WO2008081711A1 - ２－含フッ素アシル－３－アミノアクリロニトリル誘導体及びその製造方法 - Google Patents

２－含フッ素アシル－３－アミノアクリロニトリル誘導体及びその製造方法 Download PDF

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Publication number
WO2008081711A1
WO2008081711A1 PCT/JP2007/074306 JP2007074306W WO2008081711A1 WO 2008081711 A1 WO2008081711 A1 WO 2008081711A1 JP 2007074306 W JP2007074306 W JP 2007074306W WO 2008081711 A1 WO2008081711 A1 WO 2008081711A1
Authority
WO
WIPO (PCT)
Prior art keywords
fluorinated acyl
derivative
producing
aminoacrylonitrile
aminoacrylonitrile derivative
Prior art date
Application number
PCT/JP2007/074306
Other languages
English (en)
French (fr)
Inventor
Hideki Umetani
Yoji Aoki
Takeshi Kakimoto
Original Assignee
Mitsui Chemicals Agro, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsui Chemicals Agro, Inc. filed Critical Mitsui Chemicals Agro, Inc.
Priority to AU2007340689A priority Critical patent/AU2007340689A1/en
Priority to BRPI0720715-8A priority patent/BRPI0720715A2/pt
Priority to MX2009007029A priority patent/MX2009007029A/es
Priority to EP07850792A priority patent/EP2105434A4/en
Priority to US12/521,436 priority patent/US20100010216A1/en
Priority to JP2008552083A priority patent/JPWO2008081711A1/ja
Publication of WO2008081711A1 publication Critical patent/WO2008081711A1/ja

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/30—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same unsaturated acyclic carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/145—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

　２－含フッ素アシル－３－アミノアクリロニトリル誘導体及びその製造方法を提供する。 　含フッ素アシル誘導体とアミノアクリロニトリル誘導体を反応させることにより、目的とする下記一般式（３） 【化１】 （式中、Ｒｆは少なくとも１つのフッ素原子で置換されている炭素数１～６のアルキル基を表し、Ｒ１とＲ２はそれぞれ独立していて、水素原子、炭素数１～６のアルキル基等を表し、Ｒ３は、水素原子、炭素数１～６のアルキル基等を表す。）で表される２－含フッ素アシル－３－アミノアクリロニトリル誘導体を製造する。
PCT/JP2007/074306 2006-12-28 2007-12-18 ２－含フッ素アシル－３－アミノアクリロニトリル誘導体及びその製造方法 WO2008081711A1 (ja)

Priority Applications (6)

Application Number Priority Date Filing Date Title
AU2007340689A AU2007340689A1 (en) 2006-12-28 2007-12-18 2-fluorinated acyl-3-aminoacrylonitrile derivative and method for producing the same
BRPI0720715-8A BRPI0720715A2 (pt) 2006-12-28 2007-12-18 Derivado de acil-3-aminoacrilonitrila 2-fluorado e método para produzir o mesmo
MX2009007029A MX2009007029A (es) 2006-12-28 2007-12-18 Derivado de acil-3-aminoacrilonitrilo 2-fluorado y metodo para producir el mismo.
EP07850792A EP2105434A4 (en) 2006-12-28 2007-12-18 2- (ACYL FLUORINATED) -3-AMINOACRYLONITRILE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME
US12/521,436 US20100010216A1 (en) 2006-12-28 2007-12-18 2-fluorinated acyl-3-aminoacrylonitrile derivative and method for producing the same
JP2008552083A JPWO2008081711A1 (ja) 2006-12-28 2007-12-18 ２−含フッ素アシル−３−アミノアクリロニトリル誘導体及びその製造方法

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006-355146 2006-12-28
JP2006355146 2006-12-28

Publications (1)

Publication Number Publication Date
WO2008081711A1 true WO2008081711A1 (ja) 2008-07-10

Family

ID=39588395

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2007/074306 WO2008081711A1 (ja) 2006-12-28 2007-12-18 ２－含フッ素アシル－３－アミノアクリロニトリル誘導体及びその製造方法

Country Status (10)

Country Link
US (1) US20100010216A1 (ja)
EP (1) EP2105434A4 (ja)
JP (1) JPWO2008081711A1 (ja)
CN (1) CN101627008A (ja)
AU (1) AU2007340689A1 (ja)
BR (1) BRPI0720715A2 (ja)
MX (1) MX2009007029A (ja)
RU (1) RU2009124415A (ja)
TW (1) TW200837041A (ja)
WO (1) WO2008081711A1 (ja)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010540477A (ja) * 2007-09-26 2010-12-24 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト ２−ジハロアシル−３−アミノアクリル酸誘導体の調製方法
WO2012065905A1 (en) 2010-11-15 2012-05-24 Bayer Cropscience Ag Cyanoenamines and their use as fungicides

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104163800B (zh) * 2014-08-19 2016-09-28 一帆生物科技集团有限公司 一种3-二氟甲基-1-甲基-1h-吡唑-4-羧酸的制备方法
CN113354495A (zh) * 2021-05-20 2021-09-07 上海应用技术大学 一种二氟酮羰基取代不对称腈类化合物及其制备与应用

