WO2009112203A1 - Procédé de fabrication d’une diphénylazétidinone - Google Patents

Procédé de fabrication d’une diphénylazétidinone Download PDF

Info

Publication number
WO2009112203A1
WO2009112203A1 PCT/EP2009/001598 EP2009001598W WO2009112203A1 WO 2009112203 A1 WO2009112203 A1 WO 2009112203A1 EP 2009001598 W EP2009001598 W EP 2009001598W WO 2009112203 A1 WO2009112203 A1 WO 2009112203A1
Authority
WO
WIPO (PCT)
Prior art keywords
compound
formula
butyl
ethylmorpholine
ethyldiisopropylamine
Prior art date
Application number
PCT/EP2009/001598
Other languages
German (de)
English (en)
Inventor
Theodor Andreas Wollmann
Bernd Junker
Bernhard Otto
Claus-Jürgen MAIER
Original Assignee
Sanofi-Aventis Deutschland Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102008059772A external-priority patent/DE102008059772A1/de
Application filed by Sanofi-Aventis Deutschland Gmbh filed Critical Sanofi-Aventis Deutschland Gmbh
Publication of WO2009112203A1 publication Critical patent/WO2009112203A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton

Abstract

L’invention concerne un procédé amélioré de fabrication d’une diphénylazétidinone.
PCT/EP2009/001598 2008-03-14 2009-03-06 Procédé de fabrication d’une diphénylazétidinone WO2009112203A1 (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
EP08004862.2 2008-03-14
EP08004862 2008-03-14
US4529908P 2008-04-16 2008-04-16
US61/045,299 2008-04-16
DE102008059772.4 2008-12-01
DE102008059772A DE102008059772A1 (de) 2008-12-01 2008-12-01 Verfahren zur Herstellung eines Diphenylazetidinons

Publications (1)

Publication Number Publication Date
WO2009112203A1 true WO2009112203A1 (fr) 2009-09-17

Family

ID=40823593

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2009/001598 WO2009112203A1 (fr) 2008-03-14 2009-03-06 Procédé de fabrication d’une diphénylazétidinone

Country Status (1)

Country Link
WO (1) WO2009112203A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8003636B2 (en) * 2007-11-13 2011-08-23 Sanofi-Aventis Deutschland Gmbh Certain crystalline diphenylazetidinone hydrates, pharmaceutical compositions thereof and methods for their use

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004087655A1 (fr) * 2003-04-01 2004-10-14 Sanofi-Aventis Deutschland Gmbh Nouveau diphenylazetidinone a proprietes physiologiques ameliorees, procedes de production associe, medicaments contenant les composes et leurs utilisations
US7067689B1 (en) * 2005-07-08 2006-06-27 Microbia, Inc. Process for production of pentahydroxyhexylcarbamoyl alkanoic acids

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004087655A1 (fr) * 2003-04-01 2004-10-14 Sanofi-Aventis Deutschland Gmbh Nouveau diphenylazetidinone a proprietes physiologiques ameliorees, procedes de production associe, medicaments contenant les composes et leurs utilisations
US7067689B1 (en) * 2005-07-08 2006-06-27 Microbia, Inc. Process for production of pentahydroxyhexylcarbamoyl alkanoic acids

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8003636B2 (en) * 2007-11-13 2011-08-23 Sanofi-Aventis Deutschland Gmbh Certain crystalline diphenylazetidinone hydrates, pharmaceutical compositions thereof and methods for their use

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