TWI694825B - 用於長效可注射帕里皮酮（ｐａｌｉｐｅｒｉｄｏｎｅ）酯類遺漏劑量之投藥療程 - Google Patents
用於長效可注射帕里皮酮（ｐａｌｉｐｅｒｉｄｏｎｅ）酯類遺漏劑量之投藥療程 Download PDFInfo
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- Medicinal Chemistry (AREA)
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- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
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- Biomedical Technology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Inorganic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Pain & Pain Management (AREA)
- Molecular Biology (AREA)
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- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562144054P | 2015-04-07 | 2015-04-07 | |
| US62/144,054 | 2015-04-07 | ||
| US201562162596P | 2015-05-15 | 2015-05-15 | |
| US62/162,596 | 2015-05-15 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TW201642863A TW201642863A (zh) | 2016-12-16 |
| TWI694825B true TWI694825B (zh) | 2020-06-01 |
Family
ID=57072843
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW105110443A TWI694825B (zh) | 2015-04-07 | 2016-04-01 | 用於長效可注射帕里皮酮（ｐａｌｉｐｅｒｉｄｏｎｅ）酯類遺漏劑量之投藥療程 |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US10143693B2 (OSRAM) |
| EP (3) | EP4349323A3 (OSRAM) |
| JP (3) | JP6728221B2 (OSRAM) |
| KR (3) | KR102755145B1 (OSRAM) |
| AU (4) | AU2016244801B2 (OSRAM) |
| BR (1) | BR112017021383A2 (OSRAM) |
| CA (2) | CA3088401A1 (OSRAM) |
| CY (1) | CY1123203T1 (OSRAM) |
| DK (2) | DK3280416T3 (OSRAM) |
| EA (1) | EA037185B1 (OSRAM) |
| ES (2) | ES2802299T3 (OSRAM) |
| FI (1) | FI3744326T3 (OSRAM) |
| HR (2) | HRP20240022T1 (OSRAM) |
| HU (2) | HUE049485T2 (OSRAM) |
| IL (3) | IL254669B2 (OSRAM) |
| LT (2) | LT3280416T (OSRAM) |
| MA (1) | MA41917B1 (OSRAM) |
| MD (2) | MD3280416T2 (OSRAM) |
| NZ (1) | NZ735952A (OSRAM) |
| PL (2) | PL3280416T3 (OSRAM) |
| PT (2) | PT3744326T (OSRAM) |
| RS (2) | RS65024B1 (OSRAM) |
| SI (2) | SI3280416T1 (OSRAM) |
| SM (2) | SMT202000351T1 (OSRAM) |
| TW (1) | TWI694825B (OSRAM) |
| UA (1) | UA118732C2 (OSRAM) |
| WO (1) | WO2016164218A1 (OSRAM) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2802299T3 (es) | 2015-04-07 | 2021-01-18 | Janssen Pharmaceuticals Inc | Régimen de dosificación para dosis olvidadas para ésteres de paliperidona inyectables de acción prolongada |
| CA3077224A1 (en) | 2017-10-27 | 2019-05-02 | Shandong Luye Pharmaceutical Co., Ltd. | Dosage regimen of paliperidone palmitate extended-release injectable suspension |
| EP4385564A3 (en) * | 2020-11-30 | 2024-10-09 | JANSSEN Pharmaceutica NV | Dosing regimens associated with extended release paliperidone injectable formulations |
| JP2023551007A (ja) * | 2020-11-30 | 2023-12-06 | ヤンセン ファーマシューティカ エヌ．ベー． | パルミチン酸パリペリドン製剤の再懸濁を確実にする方法 |
| EP4025189B1 (en) | 2020-11-30 | 2024-06-05 | Janssen Pharmaceutica NV | Dosing regimens associated with extended release paliperidone injectable formulations |
| DK4025188T3 (da) * | 2020-11-30 | 2024-03-04 | Janssen Pharmaceutica Nv | Doseringsregimer associeret med injicerbare paliperidonformuleringer med forlænget frigivelse |
| CA3229731A1 (en) | 2021-08-20 | 2023-02-23 | Janssen Pharmaceutica Nv | Dosing regimens associated with extended release paliperidone injectable formulations |
| IL311134A (en) * | 2021-08-30 | 2024-04-01 | Janssen Pharmaceutica Nv | Dosing regimens associated with delayed-release paliperidone injection formulations |
