WO2012016314A9 - Composés dérivés de l'acide arachidonique et substitués avec des analogues de coxibs pour le traitement de la douleur - Google Patents
Composés dérivés de l'acide arachidonique et substitués avec des analogues de coxibs pour le traitement de la douleur Download PDFInfo
- Publication number
- WO2012016314A9 WO2012016314A9 PCT/BR2011/000275 BR2011000275W WO2012016314A9 WO 2012016314 A9 WO2012016314 A9 WO 2012016314A9 BR 2011000275 W BR2011000275 W BR 2011000275W WO 2012016314 A9 WO2012016314 A9 WO 2012016314A9
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- derived
- arachidonic acid
- substituted compounds
- treating pain
- coxib
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Abstract
La présente invention concerne l'obtention de composés dérivés de l'acide arachidonique et substitués avec des analogues de coxibs, ainsi que leurs sels, pour le traitement de la douleur. L'invention concerne également des compositions pharmaceutiques contenant des composés dérivés de l'acide arachidonique et substitués avec des analogues de coxibs, leurs sels et des excipients pharmaceutiquement acceptables pour le traitement de la douleur. Les analgésiques de l'invention peuvent être utilisés de manière isolée ou en association avec d'autres analgésiques, pour atténuer la douleur légère, modérée ou sévère.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
BRPI1003050-6A BRPI1003050B1 (pt) | 2010-08-04 | 2010-08-04 | Compostos derivados do ácido araquidônico substituídos com análogos de coxibes para tratamento de dor |
BRPI1003050-6 | 2010-08-04 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2012016314A1 WO2012016314A1 (fr) | 2012-02-09 |
WO2012016314A9 true WO2012016314A9 (fr) | 2012-03-22 |
Family
ID=45558870
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/BR2011/000275 WO2012016314A1 (fr) | 2010-08-04 | 2011-08-04 | Composés dérivés de l'acide arachidonique et substitués avec des analogues de coxibs pour le traitement de la douleur |
Country Status (2)
Country | Link |
---|---|
BR (1) | BRPI1003050B1 (fr) |
WO (1) | WO2012016314A1 (fr) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9562015B2 (en) | 2011-11-17 | 2017-02-07 | The Regents Of The University Of Colorado, A Body | Methods and compositions for enhanced drug delivery to the eye and extended delivery formulations |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7161016B1 (en) * | 1998-11-24 | 2007-01-09 | University Of Connecticut | Cannabimimetic lipid amides as useful medications |
US20040122089A1 (en) * | 2001-06-20 | 2004-06-24 | Martin Billy R. | Novel eicosanoid analgesics |
US20040092566A1 (en) * | 2002-11-12 | 2004-05-13 | Graneto Matthew J. | Celecoxib prodrug |
US20070105940A1 (en) * | 2005-10-19 | 2007-05-10 | Allergan, Inc. | Method for treating pain |
-
2010
- 2010-08-04 BR BRPI1003050-6A patent/BRPI1003050B1/pt active IP Right Grant
-
2011
- 2011-08-04 WO PCT/BR2011/000275 patent/WO2012016314A1/fr active Application Filing
Also Published As
Publication number | Publication date |
---|---|
BRPI1003050B1 (pt) | 2021-05-25 |
BRPI1003050A2 (pt) | 2014-03-25 |
WO2012016314A1 (fr) | 2012-02-09 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
WO2013170068A3 (fr) | Modulateurs du transport nucléaire et leurs utilisations | |
WO2012055567A3 (fr) | Utilisation de malononitrilamides dans la douleur neuropathique | |
WO2014028600A3 (fr) | Composés 3-aminocycloalkyl utilisés en tant qu'inhibiteurs de rorgammat et utilisations de ceux-ci | |
WO2012075362A3 (fr) | Modulateurs du récepteur cxcr4 de la chimiokine et leurs utilisations | |
WO2011085162A3 (fr) | Compositions topiques transdermiques de dexmédétomidine et leurs procédés d'utilisation | |
WO2012098562A3 (fr) | Compositions liquides pour administration par voie orale de sels de lanthane | |
WO2015056094A3 (fr) | Composition pharmaceutique comprenant un antagoniste de trpa1 et un agent analgésique | |
IL251543A0 (en) | Use of gel compounds in the production of medicine to prevent or treat skin diseases | |
WO2012053013A3 (fr) | Compositions pharmaceutiques d'agents anti-acné | |
WO2012162439A3 (fr) | Compositions comprenant de l'acide fusidique et leurs emballages | |
EA032271B9 (ru) | Вещества, фармацевтическая композиция и методы применения при лечении воспалительных заболеваний | |
WO2014011750A8 (fr) | Formulations de laquinimod sans agent alcalinisant | |
SG10201501579WA (en) | Composition comprising as active ingredient l-carnitine in combination with hydroxykynurennine-0-beta-dl-glucoside, for the prevention and/or treatment of pathologies of the eye due to ultraviolet radiation | |
MX363389B (es) | Composicion farmaceutica que comprende ivabradina amorfa. | |
WO2014071168A3 (fr) | Administration d'inhibiteurs de la signalisation tgfbêta, dérivés de benzothiazépine ou combinaisons de ceux-ci pour améliorer la fonction musculaire chez des patients cancéreux | |
WO2013087654A3 (fr) | Méthodes de prévention ou de traitement de troubles par l'augmentation de la biodisponibilité du fer et formulation pharmaceutique associée | |
WO2012085249A3 (fr) | Formes pharmaceutiques orales homogènes comprenant de la lercanidipine et de l'énalapril ou leurs sels pharmaceutiquement acceptables | |
WO2012029074A3 (fr) | Compositions pharmaceutiques de linézolide | |
MX2015008171A (es) | Formulacion que comprende agomelatina amorfa. | |
MX363558B (es) | Composiciones farmaceuticas que comprenden flurbiprofeno. | |
WO2012016314A9 (fr) | Composés dérivés de l'acide arachidonique et substitués avec des analogues de coxibs pour le traitement de la douleur | |
WO2013038200A3 (fr) | Troubles neurodéveloppementaux | |
WO2011107921A3 (fr) | Composition de milnacipran à libération modifiée | |
WO2014013090A3 (fr) | Formulation comprenant du fingolimod amorphe | |
WO2013072770A3 (fr) | Formulations pharmaceutiques comprenant de l'atorvastatine et du glimépiride |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
121 | Ep: the epo has been informed by wipo that ep was designated in this application |
Ref document number: 11813972 Country of ref document: EP Kind code of ref document: A1 |
|
NENP | Non-entry into the national phase |
Ref country code: DE |
|
122 | Ep: pct application non-entry in european phase |
Ref document number: 11813972 Country of ref document: EP Kind code of ref document: A1 |