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966791A (en) 1974-06-19 1976-06-29 Hoffmann-La Roche Inc. Preparation of dialkyl amino acrylonitrile
JPS55130950A (en) 1979-03-29 1980-10-11 Dynamit Nobel Ag Betaaalkoxyyacrylonitrile*33aminooacryonitrile and 22cyanoovinylester manufacture
JPS63264448A (ja) * 1988-02-29 1988-11-01 Shionogi & Co Ltd 新規β−ケトニトリル
JP2003113153A (ja) * 2001-08-02 2003-04-18 Ube Ind Ltd β−オキソニトリル誘導体又はそのアルカリ金属塩の製法
JP2003267943A (ja) * 2002-03-15 2003-09-25 Fuji Photo Film Co Ltd ジシアノメチリデン化合物及びヘテロ環化合物の合成方法
JP2005511782A (ja) 2001-12-17 2005-04-28 バイエル ケミカルズ アクチエンゲゼルシャフト ２−ハロゲンアシル−３−アミノ−アクリル酸−誘導体の製造方法
JP2006514059A (ja) 2002-12-27 2006-04-27 アムゲン インコーポレイテッド 細胞増殖及びアポトーシスに関連する疾患の処置に使用する２−オキソピリジン−３−イルチア（ジ）アゾール誘導体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6296479A (ja) * 1985-10-23 1987-05-02 Shionogi & Co Ltd ポリフルオロアルキルイソオキサゾリルアミン類
JPH08193067A (ja) * 1994-02-14 1996-07-30 Nippon Soda Co Ltd ピラゾール化合物、製法、農園芸用殺菌剤および殺虫・殺ダニ剤
WO2003014067A1 (en) * 2001-08-02 2003-02-20 Ube Industries, Ltd. PROCESS FOR PRODUCING ß-OXONITRILE COMPOUND OR ALKALI METAL SALT THEREOF
DE10349500A1 (de) * 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
US7884216B2 (en) * 2007-02-20 2011-02-08 Mitsui Chemicals Agro, Inc. Fluorine-containing pyrazolecarbonitrile derivative and method for producing the same, and fluorine-containing pyrazolecarboxylic acid derivative obtained by using the fluorine-containing pyrazolecarbonitrile derivative and method for producing the same

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966791A (en) 1974-06-19 1976-06-29 Hoffmann-La Roche Inc. Preparation of dialkyl amino acrylonitrile
JPS55130950A (en) 1979-03-29 1980-10-11 Dynamit Nobel Ag Betaaalkoxyyacrylonitrile*33aminooacryonitrile and 22cyanoovinylester manufacture
JPS63264448A (ja) * 1988-02-29 1988-11-01 Shionogi & Co Ltd 新規β−ケトニトリル
JP2003113153A (ja) * 2001-08-02 2003-04-18 Ube Ind Ltd β−オキソニトリル誘導体又はそのアルカリ金属塩の製法
JP2005511782A (ja) 2001-12-17 2005-04-28 バイエル ケミカルズ アクチエンゲゼルシャフト ２−ハロゲンアシル−３−アミノ−アクリル酸−誘導体の製造方法
JP2003267943A (ja) * 2002-03-15 2003-09-25 Fuji Photo Film Co Ltd ジシアノメチリデン化合物及びヘテロ環化合物の合成方法
JP2006514059A (ja) 2002-12-27 2006-04-27 アムゲン インコーポレイテッド 細胞増殖及びアポトーシスに関連する疾患の処置に使用する２−オキソピリジン−３−イルチア（ジ）アゾール誘導体

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
DATABASE REGISTRY [online] 30 May 2001 (2001-05-30), XP008111822, accession no. STN Database accession no. (339011-85-7) *
MAHALANABIS K.K. ET AL.: "Studies on beta-enaminonitriles: Part IV - Reaction of beta-enaminonitriles with acid chlorides", INDIAN JOURNAL OF CHEMISTRY, vol. 41B, no. 9, 2002, pages 1902 - 1906, XP008110467 *
See also references of EP2105434A4

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010540477A (ja) * 2007-09-26 2010-12-24 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト ２−ジハロアシル−３−アミノアクリル酸誘導体の調製方法
WO2012065905A1 (en) 2010-11-15 2012-05-24 Bayer Cropscience Ag Cyanoenamines and their use as fungicides
US9351489B2 (en) 2010-11-15 2016-05-31 Bayer Intellectual Property Gmbh Cyanoenamines and their use as fungicides

Also Published As

Publication number Publication date
EP2105434A4 (en) 2012-02-29
EP2105434A1 (en) 2009-09-30
RU2009124415A (ru) 2011-02-10
CN101627008A (zh) 2010-01-13
JPWO2008081711A1 (ja) 2010-04-30
AU2007340689A1 (en) 2008-07-10
TW200837041A (en) 2008-09-16
MX2009007029A (es) 2009-11-09
US20100010216A1 (en) 2010-01-14
BRPI0720715A2 (pt) 2014-04-01

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