WO2010007316A3 - NOUVEAUX DERIVES TRIAZOLO(4,3-a)PYRIDINE,LEUR PROCEDE DE PREPARATION,LEUR APPLICATION A TITRE DE MEDICAMENTS,COMPOSITIONS PHARMACEUTIQUES ET NOUVELLE UTILISATION NOTAMMENT COMME INHIBITEURS DE MET - Google Patents
NOUVEAUX DERIVES TRIAZOLO(4,3-a)PYRIDINE,LEUR PROCEDE DE PREPARATION,LEUR APPLICATION A TITRE DE MEDICAMENTS,COMPOSITIONS PHARMACEUTIQUES ET NOUVELLE UTILISATION NOTAMMENT COMME INHIBITEURS DE MET Download PDFInfo
- Publication number
- WO2010007316A3 WO2010007316A3 PCT/FR2009/051406 FR2009051406W WO2010007316A3 WO 2010007316 A3 WO2010007316 A3 WO 2010007316A3 FR 2009051406 W FR2009051406 W FR 2009051406W WO 2010007316 A3 WO2010007316 A3 WO 2010007316A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- novel
- medicaments
- preparation
- pharmaceutical compositions
- met inhibitors
- Prior art date
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P35/02—Antineoplastic agents specific for leukemia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Abstract
Priority Applications (11)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA2730959A CA2730959A1 (fr) | 2008-07-18 | 2009-07-16 | Nouveaux derives triazolo[4,3-a]pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met |
AU2009272516A AU2009272516A1 (en) | 2008-07-18 | 2009-07-16 | Novel triazolo(4,3-a)pyridine derivatives, process for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use, in particular as MET inhibitors |
JP2011517978A JP2011528337A (ja) | 2008-07-18 | 2009-07-16 | 新規トリアゾロ[4,3−a]ピリジン誘導体、これらの調製方法、医薬としてのこれらの使用、医薬組成物および、特にmet阻害剤としての、新規使用 |
US13/054,663 US20110263594A1 (en) | 2008-07-18 | 2009-07-16 | Novel triazolo(4,3-a)pyridine derivatives, process for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use, in particular as met inhibitors |
EP09736253A EP2310366A2 (fr) | 2008-07-18 | 2009-07-16 | NOUVEAUX DERIVES TRIAZOLO(4,3-a)PYRIDINE,LEUR PROCEDE DE PREPARATION,LEUR APPLICATION A TITRE DE MEDICAMENTS,COMPOSITIONS PHARMACEUTIQUES ET NOUVELLE UTILISATION NOTAMMENT COMME INHIBITEURS DE MET |
EA201170222A EA201170222A1 (ru) | 2008-07-18 | 2009-07-16 | НОВЫЕ ПРОИЗВОДНЫЕ ТРИАЗОЛО[4,3-a]ПИРИДИНА, СПОСОБ ИХ ПОЛУЧЕНИЯ, ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ЛЕКАРСТВЕННЫХ СРЕДСТВ, ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ И НОВОЕ ПРИМЕНЕНИЕ, В ЧАСТНОСТИ, В КАЧЕСТВЕ ИНГИБИТОРОВ МЕТ |
CN2009801365397A CN102159543A (zh) | 2008-07-18 | 2009-07-16 | 新颖的三唑并[4,3-a]吡啶衍生物,其制备方法,其作为药物的用途,药物组合物及新颖的尤其是作为MET抑制剂的用途 |
BRPI0916464-2A BRPI0916464A2 (pt) | 2008-07-18 | 2009-07-16 | derivados triazolo(4,3-a) piridina, o respectivo processo de preparo, a respectiva aplicação como medicamentos, composições farmacêuticas e utilização notadamente como inibidores de met |
MX2011000671A MX2011000671A (es) | 2008-07-18 | 2009-07-16 | Nuevos derivados de triazolo [4,3-a] piridina su procedimiento de preparacion, su uso como medicamentos, composiciones farmaceuticas y nuevo uso particularmente como inhibidores de met. |