| KR102869809B1 (ko) | 2023-11-21 | 2025-10-13 | 주식회사 엘지에너지솔루션 | 양극 및 이를 포함하는 전고체 전지 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110105536A1 (en) * | 2009-10-30 | 2011-05-05 | Lewyn-Briscoe Peter H | Dosing regimen associated with long-acting injectable paliperidone esters |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5158952A (en) | 1988-11-07 | 1992-10-27 | Janssen Pharmaceutica N.V. | 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use |
| US5254556A (en) | 1988-11-07 | 1993-10-19 | Janssen Pharmaceutica N.V. | 3-piperidinyl-1,2-benzisoxazoles |
| TW487572B (en) | 1996-05-20 | 2002-05-21 | Janssen Pharmaceutica Nv | Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters |
| UA72189C2 (uk) | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| EP1879890A1 (en) | 2005-04-25 | 2008-01-23 | Janssen Pharmaceutica N.V. | Preparation of aseptic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4h-pyridio[1,2-a]pyrimidin-4-one palmitate ester |
| SI2234617T2 (sl) * | 2007-12-19 | 2025-05-30 | Janssen Pharmaceutica Nv | Režim odmerjanja v zvezi z dolgodelujočimi paliperidonijevimi estri za injiciranje |
| US8758780B2 (en) * | 2009-10-06 | 2014-06-24 | Ascendis Pharma As | Subcutaneous paliperidone composition |
| PT2529757E (pt) * | 2011-05-31 | 2014-02-27 | Rovi Lab Farmaceut Sa | Formulação para implante de paliperidona |
| ES2802299T3 (es) | 2015-04-07 | 2021-01-18 | Janssen Pharmaceuticals Inc | Régimen de dosificación para dosis olvidadas para ésteres de paliperidona inyectables de acción prolongada |
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- 2016-03-30 ES ES16777058T patent/ES2802299T3/es active Active
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- 2016-03-30 DK DK16777058.5T patent/DK3280416T3/da active
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- 2016-03-30 IL IL309340A patent/IL309340A/en unknown
- 2016-03-30 MA MA41917A patent/MA41917B1/fr unknown
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- 2016-03-30 HU HUE20169861A patent/HUE065435T2/hu unknown
- 2016-03-30 SM SM20230478T patent/SMT202300478T1/it unknown
- 2016-03-30 MD MDE20180155T patent/MD3280416T2/ro unknown
- 2016-03-30 BR BR112017021383-4A patent/BR112017021383A2/pt not_active Application Discontinuation
- 2016-03-30 MD MDE20210632T patent/MD3744326T2/ro unknown
- 2016-03-30 KR KR1020177031672A patent/KR102606678B1/ko active Active
- 2016-04-01 TW TW105110443A patent/TWI694825B/zh active
- 2016-04-01 CA CA3088401A patent/CA3088401A1/en not_active Abandoned
- 2016-04-01 CA CA2925908A patent/CA2925908C/en active Active
- 2016-04-05 US US15/090,889 patent/US10143693B2/en active Active
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110105536A1 (en) * | 2009-10-30 | 2011-05-05 | Lewyn-Briscoe Peter H | Dosing regimen associated with long-acting injectable paliperidone esters |
Non-Patent Citations (3)
| Title |
|---|
| 【藥學雜誌】, Vol. 28, No. 2, Jun 30 2012「精神分裂症藥物 — Paliperidone Palmitate 之剖析」 |
| 【藥學雜誌】, Vol. 28, No. 2, Jun 30 2012「精神分裂症藥物 — Paliperidone Palmitate 之剖析」 Osborne et al. Health and Quality of Life Outcomes 2012, 10:35 http://www.hqlo.com/content/10/1/35 * |
| Osborne et al. Health and Quality of Life Outcomes 2012, 10:35 http://www.hqlo.com/content/10/1/35 |
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