UY30171A1 - Formas cristalinas de n- (benzo (b) tien-3-ilmetil) -sulfamida - Google Patents
Formas cristalinas de n- (benzo (b) tien-3-ilmetil) -sulfamidaInfo
- Publication number
- UY30171A1 UY30171A1 UY30171A UY30171A UY30171A1 UY 30171 A1 UY30171 A1 UY 30171A1 UY 30171 A UY30171 A UY 30171A UY 30171 A UY30171 A UY 30171A UY 30171 A1 UY30171 A1 UY 30171A1
- Authority
- UY
- Uruguay
- Prior art keywords
- benzo
- sulfamida
- ilmetil
- tien
- crystal forms
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/58—Radicals substituted by nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invencinn se refiere a formas cristalinas, anhidras y solvatadas de N-(benzo(b)tien-3-(ilmetil)-sulfamida, composiciones farmaccuticas que contienen dichas formas cristalinas y su utilizacinn en el tratamiento de la epilepsia y trastornos relacionados.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US77572406P | 2006-02-22 | 2006-02-22 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30171A1 true UY30171A1 (es) | 2007-07-31 |
Family
ID=38066512
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30171A UY30171A1 (es) | 2006-02-22 | 2007-02-22 | Formas cristalinas de n- (benzo (b) tien-3-ilmetil) -sulfamida |
Country Status (6)
Country | Link |
---|---|
US (1) | US20070232685A1 (es) |
AR (1) | AR059596A1 (es) |
PE (1) | PE20071016A1 (es) |
TW (1) | TW200738669A (es) |
UY (1) | UY30171A1 (es) |
WO (1) | WO2007098486A1 (es) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY147767A (en) | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
JP2008545650A (ja) | 2005-05-20 | 2008-12-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | スルファミド誘導体の製造方法 |
US8497298B2 (en) | 2005-12-19 | 2013-07-30 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels |
US8691867B2 (en) | 2005-12-19 | 2014-04-08 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction |
US8937096B2 (en) | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
EA200870556A1 (ru) | 2006-05-19 | 2009-06-30 | Янссен Фармацевтика Н.В. | Комбинированная терапия в лечении эпилепсии и родственных расстройств |
CA2696253A1 (en) | 2007-08-08 | 2009-02-12 | Janssen Pharmaceutica Nv | Sulfamide derivative useful for the treatment of epilepsy |
US20090247616A1 (en) * | 2008-03-26 | 2009-10-01 | Smith-Swintosky Virginia L | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety |
US20090247617A1 (en) * | 2008-03-26 | 2009-10-01 | Abdel-Magid Ahmed F | Process for the preparation of benzo-fused heteroaryl sulfamates |
WO2009120191A1 (en) * | 2008-03-26 | 2009-10-01 | Janssen Pharmaceutica N.V. | Process for the preparation of benzo-fused heteroaryl sulfamates and crystalline form of n- ( ( (2s) -6-chloro-2,3-dihydro-l,4-benzodioxin-2-yl) methyl-sulfamide |
NZ590682A (en) | 2008-06-23 | 2012-09-28 | Janssen Pharmaceutica Nv | Crystalline form of (2S)-(-)-N-(6-chloro-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-sulfamide |
US8815939B2 (en) * | 2008-07-22 | 2014-08-26 | Janssen Pharmaceutica Nv | Substituted sulfamide derivatives |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4513006A (en) * | 1983-09-26 | 1985-04-23 | Mcneil Lab., Inc. | Anticonvulsant sulfamate derivatives |
WO1997019682A1 (en) * | 1995-12-01 | 1997-06-05 | Synaptic Pharmaceutical Corporation | Aryl sulfonamide and sulfamide derivatives and uses thereof |
WO2002096424A1 (en) * | 2001-05-25 | 2002-12-05 | Queen's University At Kingston | Hetereocyclic beta-aminoacids and their use as anti-epileptogenic agents |
US20030047001A1 (en) * | 2001-08-28 | 2003-03-13 | Grace Liao | Ball speed detecting assembly |
CN1897950A (zh) * | 2003-10-14 | 2007-01-17 | 惠氏公司 | 稠合芳基和杂芳基衍生物及其使用方法 |
TW200612905A (en) * | 2004-06-16 | 2006-05-01 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
AU2005277134A1 (en) * | 2004-08-24 | 2006-03-02 | Janssen Pharmaceutica N.V. | Novel benzo-fused heteroaryl sulfamide derivatives useful as anticonvulsant agents |
JP2008545650A (ja) * | 2005-05-20 | 2008-12-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | スルファミド誘導体の製造方法 |
-
2007
- 2007-02-16 TW TW096105901A patent/TW200738669A/zh unknown
- 2007-02-20 PE PE2007000186A patent/PE20071016A1/es not_active Application Discontinuation
- 2007-02-21 AR ARP070100730A patent/AR059596A1/es not_active Application Discontinuation
- 2007-02-22 WO PCT/US2007/062564 patent/WO2007098486A1/en active Application Filing
- 2007-02-22 UY UY30171A patent/UY30171A1/es unknown
- 2007-02-22 US US11/677,717 patent/US20070232685A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AR059596A1 (es) | 2008-04-16 |
TW200738669A (en) | 2007-10-16 |
US20070232685A1 (en) | 2007-10-04 |
WO2007098486A1 (en) | 2007-08-30 |
PE20071016A1 (es) | 2007-10-24 |
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