WO2013046222A3 - A process for the preparation of amorphous rosuvastatin calcium - Google Patents
A process for the preparation of amorphous rosuvastatin calcium Download PDFInfo
- Publication number
- WO2013046222A3 WO2013046222A3 PCT/IN2012/000526 IN2012000526W WO2013046222A3 WO 2013046222 A3 WO2013046222 A3 WO 2013046222A3 IN 2012000526 W IN2012000526 W IN 2012000526W WO 2013046222 A3 WO2013046222 A3 WO 2013046222A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- preparation
- rosuvastatin calcium
- amorphous rosuvastatin
- amorphous
- calcium
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
Abstract
The present invention provides amorphous rosuvastatin calcium having a degree of crystallinity less than about 5% and process for preparation thereof.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2253MU2011 | 2011-08-10 | ||
IN2253/MUM/2011 | 2011-08-10 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2013046222A2 WO2013046222A2 (en) | 2013-04-04 |
WO2013046222A3 true WO2013046222A3 (en) | 2013-06-20 |
Family
ID=47996555
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/IN2012/000526 WO2013046222A2 (en) | 2011-08-10 | 2012-07-27 | A process for the preparation of amorphous rosuvastatin calcium |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2013046222A2 (en) |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0521471A1 (en) * | 1991-07-01 | 1993-01-07 | Shionogi Seiyaku Kabushiki Kaisha | Pyrimidine derivatives as HMG-CoA reductase inhibitors |
WO2005040134A1 (en) * | 2003-10-22 | 2005-05-06 | Ranbaxy Laboratories Limited | Process for the preparation of amorphous rosuvastatin calcium |
WO2006136408A2 (en) * | 2005-06-24 | 2006-12-28 | Lek Pharmaceuticals D.D. | Process for preparing pure amorphous rosuvastatin calcium |
-
2012
- 2012-07-27 WO PCT/IN2012/000526 patent/WO2013046222A2/en active Application Filing
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0521471A1 (en) * | 1991-07-01 | 1993-01-07 | Shionogi Seiyaku Kabushiki Kaisha | Pyrimidine derivatives as HMG-CoA reductase inhibitors |
WO2005040134A1 (en) * | 2003-10-22 | 2005-05-06 | Ranbaxy Laboratories Limited | Process for the preparation of amorphous rosuvastatin calcium |
WO2006136408A2 (en) * | 2005-06-24 | 2006-12-28 | Lek Pharmaceuticals D.D. | Process for preparing pure amorphous rosuvastatin calcium |
Also Published As
Publication number | Publication date |
---|---|
WO2013046222A2 (en) | 2013-04-04 |
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