IL210688A IL210688A0 (en) | 2008-07-18 | 2011-01-16 | Novel triazolo(4,3-a)pyridine derivatives, process for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use, in particular as met inhibitors |
MA33625A MA32570B1 (fr) | 2008-07-18 | 2011-02-15 | NOUVEAUX DERIVES TRIAZOLO(4,3-a)PYRIDINE,LEUR PROCEDE DE PREPARATION,LEUR APPLICATION A TITRE DE MEDICAMENTS,COMPOSITIONS PHARMACEUTIQUES ET NOUVELLE UTILISATION NOTAMMENT COMME INHIBITEURS DE MET |
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0804084 | 2008-07-18 | ||
FR0804084A FR2933980B1 (fr) | 2008-07-18 | 2008-07-18 | Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met |
FR0900245A FR2941229B1 (fr) | 2009-01-21 | 2009-01-21 | Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met |
FR0900245 | 2009-01-21 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2010007316A2 WO2010007316A2 (fr) | 2010-01-21 |
WO2010007316A3 true WO2010007316A3 (fr) | 2010-04-29 |
Family
ID=41550767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/FR2009/051406 WO2010007316A2 (fr) | 2008-07-18 | 2009-07-16 | NOUVEAUX DERIVES TRIAZOLO(4,3-a)PYRIDINE,LEUR PROCEDE DE PREPARATION,LEUR APPLICATION A TITRE DE MEDICAMENTS,COMPOSITIONS PHARMACEUTIQUES ET NOUVELLE UTILISATION NOTAMMENT COMME INHIBITEURS DE MET |
Country Status (19)
Country | Link |
---|---|
US (1) | US20110263594A1 (fr) |
EP (1) | EP2310366A2 (fr) |
JP (1) | JP2011528337A (fr) |
KR (1) | KR20110039558A (fr) |
CN (1) | CN102159543A (fr) |
AR (1) | AR072819A1 (fr) |
AU (1) | AU2009272516A1 (fr) |
BR (1) | BRPI0916464A2 (fr) |
CA (1) | CA2730959A1 (fr) |
CL (1) | CL2011000119A1 (fr) |
CO (1) | CO6331463A2 (fr) |
EA (1) | EA201170222A1 (fr) |
IL (1) | IL210688A0 (fr) |
MA (1) | MA32570B1 (fr) |
MX (1) | MX2011000671A (fr) |
PE (1) | PE20110560A1 (fr) |
TW (1) | TW201008938A (fr) |
UY (1) | UY31996A (fr) |
WO (1) | WO2010007316A2 (fr) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100041663A1 (en) | 2008-07-18 | 2010-02-18 | Novartis Ag | Organic Compounds as Smo Inhibitors |
US8759535B2 (en) | 2010-02-18 | 2014-06-24 | High Point Pharmaceuticals, Llc | Substituted fused imidazole derivatives, pharmaceutical compositions, and methods of use thereof |
FR2966151B1 (fr) * | 2010-10-14 | 2012-11-09 | Sanofi Aventis | Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met |
US9127000B2 (en) * | 2011-02-23 | 2015-09-08 | Intellikine, LLC. | Heterocyclic compounds and uses thereof |
MX339302B (es) | 2011-09-15 | 2016-05-19 | Novartis Ag | 3-(quinolin-6-il-tio)-[1,2,4]-triazolo-[4,3-a]-piridinas 6-sustituidas como cinasas de tirosina. |
AU2014262326B2 (en) * | 2013-05-10 | 2018-03-22 | Jiangsu Hansoh Pharmaceutical Co., Ltd. | [1,2,4] triazol [4,3-a] pyridine derivate, preparation method therefor or medical application thereof |
EP3004095A1 (fr) * | 2013-06-03 | 2016-04-13 | Bayer Pharma Aktiengesellschaft | Triazolopyridines utilisées comme inhibiteurs de la thrombine pour traiter des maladies thromboemboliques |
GB201321742D0 (en) * | 2013-12-09 | 2014-01-22 | Ucb Pharma Sa | Therapeutic agents |
