UA81281C2 - Avermectin derivatives, pesticide composition and method of pest control - Google Patents

Avermectin derivatives, pesticide composition and method of pest control Download PDF

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Publication number
UA81281C2
UA81281C2 UAA200507209A UA2005007209A UA81281C2 UA 81281 C2 UA81281 C2 UA 81281C2 UA A200507209 A UAA200507209 A UA A200507209A UA 2005007209 A UA2005007209 A UA 2005007209A UA 81281 C2 UA81281 C2 UA 81281C2
Authority
UA
Ukraine
Prior art keywords
alkyl
heterocyclyl
aryl
formula
group
Prior art date
Application number
UAA200507209A
Other languages
English (en)
Ukrainian (uk)
Inventor
Peter Maienfisch
Thomas Pitterna
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of UA81281C2 publication Critical patent/UA81281C2/uk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/22Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Biotechnology (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
UAA200507209A 2002-12-20 2003-12-19 Avermectin derivatives, pesticide composition and method of pest control UA81281C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0229804.0A GB0229804D0 (en) 2002-12-20 2002-12-20 Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
PCT/EP2003/014613 WO2004056844A1 (en) 2002-12-20 2003-12-19 Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4”- or 4’-position

Publications (1)

Publication Number Publication Date
UA81281C2 true UA81281C2 (en) 2007-12-25

Family

ID=9950151

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200507209A UA81281C2 (en) 2002-12-20 2003-12-19 Avermectin derivatives, pesticide composition and method of pest control

Country Status (22)

Country Link
US (3) US7737261B2 (es)
EP (1) EP1581546B1 (es)
JP (2) JP4851094B2 (es)
KR (1) KR101109500B1 (es)
CN (1) CN1738828B (es)
AR (1) AR042533A1 (es)
AU (1) AU2003302284B2 (es)
BR (1) BR0317601A (es)
CA (1) CA2507774C (es)
CO (1) CO5690647A1 (es)
ES (1) ES2742899T3 (es)
GB (1) GB0229804D0 (es)
IL (1) IL169092A (es)
MA (1) MA27646A1 (es)
MX (1) MXPA05006036A (es)
PE (1) PE20040713A1 (es)
PL (1) PL211483B1 (es)
RU (1) RU2330857C2 (es)
TW (1) TW200512214A (es)
UA (1) UA81281C2 (es)
WO (1) WO2004056844A1 (es)
ZA (1) ZA200504353B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0229804D0 (en) * 2002-12-20 2003-01-29 Syngenta Participations Ag Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position
JP2010006703A (ja) * 2006-11-07 2010-01-14 Hokko Chem Ind Co Ltd アベルメクチンモノ配糖体誘導体
RU2453553C1 (ru) * 2011-05-11 2012-06-20 Игорь Викторович Заварзин 5-о-сукциноилавермектин, способ его получения и антипаразитарное средство на его основе
RU2472801C1 (ru) * 2011-05-11 2013-01-20 Игорь Викторович Заварзин 5-о-производные авермектина, способ их получения и антипаразитарные средства на их основе
CN103613625B (zh) * 2013-12-02 2016-03-02 兰州大学 一种阿维菌素类化合物及其制备方法和在农药中的用途
CN104402953B (zh) * 2014-11-28 2017-07-28 大庆志飞生物化工有限公司 阿维菌素单糖化合物及其制备方法和用途
CN104402954A (zh) * 2014-11-28 2015-03-11 大庆志飞生物化工有限公司 甲胺基阿维菌素单糖化合物及其制备方法和用途
JP6577184B2 (ja) 2014-12-24 2019-09-18 Ntn株式会社 転がり軸受
CN107501368B (zh) * 2017-09-30 2020-02-21 中国科学院成都生物研究所 一种多拉菌素衍生物的合成及其杀虫应用
CN113150053B (zh) * 2020-01-22 2024-10-01 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用
CN113817008B (zh) * 2021-07-15 2023-05-23 湖州师范学院 新型琥珀酰基十六元大环内酯的制备方法及用途

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US18993A (en) * 1857-12-29 Cider-mill
US87519A (en) * 1869-03-02 Improvement in furnace-stoves and registers
US148520A (en) * 1874-03-10 Improvement in faucets
SE434277B (sv) 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
GB8811037D0 (en) 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
EP0353959A2 (en) 1988-08-02 1990-02-07 Beecham Group Plc Antihelmintic macrolide antibiotics
SE465605B (sv) * 1990-02-26 1991-10-07 Harry Nilsson Skivfilter
JP2622197B2 (ja) 1990-03-01 1997-06-18 三共株式会社 13−エーテル置換ミルベマイシン誘導体
US5169839A (en) 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5262400A (en) * 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
US5411737A (en) 1991-10-15 1995-05-02 Merck & Co., Inc. Slow release syneresing polymeric drug delivery device
PL174488B1 (pl) 1993-05-10 1998-08-31 Merck & Co Inc Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt
US5602107A (en) 1993-05-10 1997-02-11 Merck & Co., Inc. Pour-on formulations consisting of gylcols, glycerides and avermectin compounds
US5436355A (en) 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
AU2001278694A1 (en) 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
AU2001277712A1 (en) 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
CA2477614A1 (en) * 2002-03-05 2003-09-18 Merck & Co., Inc. Biomarker for efficacy of appetite suppressant drugs
GB0229804D0 (en) * 2002-12-20 2003-01-29 Syngenta Participations Ag Avermection b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substituent in the 4"- or 4'-position

Also Published As

Publication number Publication date
JP2011102303A (ja) 2011-05-26
RU2330857C2 (ru) 2008-08-10
US8017589B2 (en) 2011-09-13
JP5302297B2 (ja) 2013-10-02
RU2005122943A (ru) 2006-01-20
KR101109500B1 (ko) 2012-01-31
US8263566B2 (en) 2012-09-11
CA2507774C (en) 2011-06-14
IL169092A (en) 2010-12-30
MA27646A1 (fr) 2005-12-01
WO2004056844A1 (en) 2004-07-08
IL169092A0 (en) 2007-07-04
AU2003302284A1 (en) 2004-07-14
GB0229804D0 (en) 2003-01-29
BR0317601A (pt) 2005-11-29
CN1738828A (zh) 2006-02-22
AR042533A1 (es) 2005-06-22
EP1581546B1 (en) 2019-03-20
US20060148729A1 (en) 2006-07-06
JP4851094B2 (ja) 2012-01-11
MXPA05006036A (es) 2005-08-18
CN1738828B (zh) 2012-09-05
PL377497A1 (pl) 2006-02-06
ZA200504353B (en) 2006-03-29
KR20050088133A (ko) 2005-09-01
AU2003302284B2 (en) 2009-07-23
PE20040713A1 (es) 2004-12-02
US7737261B2 (en) 2010-06-15
PL211483B1 (pl) 2012-05-31
TW200512214A (en) 2005-04-01
US20100210574A1 (en) 2010-08-19
US20110230429A1 (en) 2011-09-22
JP2006515849A (ja) 2006-06-08
CO5690647A1 (es) 2006-10-31
CA2507774A1 (en) 2004-07-08
EP1581546A1 (en) 2005-10-05
ES2742899T3 (es) 2020-02-17

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