WO1981000405A1 - Di-cyano-guanidines - Google Patents

Di-cyano-guanidines Download PDF

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Publication number
WO1981000405A1
WO1981000405A1 PCT/CH1980/000091 CH8000091W WO8100405A1 WO 1981000405 A1 WO1981000405 A1 WO 1981000405A1 CH 8000091 W CH8000091 W CH 8000091W WO 8100405 A1 WO8100405 A1 WO 8100405A1
Authority
WO
WIPO (PCT)
Prior art keywords
cyano
methyl
que
ethyl
dans
Prior art date
Application number
PCT/CH1980/000091
Other languages
German (de)
English (en)
Inventor
P Baudet
Original Assignee
Rech Syntheses Organ
P Baudet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rech Syntheses Organ, P Baudet filed Critical Rech Syntheses Organ
Publication of WO1981000405A1 publication Critical patent/WO1981000405A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
    • C07C323/43—Y being a hetero atom
    • C07C323/44—X or Y being nitrogen atoms

Definitions

  • IR (nujol): 3470, 3230, 3150, 2700, 2600, 2170, 1610, 160 1650, 1500, 1345, (double) 1295, 1280, 1240, 1220, 1180, 1120 (double) 1085, 1050, 955, 900 , 860, 750 (epaul.), 725 cm -1 .

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Di-cyano-guanidines de formule: (FORMULE) dans laquelle (FORMULE) et plusieurs procedes de leur preparation. Le compose (b) possede une activite antihistaminique.
PCT/CH1980/000091 1979-07-30 1980-07-29 Di-cyano-guanidines WO1981000405A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH6994/79 1979-07-30
CH699479 1979-07-30

Publications (1)

Publication Number Publication Date
WO1981000405A1 true WO1981000405A1 (fr) 1981-02-19

Family

ID=4318265

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/CH1980/000091 WO1981000405A1 (fr) 1979-07-30 1980-07-29 Di-cyano-guanidines

Country Status (3)

Country Link
EP (1) EP0032916A1 (fr)
JP (1) JPS56501008A (fr)
WO (1) WO1981000405A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20230349922A1 (en) 2020-08-11 2023-11-02 Université De Strasbourg H2 Blockers Targeting Liver Macrophages for the Prevention and Treatment of Liver Disease and Cancer

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1979000466A1 (fr) * 1977-12-30 1979-07-26 Crc Ricerca Chim Procede d'alkylation du 4(5)-mercaptomethyl-imidazole avec des derives d'aziridine

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1979000466A1 (fr) * 1977-12-30 1979-07-26 Crc Ricerca Chim Procede d'alkylation du 4(5)-mercaptomethyl-imidazole avec des derives d'aziridine

Also Published As

Publication number Publication date
EP0032916A1 (fr) 1981-08-05
JPS56501008A (fr) 1981-07-23

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