WO2016089648A1 (fr) | 2014-12-01 | 2016-06-09 | Vtv Therapeutics Llc | Inhibiteurs de bach1 en combinaison avec des activateurs de nrf2 et compositions pharmaceutiques les contenant |
CN106489962B (zh) * | 2016-10-20 | 2019-02-22 | 贵州大学 | 一种[1,2,4]三唑[4,3-a]吡啶类含硫化合物在制备杀虫剂中的应用 |
AU2018378935A1 (en) | 2017-12-07 | 2020-06-25 | The Regents Of The University Of Michigan | NSD family inhibitors and methods of treatment therewith |
US20220143049A1 (en) | 2019-03-21 | 2022-05-12 | Onxeo | A dbait molecule in combination with kinase inhibitor for the treatment of cancer |
JP2023500906A (ja) | 2019-11-08 | 2023-01-11 | インサーム(インスティテュ ナシオナル ドゥ ラ サンテ エ ドゥ ラ ルシェルシェ メディカル) | キナーゼ阻害剤に対する獲得抵抗性を有するがんの処置方法 |
WO2021148581A1 (fr) | 2020-01-22 | 2021-07-29 | Onxeo | Nouvelle molécule dbait et son utilisation |
Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2857371A (en) * | 1954-09-10 | 1958-10-21 | Eastman Kodak Co | Benzothiazole azo diphenylamine compounds |
EP0048555A1 (fr) * | 1980-08-27 | 1982-03-31 | Glaxo Group Limited | Dérivés aminés du 1,2,4 triazole, leur procédé de préparation et médicaments les contenant |
EP0254623A1 (fr) * | 1986-07-23 | 1988-01-27 | Laboratoires Upsa | Nouveaux dérivés amino alkyl thio de triazolopyridine ou triazoloquinoline, leurs procédés de préparation, médicaments les contenant, utiles notamment comme antalgiques |
US20060057510A1 (en) * | 2004-09-07 | 2006-03-16 | Eastman Kodak Company | Silver salt-toner co-precipitates and imaging materials |
WO2007075567A1 (fr) * | 2005-12-21 | 2007-07-05 | Janssen Pharmaceutica, N.V. | Triazolopyridazines en tant que modulateurs de la tyrosine kinase |
WO2008092888A1 (fr) * | 2007-02-01 | 2008-08-07 | Glaxo Group Limited | Dérivés 1-oxa-3-azaspiro [4,5] décane-2-one pour le traitement de troubles de l'alimentation |
WO2009056692A2 (fr) * | 2007-08-09 | 2009-05-07 | Sanofi-Aventis | Nouveaux derives de 6-triazolopyridazine-sulfanyl benzothiazole et benzimidazole, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met |
-
2009
- 2009-07-16 BR BRPI0916464-2A patent/BRPI0916464A2/pt not_active IP Right Cessation
- 2009-07-16 KR KR1020117003697A patent/KR20110039558A/ko not_active Application Discontinuation
- 2009-07-16 MX MX2011000671A patent/MX2011000671A/es not_active Application Discontinuation
- 2009-07-16 CN CN2009801365397A patent/CN102159543A/zh active Pending
- 2009-07-16 US US13/054,663 patent/US20110263594A1/en not_active Abandoned
- 2009-07-16 PE PE2011000048A patent/PE20110560A1/es not_active Application Discontinuation
- 2009-07-16 CA CA2730959A patent/CA2730959A1/fr not_active Abandoned
- 2009-07-16 AU AU2009272516A patent/AU2009272516A1/en not_active Abandoned
- 2009-07-16 EA EA201170222A patent/EA201170222A1/ru unknown
- 2009-07-16 JP JP2011517978A patent/JP2011528337A/ja not_active Withdrawn
- 2009-07-16 EP EP09736253A patent/EP2310366A2/fr not_active Withdrawn
- 2009-07-16 TW TW098124130A patent/TW201008938A/zh unknown
- 2009-07-16 WO PCT/FR2009/051406 patent/WO2010007316A2/fr active Application Filing
