YU33390B - Postupak za izradu n-oksida benzilpirimidina - Google Patents

Postupak za izradu n-oksida benzilpirimidina

Info

Publication number
YU33390B
YU33390B YU01328/70A YU132870A YU33390B YU 33390 B YU33390 B YU 33390B YU 01328/70 A YU01328/70 A YU 01328/70A YU 132870 A YU132870 A YU 132870A YU 33390 B YU33390 B YU 33390B
Authority
YU
Yugoslavia
Prior art keywords
oksida
izradu
benzilpirimidina
postupak
oksida benzilpirimidina
Prior art date
Application number
YU01328/70A
Other languages
English (en)
Other versions
YU132870A (en
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of YU132870A publication Critical patent/YU132870A/xx
Publication of YU33390B publication Critical patent/YU33390B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Structures Of Non-Positive Displacement Pumps (AREA)
YU01328/70A 1969-06-12 1970-05-25 Postupak za izradu n-oksida benzilpirimidina YU33390B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH897069A CH513181A (de) 1969-06-12 1969-06-12 Verfahren zur Herstellung von N-Oxyden von Benzylpyrimidinen

Publications (2)

Publication Number Publication Date
YU132870A YU132870A (en) 1976-06-30
YU33390B true YU33390B (en) 1976-12-31

Family

ID=4346865

Family Applications (1)

Application Number Title Priority Date Filing Date
YU01328/70A YU33390B (en) 1969-06-12 1970-05-25 Postupak za izradu n-oksida benzilpirimidina

Country Status (18)

Country Link
US (1) US3715357A (de)
AT (1) AT294843B (de)
BE (1) BE751790A (de)
BR (1) BR6915095D0 (de)
CA (1) CA955944A (de)
CH (1) CH513181A (de)
DE (1) DE2026997A1 (de)
DK (1) DK124682B (de)
ES (1) ES380642A1 (de)
FR (1) FR2052954B1 (de)
GB (1) GB1256849A (de)
IE (1) IE34683B1 (de)
IL (1) IL34632A (de)
NL (1) NL7008610A (de)
NO (1) NO127237B (de)
SE (1) SE367412B (de)
YU (1) YU33390B (de)
ZA (1) ZA703569B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3993761A (en) * 1971-12-01 1976-11-23 Hoffmann-La Roche Inc. Antibacterial compositions
BE792096A (fr) * 1971-12-01 1973-05-30 Hoffmann La Roche Nouvelles benzylpyrimidines
AR204082A1 (es) * 1972-06-26 1975-11-20 Hoffmann La Roche Procedimiento para preparar derivados de n-oxidos de 2,4-diamino-5-(3-metoxi-4,5-metilendioxibencil)pirimidina
US4515948A (en) * 1973-09-12 1985-05-07 Hoffmann-La Roche Inc. 2,4-Diamino-5-(4-amino and 4-dimethylamino-3,5-dimethoxy benzyl)pyrimidines
US4076810A (en) * 1973-11-08 1978-02-28 Hoffmann-La Roche Inc. Benzylpyrimidine antibacterial composition
CH591457A5 (de) * 1973-11-08 1977-09-15 Hoffmann La Roche
WO2003043979A2 (en) * 2001-11-20 2003-05-30 Dana Farber Cancer Institute Pharmaceutically active compounds and methods of use thereof
DK1725540T5 (da) 2004-03-05 2012-10-22 Hoffmann La Roche Diaminopyrimidiner som p2x3- og p2x2/3-antagonister
EP1924566B1 (de) * 2005-09-01 2016-01-13 F.Hoffmann-La Roche Ag Diaminopyrimidine als p2x3- und p3x2/3-modulatoren
CA2619919C (en) * 2005-09-01 2014-04-01 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
CN101253159B (zh) * 2005-09-01 2011-12-07 弗·哈夫曼-拉罗切有限公司 作为p2x3和p2x2/3调节剂的二氨基嘧啶类化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2518130A (en) * 1945-04-26 1950-08-08 Evans N-oxides of tertiary amines and process of preparing same
US2500131A (en) * 1945-06-27 1950-03-07 Ralph L Evans Di-nu-oxides of amino-substituted acridines and quinolines
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
FR1453056A (fr) * 1964-11-12 1966-04-15 Hoffmann La Roche Procédé pour la préparation de dérivés de pyrimidine
US3485840A (en) * 1964-11-12 1969-12-23 Hoffmann La Roche 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes
US3461461A (en) * 1965-11-01 1969-08-12 Upjohn Co 6-amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidines
US3464987A (en) * 1966-02-21 1969-09-02 Upjohn Co 1,2-dihydro-1-hydroxy-2-imino-6-(lower alkyl)pyrimidines

Also Published As

Publication number Publication date
CH513181A (de) 1971-09-30
BR6915095D0 (pt) 1973-03-08
IL34632A0 (en) 1970-08-19
ES380642A1 (es) 1972-10-16
YU132870A (en) 1976-06-30
SE367412B (de) 1974-05-27
NL7008610A (de) 1970-12-15
AT294843B (de) 1971-12-10
FR2052954A1 (de) 1971-04-16
ZA703569B (en) 1971-01-27
GB1256849A (de) 1971-12-15
CA955944A (en) 1974-10-08
BE751790A (fr) 1970-12-11
FR2052954B1 (de) 1973-08-10
US3715357A (en) 1973-02-06
IL34632A (en) 1973-08-29
NO127237B (de) 1973-05-28
DK124682B (da) 1972-11-13
DE2026997A1 (de) 1970-12-23
IE34683L (en) 1970-12-12
IE34683B1 (en) 1975-07-23

Similar Documents

Publication Publication Date Title
YU19170A (en) Spremiste za nozice za brijanje
YU213370A (en) Postupa za kataliticko dehidrogenovanje ugjovodnika
YU125469A (en) Postupak za dobivanje tiadiazol proizvoda
YU20070A (en) Priprava za tesnjenje rotirajoce gredi
YU127170A (en) Pokretna masina za utiskivanje zastora koloseka
YU33390B (en) Postupak za izradu n-oksida benzilpirimidina
YU123869A (en) Rezna glava za profiliranje okruglih drvenih trupaca
YU135070A (en) Okvir za tro- ili viseosovna obrtna postolja sinskih vozila
YU204070A (en) Mrezica aparata za suvo brijanje
YU214170A (en) Rotaciona vakuum-masina za kalupovanje termoplasticne odnosno penoplasticne folije
YU141370A (en) Sprednja celjust za varnostne smucarske vezi
YU162470A (en) Postupak za dobijanje cistog p-ksilola
YU157270A (en) Uredaj za upravljanje vozila
YU168070A (en) Okvir za zidno odprtino
YU126570A (en) Postupak za dobijanje novih derivata benzofurana
YU159270A (en) Hidraulicni uredaj za kocenje
YU195870A (en) Razdovojiva frikciona spojnica za vozila
YU198670A (en) Klatna spona za vesanje gibnjeva
YU189270A (en) Uredaj za mesanje stocne hrane
YU143270A (en) Postopek za propravo nizkoogljicnih jekel
YU134870A (en) Postopek za pripravo termoplasticnih polimernih sestavkov
YU12470A (en) Priprava za izdelavo toplotnega izmenjalnika
YU146070A (en) Srednja celjust za varnostne smucarske vezi
YU172169A (en) Postopek za pripravo derivatov imidazola
YU148969A (en) Priprava za funkcionalno elektricno stimulacijo ekstremitete