WO2002089734A2 - Methode de traitement et de prevention de troubles du systeme nerveux central associes a une alteration de la neurotransmission glutamatergique par administration de derives de 2-aminobenzenesulfonamide - Google Patents
Methode de traitement et de prevention de troubles du systeme nerveux central associes a une alteration de la neurotransmission glutamatergique par administration de derives de 2-aminobenzenesulfonamide Download PDFInfo
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- WO2002089734A2 WO2002089734A2 PCT/US2002/014262 US0214262W WO02089734A2 WO 2002089734 A2 WO2002089734 A2 WO 2002089734A2 US 0214262 W US0214262 W US 0214262W WO 02089734 A2 WO02089734 A2 WO 02089734A2
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- A61K31/18—Sulfonamides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/136—Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
Abstract
L'invention porte sur des dérivés de 2-aminobenzènesulfonamide utilisés pour le traitement ou la prévention de troubles du système nerveux central associés à une modulation positive ou négative de la neurotransmission glutamatergique, notamment des troubles de la mémoire et de l'apprentissage, de la schizophrénie, des dysfonctionnements sexuels, d'attaques ischémiques, d'ictus, etc. A titre d'exemple, un composé de formule I est administré afin de traiter ou de prévenir des maladies du système nerveux central présentant une modulation positive ou négative des récepteurs AMPA-Kainate et une modulation négative des récepteurs NMDA.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02769353A EP1435926A4 (fr) | 2001-05-08 | 2002-05-07 | Methode de traitement et de prevention de troubles du systeme nerveux central associes a une alteration de la neurotransmission glutamatergique par administration de derives de 2-aminobenzenesulfonamide |
| AU2002308614A AU2002308614A1 (en) | 2001-05-08 | 2002-05-07 | Method for treatment and prevention of disturbances of the central nervous system associated with an alteration of glutamatergic neurotransmission by administration of 2-aminobenzenesulfonamide derivatives |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITBO2001A000271 | 2001-05-08 | ||
| IT2001BO000271A ITBO20010271A1 (it) | 2001-05-08 | 2001-05-08 | Metodo per il trattamento e la prevenzione dei disturbi del sistema nervoso centrale associati ad una alterazione della neurotrasmissione gl |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2002089734A2 true WO2002089734A2 (fr) | 2002-11-14 |
| WO2002089734A3 WO2002089734A3 (fr) | 2003-03-06 |
Family
ID=11439316
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/US2002/014262 WO2002089734A2 (fr) | 2001-05-08 | 2002-05-07 | Methode de traitement et de prevention de troubles du systeme nerveux central associes a une alteration de la neurotransmission glutamatergique par administration de derives de 2-aminobenzenesulfonamide |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP1435926A4 (fr) |
| AU (1) | AU2002308614A1 (fr) |
| IT (1) | ITBO20010271A1 (fr) |
| WO (1) | WO2002089734A2 (fr) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007076875A2 (fr) * | 2006-01-06 | 2007-07-12 | Aarhus Universitet | Composes agissant sur le transporteur de la serotonine |
| US7297713B2 (en) | 2005-07-29 | 2007-11-20 | Wyeth | Cyanopyrrole-phenyl amide progesterone receptor modulators and uses thereof |
| EP3311842A1 (fr) | 2013-06-13 | 2018-04-25 | VeroScience LLC | Compositions et procédés de traitement des troubles métaboliques |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5536719A (en) * | 1994-07-12 | 1996-07-16 | Adir Et Compagnie | Benzothiadiazine compound |
| US6083947A (en) * | 1996-01-29 | 2000-07-04 | The Regents Of The University Of California | Method for treating sexual dysfunctions |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5939451A (en) * | 1996-06-28 | 1999-08-17 | Hoffmann-La Roche Inc. | Use of sulfonamides |
| GB9818916D0 (en) * | 1998-08-28 | 1998-10-21 | Smithkline Beecham Plc | Use |
-
2001
- 2001-05-08 IT IT2001BO000271A patent/ITBO20010271A1/it unknown
-
2002
- 2002-05-07 AU AU2002308614A patent/AU2002308614A1/en not_active Abandoned
- 2002-05-07 WO PCT/US2002/014262 patent/WO2002089734A2/fr not_active Application Discontinuation
- 2002-05-07 EP EP02769353A patent/EP1435926A4/fr not_active Withdrawn
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5536719A (en) * | 1994-07-12 | 1996-07-16 | Adir Et Compagnie | Benzothiadiazine compound |
| US6083947A (en) * | 1996-01-29 | 2000-07-04 | The Regents Of The University Of California | Method for treating sexual dysfunctions |
Non-Patent Citations (1)
| Title |
|---|
| See also references of EP1435926A2 * |
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7297713B2 (en) | 2005-07-29 | 2007-11-20 | Wyeth | Cyanopyrrole-phenyl amide progesterone receptor modulators and uses thereof |
| US7652062B2 (en) | 2005-07-29 | 2010-01-26 | Wyeth Llc | Cyanopyrrole-phenyl amide progesterone receptor modulators and uses thereof |
| WO2007076875A2 (fr) * | 2006-01-06 | 2007-07-12 | Aarhus Universitet | Composes agissant sur le transporteur de la serotonine |
| WO2007076875A3 (fr) * | 2006-01-06 | 2007-11-15 | Univ Aarhus | Composes agissant sur le transporteur de la serotonine |
| EP3311842A1 (fr) | 2013-06-13 | 2018-04-25 | VeroScience LLC | Compositions et procédés de traitement des troubles métaboliques |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2002308614A1 (en) | 2002-11-18 |
| ITBO20010271A1 (it) | 2002-11-08 |
| WO2002089734A3 (fr) | 2003-03-06 |
| ITBO20010271A0 (it) | 2001-05-08 |
| EP1435926A4 (fr) | 2005-11-23 |
| EP1435926A2 (fr) | 2004-07-14 |
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