kojem se novo jedinjenje formule I meša sa farmaceutski prihvatljivim sastojkom na standardni način.
YU60790A 1989-04-14 1990-03-28 Postupak za dobijanje 5-fenilpirimidin jedinjenja i njihovih soli YU47557B (sh)

Priority Applications (2)

Application Number Priority Date Filing Date Title
SI9010607A SI9010607B (sl) 1989-04-14 1990-03-28 Farmakolosko aktivne CNS spojine
HR940540A HRP940540B1 (en) 1989-04-14 1994-09-16 Pharmacologically active cns compounds

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898908561A GB8908561D0 (en) 1989-04-14 1989-04-14 Pharmaceutically active cns compounds

Publications (2)

Publication Number Publication Date
YU60790A true YU60790A (sh) 1994-04-05
YU47557B YU47557B (sh) 1995-10-03

Family

ID=10655105

Family Applications (1)

Application Number Title Priority Date Filing Date
YU60790A YU47557B (sh) 1989-04-14 1990-03-28 Postupak za dobijanje 5-fenilpirimidin jedinjenja i njihovih soli

Country Status (5)

Country Link
CZ (1) CZ287351B6 (sh)
GB (1) GB8908561D0 (sh)
HR (1) HRP940540B1 (sh)
SI (1) SI9010607B (sh)
YU (1) YU47557B (sh)

Also Published As

Publication number Publication date
HRP940540A2 (en) 1996-08-31
HRP940540B1 (en) 2000-12-31
CZ287351B6 (cs) 2000-10-11
SI9010607A (en) 1997-06-30
SI9010607B (sl) 2006-06-30
GB8908561D0 (en) 1989-06-01
YU47557B (sh) 1995-10-03

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