- 2009-07-17 UY UY0001031996A patent/UY31996A/es not_active Application Discontinuation
- 2009-07-17 AR ARP090102727A patent/AR072819A1/es unknown
-
2011
- 2011-01-16 IL IL210688A patent/IL210688A0/en unknown
- 2011-01-18 CO CO11004610A patent/CO6331463A2/es not_active Application Discontinuation
- 2011-01-18 CL CL2011000119A patent/CL2011000119A1/es unknown
- 2011-02-15 MA MA33625A patent/MA32570B1/fr unknown
Patent Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2857371A (en) * | 1954-09-10 | 1958-10-21 | Eastman Kodak Co | Benzothiazole azo diphenylamine compounds |
EP0048555A1 (fr) * | 1980-08-27 | 1982-03-31 | Glaxo Group Limited | Dérivés aminés du 1,2,4 triazole, leur procédé de préparation et médicaments les contenant |
EP0254623A1 (fr) * | 1986-07-23 | 1988-01-27 | Laboratoires Upsa | Nouveaux dérivés amino alkyl thio de triazolopyridine ou triazoloquinoline, leurs procédés de préparation, médicaments les contenant, utiles notamment comme antalgiques |
US20060057510A1 (en) * | 2004-09-07 | 2006-03-16 | Eastman Kodak Company | Silver salt-toner co-precipitates and imaging materials |
WO2007075567A1 (fr) * | 2005-12-21 | 2007-07-05 | Janssen Pharmaceutica, N.V. | Triazolopyridazines en tant que modulateurs de la tyrosine kinase |
WO2008092888A1 (fr) * | 2007-02-01 | 2008-08-07 | Glaxo Group Limited | Dérivés 1-oxa-3-azaspiro [4,5] décane-2-one pour le traitement de troubles de l'alimentation |
WO2009056692A2 (fr) * | 2007-08-09 | 2009-05-07 | Sanofi-Aventis | Nouveaux derives de 6-triazolopyridazine-sulfanyl benzothiazole et benzimidazole, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met |
Non-Patent Citations (2)
Title |
---|
DATABASE CHEMCATS, [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; 4 December 2008 (2008-12-04), SPECS: "Compounds for screening", XP002543539, retrieved from CHEMCATS * |
EDMONDSON, SCOTT D. ET AL: "(2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4- [1,2,4]triazolo[1,5-a]- pyridin-6-ylphenyl)butanamide: A selective .alpha.-amino amide dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes", JOURNAL OF MEDICINAL CHEMISTRY, vol. 49, no. 12, 2006, pages 3614 - 3627, XP002543538, ISSN: 0022-2623 * |
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Publication number | Publication date |
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TW201008938A (en) | 2010-03-01 |
KR20110039558A (ko) | 2011-04-19 |
JP2011528337A (ja) | 2011-11-17 |
PE20110560A1 (es) | 2011-08-29 |
WO2010007316A2 (fr) | 2010-01-21 |
BRPI0916464A2 (pt) | 2018-06-12 |
MX2011000671A (es) | 2011-04-11 |
US20110263594A1 (en) | 2011-10-27 |
CA2730959A1 (fr) | 2010-01-21 |
CO6331463A2 (es) | 2011-10-20 |
MA32570B1 (fr) | 2011-08-01 |
CL2011000119A1 (es) | 2011-06-17 |
UY31996A (es) | 2010-02-26 |
AR072819A1 (es) | 2010-09-22 |
CN102159543A (zh) | 2011-08-17 |
IL210688A0 (en) | 2011-03-31 |
EP2310366A2 (fr) | 2011-04-20 |
AU2009272516A1 (en) | 2010-01-21 |
EA201170222A1 (ru) | 2011-08-30 |
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