AU1824576A - "7-(2-substituted-4-(4-hydroxy phenyl) -5 ketoterahydroimidazo-1-yl) - 3- substituted thiomethyl-3-cephem-4-carboxylic acid derivatives - Google Patents

"7-(2-substituted-4-(4-hydroxy phenyl) -5 ketoterahydroimidazo-1-yl) - 3- substituted thiomethyl-3-cephem-4-carboxylic acid derivatives

Info

Publication number
AU1824576A
AU1824576A AU18245/76A AU1824576A AU1824576A AU 1824576 A AU1824576 A AU 1824576A AU 18245/76 A AU18245/76 A AU 18245/76A AU 1824576 A AU1824576 A AU 1824576A AU 1824576 A AU1824576 A AU 1824576A
Authority
AU
Australia
Prior art keywords
substituted
ketoterahydroimidazo
cephem
carboxylic acid
acid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU18245/76A
Other versions
AU511344B2 (en
Inventor
Murray Arthur Kaplan
William J Gottstein
Alphonse Peter Granatek
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/653,999 external-priority patent/US4026888A/en
Priority claimed from US05/654,314 external-priority patent/US4061862A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of AU1824576A publication Critical patent/AU1824576A/en
Application granted granted Critical
Publication of AU511344B2 publication Critical patent/AU511344B2/en
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/58—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with a nitrogen atom, which is a member of a hetero ring, attached in position 7
AU18245/76A 1975-10-06 1976-09-30 "7-(2-substituted-4-(4-hydroxy phenyl) -5 ketoterahydroimidazo-1-yl) - 3- substituted thiomethyl-3-cephem-4-carboxylic acid derivatives Expired AU511344B2 (en)

Applications Claiming Priority (10)

Application Number Priority Date Filing Date Title
US62000575A 1975-10-06 1975-10-06
USUS620005 1975-10-06
US62230675A 1975-10-10 1975-10-10
USUS622,306 1975-10-10
US64031775A 1975-12-12 1975-12-12
USUS640,317 1975-12-12
USUS653,999 1976-01-30
US05/653,999 US4026888A (en) 1975-10-10 1976-01-30 Certain derivatives of particular 3-thiolated cephalosporins
US05/654,314 US4061862A (en) 1975-10-06 1976-02-02 Derivatives of 7-(cyclized)phenylglycyl-3-triazolo-thio methyl cephalosporin
USUS654,314 1976-02-02

Publications (2)

Publication Number Publication Date
AU1824576A true AU1824576A (en) 1978-04-06
AU511344B2 AU511344B2 (en) 1980-08-14

Family

ID=27542000

Family Applications (1)

Application Number Title Priority Date Filing Date
AU18245/76A Expired AU511344B2 (en) 1975-10-06 1976-09-30 "7-(2-substituted-4-(4-hydroxy phenyl) -5 ketoterahydroimidazo-1-yl) - 3- substituted thiomethyl-3-cephem-4-carboxylic acid derivatives

Country Status (17)

Country Link
JP (1) JPS6052718B2 (en)
AU (1) AU511344B2 (en)
BE (1) BE846890A (en)
CA (1) CA1113927A (en)
CH (1) CH629500A5 (en)
CY (1) CY1121A (en)
DE (1) DE2645144C2 (en)
DK (2) DK158673C (en)
FR (1) FR2326926A1 (en)
GB (1) GB1521419A (en)
HK (1) HK41281A (en)
IE (1) IE43666B1 (en)
KE (1) KE3154A (en)
LU (1) LU75935A1 (en)
NL (1) NL189670C (en)
SE (1) SE434952B (en)
YU (1) YU40287B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54112892A (en) * 1978-02-23 1979-09-04 Shionogi & Co Ltd Substituted imidazolidinyl-3-chloro-3-cephem-4-carboxylic acid
JPS54115354A (en) * 1978-02-27 1979-09-07 Chugai Pharmaceut Co Ltd Biphenylylglycine derivative
WO2019168164A1 (en) * 2018-03-02 2019-09-06 国立大学法人大阪大学 Molecule for protein and/or peptide design

Also Published As

Publication number Publication date
DK158673B (en) 1990-07-02
DK158673C (en) 1991-01-14
FR2326926A1 (en) 1977-05-06
DK200488A (en) 1988-04-12
IE43666L (en) 1977-04-06
FR2326926B1 (en) 1980-07-11
LU75935A1 (en) 1977-05-25
NL189670B (en) 1993-01-18
SE434952B (en) 1984-08-27
IE43666B1 (en) 1981-04-22
SE7610989L (en) 1977-04-07
KE3154A (en) 1981-09-18
DK200488D0 (en) 1988-04-12
YU243176A (en) 1982-06-30
YU40287B (en) 1985-12-31
CY1121A (en) 1981-12-04
JPS6052718B2 (en) 1985-11-20
CA1113927A (en) 1981-12-08
JPS5246094A (en) 1977-04-12
DK164225B (en) 1992-05-25
DK446576A (en) 1977-04-07
NL189670C (en) 1993-06-16
NL7611026A (en) 1977-04-12
DE2645144A1 (en) 1977-04-14
GB1521419A (en) 1978-08-16
CH629500A5 (en) 1982-04-30
DE2645144C2 (en) 1986-11-27
HK41281A (en) 1981-08-28
DK164225C (en) 1992-10-19
BE846890A (en) 1977-04-01
AU511344B2 (en) 1980-08-14

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