UA93348C2 - Индазолы, бензотиазолы, бензоизотиазолы, их получение и применение - Google Patents
Индазолы, бензотиазолы, бензоизотиазолы, их получение и применениеInfo
- Publication number
- UA93348C2 UA93348C2 UAA200611224A UAA200611224A UA93348C2 UA 93348 C2 UA93348 C2 UA 93348C2 UA A200611224 A UAA200611224 A UA A200611224A UA A200611224 A UAA200611224 A UA A200611224A UA 93348 C2 UA93348 C2 UA 93348C2
- Authority
- UA
- Ukraine
- Prior art keywords
- indazoles
- benzothiazoles
- receptors
- nach
- benzoisothiazoles
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Данное изобретение в целом касается области лигандов никотиновых ацетилхолиновых рецепторов (рецепторов nACh), активации рецепторов nACh и лечения патологических состояний, связанных с дефектными или неправильно функционирующими никотиновыми ацетилхолиновыми рецепторами, особенно в головном мозге. Кроме того, в заявке описаны соединения (например, индазолы и бензотиазолы), которые действуют как лиганды для подтипа (7 рецепторов nACh, способы получения таких соединений и их применение.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US55595104P | 2004-03-25 | 2004-03-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
UA93348C2 true UA93348C2 (ru) | 2011-02-10 |
Family
ID=38693326
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200611224A UA93348C2 (ru) | 2004-03-25 | 2005-03-25 | Индазолы, бензотиазолы, бензоизотиазолы, их получение и применение |
Country Status (4)
Country | Link |
---|---|
CN (1) | CN101001856A (ru) |
TN (1) | TNSN06301A1 (ru) |
UA (1) | UA93348C2 (ru) |
ZA (1) | ZA200608812B (ru) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JOP20130213B1 (ar) | 2012-07-17 | 2021-08-17 | Takeda Pharmaceuticals Co | معارضات لمستقبلht3-5 |
PL3201203T3 (pl) | 2014-09-29 | 2021-11-22 | Takeda Pharmaceutical Company Limited | Krystaliczna postać 1-(1-metylo-1h-pirazol-4-ilo)-n-((1r,5s,7s)-9-metylo-3-oksa-9-azabicyklo[3.3.1]nonan-7-ylo)-1h-indolo-3-karboksyamidu |
CN110582500B (zh) * | 2017-05-04 | 2022-04-05 | 上海长森药业有限公司 | 双并环类核衣壳抑制剂和其作为药物用于治疗乙型肝炎的用途 |
BR112020017087A2 (pt) | 2018-02-23 | 2020-12-22 | Samumed, Llc | Indazol-3-carboxamidas substituídas 5-heteroarila e preparação e uso das mesmas |
CN110437132B (zh) * | 2018-05-04 | 2022-04-01 | 上海长森药业有限公司 | 双并杂环核衣壳抑制剂及其药物用途 |
CN114605329B (zh) * | 2022-03-28 | 2024-01-26 | 河南中医药大学 | 取代的吲唑甲酰胺或取代的氮杂吲唑甲酰胺类flt3抑制剂及其用途 |
-
2005
- 2005-03-25 UA UAA200611224A patent/UA93348C2/ru unknown
- 2005-03-25 CN CN 200580016742 patent/CN101001856A/zh active Pending
-
2006
- 2006-09-22 TN TNP2006000301A patent/TNSN06301A1/en unknown
- 2006-10-23 ZA ZA200608812A patent/ZA200608812B/en unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200608812B (en) | 2008-04-30 |
TNSN06301A1 (en) | 2007-12-03 |
CN101001856A (zh) | 2007-07-18 |
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