UA93489C2 - Гетероциклические соединения kak антагонисты ccr2b - Google Patents

Гетероциклические соединения kak антагонисты ccr2b

Info

Publication number
UA93489C2
UA93489C2 UAA200706266A UAA200706266A UA93489C2 UA 93489 C2 UA93489 C2 UA 93489C2 UA A200706266 A UAA200706266 A UA A200706266A UA A200706266 A UAA200706266 A UA A200706266A UA 93489 C2 UA93489 C2 UA 93489C2
Authority
UA
Ukraine
Prior art keywords
heterocyclic compounds
formula
yand
alkyl
ccr2b
Prior art date
Application number
UAA200706266A
Other languages
English (en)
Ukrainian (uk)
Inventor
Джастин Ферфилд Бауэр
Джеффри Филип Пойзер
Пол Тернер
Дейвид Вотерсон
Джон Винтер
Original Assignee
Астразенека Аб
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Астразенека Аб filed Critical Астразенека Аб
Publication of UA93489C2 publication Critical patent/UA93489C2/ru

Links

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Соединения формулы (I)(I)и их фармацевтически приемлемые соли или сольваты, которые являются полезными в лечении опосредованных хемокином С-С состояний.
UAA200706266A 2004-12-24 2005-12-19 Гетероциклические соединения kak антагонисты ccr2b UA93489C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB0428327A GB0428327D0 (en) 2004-12-24 2004-12-24 Method

Publications (1)

Publication Number Publication Date
UA93489C2 true UA93489C2 (ru) 2011-02-25

Family

ID=34130900

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200706266A UA93489C2 (ru) 2004-12-24 2005-12-19 Гетероциклические соединения kak антагонисты ccr2b

Country Status (4)

Country Link
CN (1) CN101128427B (ru)
GB (1) GB0428327D0 (ru)
UA (1) UA93489C2 (ru)
ZA (1) ZA200705159B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100152197A1 (en) * 2008-12-15 2010-06-17 Astrazeneca Ab (4-tert-butylpiperazin-2-yl)(piperazin-1-yl)methanone-n-carboxamide derivatives
MX2022002720A (es) * 2019-09-05 2022-08-10 Lunan Pharmaceutical Group Corp Inhibidor de magl, procedimiento de preparacion y uso del mismo.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07502014A (ja) * 1991-06-21 1995-03-02 ベーリンガー マンハイム イタリア エス.ピー.エイ. 気道に対して抗喘息性、抗炎症性活性を有する2−アミノ−4−アリール−チアゾール
EP1334089A1 (en) * 2000-11-13 2003-08-13 GlaxoSmithKline S.p.A. Quinoline derivatives as nk-3 and nk-2 antagonists
GB0031088D0 (en) * 2000-12-20 2001-01-31 Smithkline Beecham Plc Medicaments
WO2002079151A1 (en) * 2001-03-29 2002-10-10 Smithkline Beecham P.L.C. 3-substituted indoels or fused pyrroles as antagonists of the chemokine mcp-1 (ccr2b) receptor
CA2502178A1 (en) * 2002-10-30 2004-05-21 Merck & Co., Inc. Heteroarylpiperidine modulators of chemokine receptor activity
FR2872813B1 (fr) * 2004-07-09 2007-01-19 Sanofi Synthelabo Derives de 2-carbamide-4-phenylthiazole, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
CN101128427B (zh) 2013-03-27
ZA200705159B (en) 2008-06-25
CN101128427A (zh) 2008-02-20
GB0428327D0 (en) 2005-02-02

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