YU2397A - 2-phenyl-3-aroylbenzothiophenes using for medicaments obtaining - Google Patents
2-phenyl-3-aroylbenzothiophenes using for medicaments obtainingInfo
- Publication number
- YU2397A YU2397A YU2397A YU2397A YU2397A YU 2397 A YU2397 A YU 2397A YU 2397 A YU2397 A YU 2397A YU 2397 A YU2397 A YU 2397A YU 2397 A YU2397 A YU 2397A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- phenyl
- aroylbenzothiophenes
- medicaments
- obtaining
- hexamethyleneimino
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4535—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
Opisana je upotreba jedinjenja formule I u kojoj su R1 i R3 nezavisno vodonik, -CH3, -C(=O)-(C1-C6 alkil), ili -C(O=)- Ar, gde je Ar opciono supstituisan fenil; R2 je izabran od grupe koja sadrži pirolidin, heksametilenimino i piperidino; ili farmaceutski prihvatljive soli i njihove rastvore; za dobijanje medikamenta upotrebljivog za inhibiciju kancera debelog creva.Described is the use of a compound of formula I wherein R 1 and R 3 are independently hydrogen, -CH 3, -C (= O) - (C 1 -C 6 alkyl), or -C (O =) - Ar, wherein Ar is optionally substituted phenyl; R2 is selected from the group consisting of pyrrolidine, hexamethyleneimino and piperidino; or pharmaceutically acceptable salts and solutions thereof; to obtain a medicament useful for the inhibition of colon cancer.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1077296P | 1996-01-29 | 1996-01-29 | |
| GBGB9603150.5A GB9603150D0 (en) | 1996-02-15 | 1996-02-15 | Methods of inhibiting colon tumors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| YU2397A true YU2397A (en) | 1999-11-22 |
Family
ID=26308709
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU2397A YU2397A (en) | 1996-01-29 | 1997-01-24 | 2-phenyl-3-aroylbenzothiophenes using for medicaments obtaining |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP0921799A4 (en) |
| JP (1) | JP2000503994A (en) |
| KR (1) | KR19990082054A (en) |
| CN (1) | CN1209745A (en) |
| AR (1) | AR010978A1 (en) |
| AU (1) | AU707892B2 (en) |
| BR (1) | BR9700778A (en) |
| CO (1) | CO4761062A1 (en) |
| CZ (1) | CZ235498A3 (en) |
| EA (1) | EA001104B1 (en) |
| ID (1) | ID15917A (en) |
| IL (1) | IL125521A (en) |
| MX (1) | MX9806036A (en) |
| NO (1) | NO983451L (en) |
| NZ (1) | NZ331105A (en) |
| PL (1) | PL328147A1 (en) |
| TW (1) | TW446560B (en) |
| WO (1) | WO1997026877A1 (en) |
| YU (1) | YU2397A (en) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW366342B (en) * | 1992-07-28 | 1999-08-11 | Lilly Co Eli | The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss |
| IL111287A0 (en) * | 1993-10-15 | 1994-12-29 | Lilly Co Eli | Methods for treating resistant neoplasms |
| US5574047A (en) * | 1993-12-21 | 1996-11-12 | Eli Lilly And Company | Methods of inhibiting imperfect tissue repair |
-
1997
- 1997-01-22 ID IDP970182A patent/ID15917A/en unknown
- 1997-01-24 YU YU2397A patent/YU2397A/en unknown
- 1997-01-24 AR ARP970100300A patent/AR010978A1/en unknown
- 1997-01-25 TW TW086100832A patent/TW446560B/en not_active IP Right Cessation
- 1997-01-27 BR BR9700778A patent/BR9700778A/en active Search and Examination
- 1997-01-27 WO PCT/US1997/002286 patent/WO1997026877A1/en not_active Application Discontinuation
- 1997-01-27 EA EA199800677A patent/EA001104B1/en not_active IP Right Cessation
- 1997-01-27 NZ NZ331105A patent/NZ331105A/en unknown
- 1997-01-27 KR KR1019980705775A patent/KR19990082054A/en not_active Application Discontinuation
- 1997-01-27 IL IL12552197A patent/IL125521A/en not_active IP Right Cessation
- 1997-01-27 EP EP97906587A patent/EP0921799A4/en not_active Withdrawn
- 1997-01-27 PL PL97328147A patent/PL328147A1/en unknown
- 1997-01-27 JP JP9527132A patent/JP2000503994A/en active Pending
- 1997-01-27 CN CN97191791A patent/CN1209745A/en active Pending
- 1997-01-27 CZ CZ982354A patent/CZ235498A3/en unknown
- 1997-01-27 AU AU21239/97A patent/AU707892B2/en not_active Ceased
- 1997-01-28 CO CO97003856A patent/CO4761062A1/en unknown
-
1998
- 1998-07-27 MX MX9806036A patent/MX9806036A/en unknown
- 1998-07-27 NO NO983451A patent/NO983451L/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| TW446560B (en) | 2001-07-21 |
| IL125521A (en) | 2001-11-25 |
| PL328147A1 (en) | 1999-01-18 |
| AR010978A1 (en) | 2000-08-02 |
| CN1209745A (en) | 1999-03-03 |
| NO983451D0 (en) | 1998-07-27 |
| AU707892B2 (en) | 1999-07-22 |
| BR9700778A (en) | 1998-10-06 |
| WO1997026877A1 (en) | 1997-07-31 |
| IL125521A0 (en) | 1999-03-12 |
| EP0921799A4 (en) | 2002-03-13 |
| JP2000503994A (en) | 2000-04-04 |
| EP0921799A1 (en) | 1999-06-16 |
| EA199800677A1 (en) | 1999-02-25 |
| ID15917A (en) | 1997-08-21 |
| EA001104B1 (en) | 2000-10-30 |
| KR19990082054A (en) | 1999-11-15 |
| NO983451L (en) | 1998-07-27 |
| CZ235498A3 (en) | 1999-02-17 |
| CO4761062A1 (en) | 1999-04-27 |
| NZ331105A (en) | 2000-06-23 |
| MX9806036A (en) | 1998-11-29 |
| AU2123997A (en) | 1997-08-20 |
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