WO2009057138A3 - Compositions pharmaceutiques à libération régulée de toltérodine - Google Patents
Compositions pharmaceutiques à libération régulée de toltérodine Download PDFInfo
- Publication number
- WO2009057138A3 WO2009057138A3 PCT/IN2008/000695 IN2008000695W WO2009057138A3 WO 2009057138 A3 WO2009057138 A3 WO 2009057138A3 IN 2008000695 W IN2008000695 W IN 2008000695W WO 2009057138 A3 WO2009057138 A3 WO 2009057138A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- tolterodine
- controlled release
- release pharmaceutical
- pharmaceutical compositions
- pharmaceutically acceptable
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
L'invention porte sur une composition pharmaceutique à libération régulée qui contient un noyau comportant de la toltérodine ou des sels acceptables du point de vue pharmaceutique de celle-ci, des excipients auxiliaires et une seule couche d'enrobage comportant un ou des agents de régulation de vitesse. L'invention porte également sur une composition pharmaceutique à libération régulée qui comporte de la toltérodine ou des sels acceptables du point de vue pharmaceutique de celle-ci, le noyau comportant de la toltérodine ou des sels acceptables du point de vue pharmaceutique de celle-ci, des excipients auxiliaires et une seule couche d'enrobage comportant un ou des agents de régulation de la vitesse, ladite composition comportant en outre un ou des agents améliorant la dissolution.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2010531645A JP2011502140A (ja) | 2007-10-29 | 2008-10-22 | トルテロジンの制御放出型医薬組成物 |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1475/KOL/2007 | 2007-10-29 | ||
IN1475KO2007 | 2007-10-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2009057138A2 WO2009057138A2 (fr) | 2009-05-07 |
WO2009057138A3 true WO2009057138A3 (fr) | 2009-07-23 |
Family
ID=40405020
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/IN2008/000695 WO2009057138A2 (fr) | 2007-10-29 | 2008-10-22 | Compositions pharmaceutiques à libération régulée de toltérodine |
Country Status (2)
Country | Link |
---|---|
JP (1) | JP2011502140A (fr) |
WO (1) | WO2009057138A2 (fr) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8871275B2 (en) | 2007-08-08 | 2014-10-28 | Inventia Healthcare Private Limited | Extended release compositions comprising tolterodine |
CA2761602C (fr) * | 2009-05-11 | 2015-07-07 | Ratiopharm Gmbh | Desfesoterodine sous forme de sel d'acide tartrique |
TR201111143T1 (tr) * | 2009-05-11 | 2012-05-21 | Lupin Limited | Yeni̇ farmasöti̇k koli̇n fenofi̇brat bi̇leşi̇mleri̇ |
ES2600894T3 (es) * | 2010-02-22 | 2017-02-13 | Daiichi Sankyo Company, Limited | Preparación sólida de liberación sostenida para uso oral |
WO2011102504A1 (fr) | 2010-02-22 | 2011-08-25 | 第一三共株式会社 | Préparation solide à libération prolongée pour utilisation orale |
SG174658A1 (en) * | 2010-04-01 | 2011-10-28 | Theravida Inc | Pharmaceutical formulations for the treatment of overactive bladder |
SG194809A1 (en) | 2011-05-10 | 2013-12-30 | Theravida Inc | Combinations of solifenacin and salivary stimulants for the treatment of overactive bladder |
WO2014034929A1 (fr) | 2012-09-03 | 2014-03-06 | 第一三共株式会社 | Composition pharmaceutique à libération prolongée administrée par voie orale contenant du chlorhydrate d'hydromorphone |
CA2993823C (fr) | 2015-07-28 | 2024-01-02 | Board Of Regents, The University Of Texas System | Compositions d'implant destinees a l'apport unidirectionnel de composes therapeutiques au cerveau |
JP6841834B2 (ja) | 2016-01-20 | 2021-03-10 | テラヴィダ, インコーポレイテッドTheraVida, Inc. | 多汗症の処置のための方法および組成物 |
Citations (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2004105735A1 (fr) * | 2003-05-30 | 2004-12-09 | Ranbaxy Laboratories Limited | Compositions pharmaceutiques de tolterodine a liberation controlee et leurs procedes de preparation |
WO2005105036A1 (fr) * | 2004-04-28 | 2005-11-10 | Natco Pharma Limited | Matrice muco-adhesive a liberation controlee contenant de la tolterodine, et procede d'elaboration |
WO2007029087A2 (fr) * | 2005-09-05 | 2007-03-15 | Ranbaxy Laboratories Limited | Preparations multi-unites a liberation controlee |
WO2007113207A2 (fr) * | 2006-03-31 | 2007-10-11 | Lek Pharmaceuticals D.D. | Formulations enduites |
WO2008012346A1 (fr) * | 2006-07-28 | 2008-01-31 | Farmaprojects, S. A. | Préparation pharmaceutique de métoprolol à libération prolongée et son procédé de préparation |
WO2009019599A2 (fr) * | 2007-08-08 | 2009-02-12 | Themis Laboratories Private Limited | Compositions à libération prolongée comprenant de la toltérodine |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS59175414A (ja) * | 1983-03-23 | 1984-10-04 | Toyo Jozo Co Ltd | マクロライド抗生物質の安定な経口用製剤および安定化法 |
JP2001316292A (ja) * | 1999-09-03 | 2001-11-13 | Takeda Chem Ind Ltd | 医 薬 |
-
2008
- 2008-10-22 WO PCT/IN2008/000695 patent/WO2009057138A2/fr active Application Filing
- 2008-10-22 JP JP2010531645A patent/JP2011502140A/ja active Pending
Patent Citations (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2004105735A1 (fr) * | 2003-05-30 | 2004-12-09 | Ranbaxy Laboratories Limited | Compositions pharmaceutiques de tolterodine a liberation controlee et leurs procedes de preparation |
WO2005105036A1 (fr) * | 2004-04-28 | 2005-11-10 | Natco Pharma Limited | Matrice muco-adhesive a liberation controlee contenant de la tolterodine, et procede d'elaboration |
WO2007029087A2 (fr) * | 2005-09-05 | 2007-03-15 | Ranbaxy Laboratories Limited | Preparations multi-unites a liberation controlee |
WO2007113207A2 (fr) * | 2006-03-31 | 2007-10-11 | Lek Pharmaceuticals D.D. | Formulations enduites |
WO2008012346A1 (fr) * | 2006-07-28 | 2008-01-31 | Farmaprojects, S. A. | Préparation pharmaceutique de métoprolol à libération prolongée et son procédé de préparation |
WO2009019599A2 (fr) * | 2007-08-08 | 2009-02-12 | Themis Laboratories Private Limited | Compositions à libération prolongée comprenant de la toltérodine |
Also Published As
Publication number | Publication date |
---|---|
WO2009057138A2 (fr) | 2009-05-07 |
JP2011502140A (ja) | 2011-01-20 |
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