WO2009004873A1 - プロスタグランジン誘導体含有水性液剤 - Google Patents

プロスタグランジン誘導体含有水性液剤 Download PDF

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Publication number
WO2009004873A1
WO2009004873A1 PCT/JP2008/059774 JP2008059774W WO2009004873A1 WO 2009004873 A1 WO2009004873 A1 WO 2009004873A1 JP 2008059774 W JP2008059774 W JP 2008059774W WO 2009004873 A1 WO2009004873 A1 WO 2009004873A1
Authority
WO
WIPO (PCT)
Prior art keywords
aqueous liquid
liquid agent
prostaglandin derivative
containing aqueous
glycol
Prior art date
Application number
PCT/JP2008/059774
Other languages
English (en)
French (fr)
Inventor
Kaori Nishizaki
Takayuki Sato
Kentaro Goto
Kuniaki Ishii
Original Assignee
Taisho Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taisho Pharmaceutical Co., Ltd. filed Critical Taisho Pharmaceutical Co., Ltd.
Priority to EP08764790A priority Critical patent/EP2172202A4/en
Priority to US12/666,804 priority patent/US8044104B2/en
Priority to JP2009521556A priority patent/JPWO2009004873A1/ja
Publication of WO2009004873A1 publication Critical patent/WO2009004873A1/ja

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Medicinal Preparation (AREA)

Abstract

（ａ）下記式（Ｉ） で表されるプロスタグランジン誘導体若しくはその製薬学的に許容される塩又はそれらの水和物、並びに、（ｂ）グリセリン、プロピレングリコール、ジプロピレングリコール及び１，３－ブチレングリコールの少なくとも１種の多価アルコール、を含有することを特徴とする水性液剤を提供する。
PCT/JP2008/059774 2007-06-29 2008-05-28 プロスタグランジン誘導体含有水性液剤 WO2009004873A1 (ja)

Priority Applications (3)

Application Number Priority Date Filing Date Title
EP08764790A EP2172202A4 (en) 2007-06-29 2008-05-28 AQUEOUS LIQUID AGENT CONTAINING A PROSTAGLANDINE DERIVATIVE
US12/666,804 US8044104B2 (en) 2007-06-29 2008-05-28 Prostaglandin derivative-containing aqueous liquid preparation
JP2009521556A JPWO2009004873A1 (ja) 2007-06-29 2008-05-28 プロスタグランジン誘導体含有水性液剤

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007172331 2007-06-29
JP2007-172331 2007-06-29

Publications (1)

Publication Number Publication Date
WO2009004873A1 true WO2009004873A1 (ja) 2009-01-08

Family

ID=40225929

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2008/059774 WO2009004873A1 (ja) 2007-06-29 2008-05-28 プロスタグランジン誘導体含有水性液剤

Country Status (4)

Country Link
US (1) US8044104B2 (ja)
EP (1) EP2172202A4 (ja)
JP (1) JPWO2009004873A1 (ja)
WO (1) WO2009004873A1 (ja)

Citations (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02282329A (ja) * 1989-04-25 1990-11-19 Green Cross Corp:The プロスタグランジン含有液状組成物
JPH05229928A (ja) * 1992-02-24 1993-09-07 Kao Corp 化粧水
WO1997030696A1 (fr) * 1996-02-26 1997-08-28 Daiichi Pharmaceutical Co., Ltd. Liposome et dispersion de liposome
JP2000319163A (ja) * 1999-05-07 2000-11-21 Masako Motomura 肌洗浄液、および肌払拭材
JP2003238328A (ja) * 2002-02-13 2003-08-27 Fancl Corp 低刺激性皮膚外用剤
JP2003238336A (ja) * 2002-02-13 2003-08-27 Fancl Corp 化粧料組成物
JP2003528895A (ja) * 2000-03-31 2003-09-30 ザ プロクター アンド ギャンブル カンパニー オキシミルプロスタグランジン及びヒドロキシルアミノプロスタグランジンを使用した脱毛症治療用組成物及びその治療方法
WO2004014394A1 (ja) 2002-08-09 2004-02-19 Taisho Pharmaceutical Co.,Ltd. 止痒剤
WO2005044276A1 (ja) * 2003-11-07 2005-05-19 Senju Pharmaceutical Co., Ltd. プロスタグランジン含有医薬組成物
JP2005247842A (ja) * 2004-02-06 2005-09-15 Taisho Pharmaceut Co Ltd 乾皮症治療剤
WO2006085655A1 (ja) 2005-02-14 2006-08-17 Taisho Pharmaceutical Co., Ltd. 軟膏剤

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7737182B2 (en) * 2002-08-09 2010-06-15 Taisho Pharmaceutical Co., Ltd. Pharmaceuticals for xerosis
US7254362B2 (en) * 2003-11-07 2007-08-07 Ricoh Company, Ltd. Fixing device, image forming apparatus using the fixing device, and heat insulating member

Patent Citations (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02282329A (ja) * 1989-04-25 1990-11-19 Green Cross Corp:The プロスタグランジン含有液状組成物
JPH05229928A (ja) * 1992-02-24 1993-09-07 Kao Corp 化粧水
WO1997030696A1 (fr) * 1996-02-26 1997-08-28 Daiichi Pharmaceutical Co., Ltd. Liposome et dispersion de liposome
JP2000319163A (ja) * 1999-05-07 2000-11-21 Masako Motomura 肌洗浄液、および肌払拭材
JP2003528895A (ja) * 2000-03-31 2003-09-30 ザ プロクター アンド ギャンブル カンパニー オキシミルプロスタグランジン及びヒドロキシルアミノプロスタグランジンを使用した脱毛症治療用組成物及びその治療方法
JP2003238328A (ja) * 2002-02-13 2003-08-27 Fancl Corp 低刺激性皮膚外用剤
JP2003238336A (ja) * 2002-02-13 2003-08-27 Fancl Corp 化粧料組成物
WO2004014394A1 (ja) 2002-08-09 2004-02-19 Taisho Pharmaceutical Co.,Ltd. 止痒剤
WO2005044276A1 (ja) * 2003-11-07 2005-05-19 Senju Pharmaceutical Co., Ltd. プロスタグランジン含有医薬組成物
JP2005247842A (ja) * 2004-02-06 2005-09-15 Taisho Pharmaceut Co Ltd 乾皮症治療剤
WO2006085655A1 (ja) 2005-02-14 2006-08-17 Taisho Pharmaceutical Co., Ltd. 軟膏剤

Non-Patent Citations (4)

* Cited by examiner, † Cited by third party
Title
DRAIZE: "Appraisal of the safety of chemicals in foods, drugs and cosmetics", 1959, ASSOCIATION OF FOOD & DRUG OFFICIALS OF THE UNITED STATES, pages: 46 - 59
KAY; CALANDRA: "Interpretation of eye irritation tests", J. SOC. COSM. CHEM., vol. 13, 1962, pages 281 - 289
See also references of EP2172202A4
TAKANO N ET AL., EUROPEAN JOURNAL OF PHARMACOLOGY, vol. 471, 2003, pages 223 - 8

Also Published As

Publication number Publication date
US20100204331A1 (en) 2010-08-12
EP2172202A4 (en) 2010-06-30
JPWO2009004873A1 (ja) 2010-08-26
US8044104B2 (en) 2011-10-25
EP2172202A1 (en) 2010-04-07

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