WO2000014098A1 - Methods for the preparation of conjugated oligomers - Google Patents

Methods for the preparation of conjugated oligomers Download PDF

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Publication number
WO2000014098A1
WO2000014098A1 PCT/US1999/019828 US9919828W WO0014098A1 WO 2000014098 A1 WO2000014098 A1 WO 2000014098A1 US 9919828 W US9919828 W US 9919828W WO 0014098 A1 WO0014098 A1 WO 0014098A1
Authority
WO
WIPO (PCT)
Prior art keywords
compound
formula
alkyl
oligonucleotide
group
Prior art date
Application number
PCT/US1999/019828
Other languages
English (en)
French (fr)
Inventor
Muthiah Manoharan
Original Assignee
Isis Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Isis Pharmaceuticals, Inc. filed Critical Isis Pharmaceuticals, Inc.
Priority to EP99942546A priority Critical patent/EP1112279A4/en
Priority to AU55899/99A priority patent/AU5589999A/en
Publication of WO2000014098A1 publication Critical patent/WO2000014098A1/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PCT/US1999/019828 1998-09-07 1999-08-27 Methods for the preparation of conjugated oligomers WO2000014098A1 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
EP99942546A EP1112279A4 (en) 1998-09-07 1999-08-27 METHOD FOR THE PRODUCTION OF CONJUGATED OLIGOMERS
AU55899/99A AU5589999A (en) 1998-09-07 1999-08-27 Methods for the preparation of conjugated oligomers

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/149,156 1998-09-07
US09/149,156 US6335437B1 (en) 1998-09-07 1998-09-07 Methods for the preparation of conjugated oligomers

Publications (1)

Publication Number Publication Date
WO2000014098A1 true WO2000014098A1 (en) 2000-03-16

Family

ID=22529021

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US1999/019828 WO2000014098A1 (en) 1998-09-07 1999-08-27 Methods for the preparation of conjugated oligomers

Country Status (4)

Country Link
US (1) US6335437B1 (US06335437-20020101-C00041.png)
EP (1) EP1112279A4 (US06335437-20020101-C00041.png)
AU (1) AU5589999A (US06335437-20020101-C00041.png)
WO (1) WO2000014098A1 (US06335437-20020101-C00041.png)

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Also Published As

Publication number Publication date
AU5589999A (en) 2000-03-27
US6335437B1 (en) 2002-01-01
EP1112279A1 (en) 2001-07-04
EP1112279A4 (en) 2002-06-19

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