BR6915095D0 - Processo para a preparacao de n-oxidos de benzilpirimidinas - Google Patents

Processo para a preparacao de n-oxidos de benzilpirimidinas

Info

Publication number
BR6915095D0
BR6915095D0 BR215095/69A BR21509569A BR6915095D0 BR 6915095 D0 BR6915095 D0 BR 6915095D0 BR 215095/69 A BR215095/69 A BR 215095/69A BR 21509569 A BR21509569 A BR 21509569A BR 6915095 D0 BR6915095 D0 BR 6915095D0
Authority
BR
Brazil
Prior art keywords
benzylpyrimidines
oxides
preparation
Prior art date
Application number
BR215095/69A
Other languages
English (en)
Inventor
Bellet G Rey
D Schwartz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR6915095D0 publication Critical patent/BR6915095D0/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Structures Of Non-Positive Displacement Pumps (AREA)
BR215095/69A 1969-06-12 1969-12-15 Processo para a preparacao de n-oxidos de benzilpirimidinas BR6915095D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH897069A CH513181A (de) 1969-06-12 1969-06-12 Verfahren zur Herstellung von N-Oxyden von Benzylpyrimidinen

Publications (1)

Publication Number Publication Date
BR6915095D0 true BR6915095D0 (pt) 1973-03-08

Family

ID=4346865

Family Applications (1)

Application Number Title Priority Date Filing Date
BR215095/69A BR6915095D0 (pt) 1969-06-12 1969-12-15 Processo para a preparacao de n-oxidos de benzilpirimidinas

Country Status (18)

Country Link
US (1) US3715357A (pt)
AT (1) AT294843B (pt)
BE (1) BE751790A (pt)
BR (1) BR6915095D0 (pt)
CA (1) CA955944A (pt)
CH (1) CH513181A (pt)
DE (1) DE2026997A1 (pt)
DK (1) DK124682B (pt)
ES (1) ES380642A1 (pt)
FR (1) FR2052954B1 (pt)
GB (1) GB1256849A (pt)
IE (1) IE34683B1 (pt)
IL (1) IL34632A (pt)
NL (1) NL7008610A (pt)
NO (1) NO127237B (pt)
SE (1) SE367412B (pt)
YU (1) YU33390B (pt)
ZA (1) ZA703569B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE792096A (fr) * 1971-12-01 1973-05-30 Hoffmann La Roche Nouvelles benzylpyrimidines
US3993761A (en) * 1971-12-01 1976-11-23 Hoffmann-La Roche Inc. Antibacterial compositions
AR204082A1 (es) * 1972-06-26 1975-11-20 Hoffmann La Roche Procedimiento para preparar derivados de n-oxidos de 2,4-diamino-5-(3-metoxi-4,5-metilendioxibencil)pirimidina
US4515948A (en) * 1973-09-12 1985-05-07 Hoffmann-La Roche Inc. 2,4-Diamino-5-(4-amino and 4-dimethylamino-3,5-dimethoxy benzyl)pyrimidines
US4076810A (en) * 1973-11-08 1978-02-28 Hoffmann-La Roche Inc. Benzylpyrimidine antibacterial composition
CH591457A5 (pt) * 1973-11-08 1977-09-15 Hoffmann La Roche
WO2003043979A2 (en) * 2001-11-20 2003-05-30 Dana Farber Cancer Institute Pharmaceutically active compounds and methods of use thereof
ES2391636T3 (es) * 2004-03-05 2012-11-28 F. Hoffmann-La Roche Ag Diaminopirimidinas como antagonistas de P2X3 y P2X2/3
CA2620129C (en) * 2005-09-01 2014-12-23 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
ES2601178T3 (es) * 2005-09-01 2017-02-14 F. Hoffmann-La Roche Ag Diaminopirimidinas como moduladores de P2X3 y P3X2/3
CA2619919C (en) * 2005-09-01 2014-04-01 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2518130A (en) * 1945-04-26 1950-08-08 Evans N-oxides of tertiary amines and process of preparing same
US2500131A (en) * 1945-06-27 1950-03-07 Ralph L Evans Di-nu-oxides of amino-substituted acridines and quinolines
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
US3485840A (en) * 1964-11-12 1969-12-23 Hoffmann La Roche 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes
FR1453056A (fr) * 1964-11-12 1966-04-15 Hoffmann La Roche Procédé pour la préparation de dérivés de pyrimidine
US3382247A (en) * 1965-11-01 1968-05-07 Upjohn Co 6-amino-1, 2-dihydro-1-hydroxy-2-imino-4-phenoxypyrimidines
US3464987A (en) * 1966-02-21 1969-09-02 Upjohn Co 1,2-dihydro-1-hydroxy-2-imino-6-(lower alkyl)pyrimidines

Also Published As

Publication number Publication date
SE367412B (pt) 1974-05-27
CH513181A (de) 1971-09-30
YU33390B (en) 1976-12-31
FR2052954A1 (pt) 1971-04-16
ES380642A1 (es) 1972-10-16
IL34632A (en) 1973-08-29
AT294843B (de) 1971-12-10
DE2026997A1 (pt) 1970-12-23
GB1256849A (pt) 1971-12-15
FR2052954B1 (pt) 1973-08-10
ZA703569B (en) 1971-01-27
CA955944A (en) 1974-10-08
US3715357A (en) 1973-02-06
NO127237B (pt) 1973-05-28
IE34683B1 (en) 1975-07-23
YU132870A (en) 1976-06-30
BE751790A (fr) 1970-12-11
IL34632A0 (en) 1970-08-19
IE34683L (en) 1970-12-12
NL7008610A (pt) 1970-12-15
DK124682B (da) 1972-11-13

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