YU40287B - Process for obtaining antibacterial agents, unsubstituted 3-thiole-cephalosporins - Google Patents

Process for obtaining antibacterial agents, unsubstituted 3-thiole-cephalosporins

Info

Publication number
YU40287B
YU40287B YU2431/76A YU243176A YU40287B YU 40287 B YU40287 B YU 40287B YU 2431/76 A YU2431/76 A YU 2431/76A YU 243176 A YU243176 A YU 243176A YU 40287 B YU40287 B YU 40287B
Authority
YU
Yugoslavia
Prior art keywords
thiole
cephalosporins
unsubstituted
antibacterial agents
obtaining antibacterial
Prior art date
Application number
YU2431/76A
Other versions
YU243176A (en
Inventor
M A Kaplan
W Gottstein
A P Granatek
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/653,999 external-priority patent/US4026888A/en
Priority claimed from US05/654,314 external-priority patent/US4061862A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of YU243176A publication Critical patent/YU243176A/en
Publication of YU40287B publication Critical patent/YU40287B/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/58—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with a nitrogen atom, which is a member of a hetero ring, attached in position 7

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
YU2431/76A 1975-10-06 1976-10-04 Process for obtaining antibacterial agents, unsubstituted 3-thiole-cephalosporins YU40287B (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US62000575A 1975-10-06 1975-10-06
US62230675A 1975-10-10 1975-10-10
US64031775A 1975-12-12 1975-12-12
US05/653,999 US4026888A (en) 1975-10-10 1976-01-30 Certain derivatives of particular 3-thiolated cephalosporins
US05/654,314 US4061862A (en) 1975-10-06 1976-02-02 Derivatives of 7-(cyclized)phenylglycyl-3-triazolo-thio methyl cephalosporin

Publications (2)

Publication Number Publication Date
YU243176A YU243176A (en) 1982-06-30
YU40287B true YU40287B (en) 1985-12-31

Family

ID=27542000

Family Applications (1)

Application Number Title Priority Date Filing Date
YU2431/76A YU40287B (en) 1975-10-06 1976-10-04 Process for obtaining antibacterial agents, unsubstituted 3-thiole-cephalosporins

Country Status (17)

Country Link
JP (1) JPS6052718B2 (en)
AU (1) AU511344B2 (en)
BE (1) BE846890A (en)
CA (1) CA1113927A (en)
CH (1) CH629500A5 (en)
CY (1) CY1121A (en)
DE (1) DE2645144C2 (en)
DK (2) DK158673C (en)
FR (1) FR2326926A1 (en)
GB (1) GB1521419A (en)
HK (1) HK41281A (en)
IE (1) IE43666B1 (en)
KE (1) KE3154A (en)
LU (1) LU75935A1 (en)
NL (1) NL189670C (en)
SE (1) SE434952B (en)
YU (1) YU40287B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54112892A (en) * 1978-02-23 1979-09-04 Shionogi & Co Ltd Substituted imidazolidinyl-3-chloro-3-cephem-4-carboxylic acid
JPS54115354A (en) * 1978-02-27 1979-09-07 Chugai Pharmaceut Co Ltd Biphenylylglycine derivative
WO2019168164A1 (en) * 2018-03-02 2019-09-06 国立大学法人大阪大学 Molecule for protein and/or peptide design

Also Published As

Publication number Publication date
DK158673B (en) 1990-07-02
DK158673C (en) 1991-01-14
FR2326926A1 (en) 1977-05-06
DK200488A (en) 1988-04-12
IE43666L (en) 1977-04-06
FR2326926B1 (en) 1980-07-11
LU75935A1 (en) 1977-05-25
NL189670B (en) 1993-01-18
SE434952B (en) 1984-08-27
IE43666B1 (en) 1981-04-22
SE7610989L (en) 1977-04-07
KE3154A (en) 1981-09-18
DK200488D0 (en) 1988-04-12
YU243176A (en) 1982-06-30
CY1121A (en) 1981-12-04
JPS6052718B2 (en) 1985-11-20
CA1113927A (en) 1981-12-08
JPS5246094A (en) 1977-04-12
DK164225B (en) 1992-05-25
DK446576A (en) 1977-04-07
NL189670C (en) 1993-06-16
AU1824576A (en) 1978-04-06
NL7611026A (en) 1977-04-12
DE2645144A1 (en) 1977-04-14
GB1521419A (en) 1978-08-16
CH629500A5 (en) 1982-04-30
DE2645144C2 (en) 1986-11-27
HK41281A (en) 1981-08-28
DK164225C (en) 1992-10-19
BE846890A (en) 1977-04-01
AU511344B2 (en) 1980-08-14

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