UY32975A - AMINOPIRIDINE DERIVATIVES - Google Patents

AMINOPIRIDINE DERIVATIVES

Info

Publication number
UY32975A
UY32975A UY0001032975A UY32975A UY32975A UY 32975 A UY32975 A UY 32975A UY 0001032975 A UY0001032975 A UY 0001032975A UY 32975 A UY32975 A UY 32975A UY 32975 A UY32975 A UY 32975A
Authority
UY
Uruguay
Prior art keywords
aminopiridine
derivatives
compounds
copd
asthma
Prior art date
Application number
UY0001032975A
Other languages
Spanish (es)
Inventor
David Michael Evans
Christine Elizabeth Allan
Original Assignee
Vantia Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vantia Ltd filed Critical Vantia Ltd
Publication of UY32975A publication Critical patent/UY32975A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/73Unsubstituted amino or imino radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

La presente invención proporciona compuestos de fórmula (I), composiciones que comprenden dichos compuestos; el uso de dichos compuestos en terapia (tal como asma o EPOC); y métodos para tratar pacientes con tales compuestos; en donde R1 ? R10 y A1 son tal como se definen en la presente.The present invention provides compounds of formula (I), compositions comprising said compounds; the use of said compounds in therapy (such as asthma or COPD); and methods for treating patients with such compounds; where R1? R10 and A1 are as defined herein.

UY0001032975A 2009-10-28 2010-10-27 AMINOPIRIDINE DERIVATIVES UY32975A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25560609P 2009-10-28 2009-10-28
GBGB0918922.6A GB0918922D0 (en) 2009-10-28 2009-10-28 Aminopyridine derivatives

Publications (1)

Publication Number Publication Date
UY32975A true UY32975A (en) 2011-05-31

Family

ID=41434814

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032975A UY32975A (en) 2009-10-28 2010-10-27 AMINOPIRIDINE DERIVATIVES

Country Status (5)

Country Link
AR (1) AR078817A1 (en)
GB (1) GB0918922D0 (en)
TW (1) TW201119654A (en)
UY (1) UY32975A (en)
WO (1) WO2011051671A1 (en)

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US9409880B2 (en) 2011-01-20 2016-08-09 The Regents Of The University Of Colorado, A Body Corporate Modulators of TLR3/dsRNA complex and uses thereof
GB2510407A (en) * 2013-02-04 2014-08-06 Kalvista Pharmaceuticals Ltd Aqueous suspensions of kallikrein inhibitors for parenteral administration
JP2016152772A (en) * 2013-06-27 2016-08-25 味の素株式会社 Novel umami-taste imparting agent
WO2020094008A1 (en) * 2018-11-06 2020-05-14 天津药物研究院有限公司 2-oxo-1,2-dihydroquinoline derivatives, preparation method therefor, and pharmaceutical applications thereof
EP4010333A1 (en) 2019-08-09 2022-06-15 Kalvista Pharmaceuticals Limited Plasma kallikrein inhibitors

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Also Published As

Publication number Publication date
TW201119654A (en) 2011-06-16
AR078817A1 (en) 2011-12-07
GB0918922D0 (en) 2009-12-16
WO2011051671A1 (en) 2011-05-05

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Effective date: 20121113