TW348178B - Octacyclodepsipeptides having an action for killing endoparasites in animals - Google Patents

Octacyclodepsipeptides having an action for killing endoparasites in animals

Info

Publication number
TW348178B
TW348178B TW083102609A TW83102609A TW348178B TW 348178 B TW348178 B TW 348178B TW 083102609 A TW083102609 A TW 083102609A TW 83102609 A TW83102609 A TW 83102609A TW 348178 B TW348178 B TW 348178B
Authority
TW
Taiwan
Prior art keywords
octacyclodepsipeptides
animals
action
endoparasites
killing
Prior art date
Application number
TW083102609A
Other languages
English (en)
Inventor
Scherkenbeck Jurgen
Jeschker Peter
Lerchen Hans-Geofg
Hagemann Hermann
Harder Achim
Mencke Norbert
Plant Andrew
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Application granted granted Critical
Publication of TW348178B publication Critical patent/TW348178B/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
TW083102609A 1993-05-26 1994-03-25 Octacyclodepsipeptides having an action for killing endoparasites in animals TW348178B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4317432A DE4317432A1 (de) 1993-05-26 1993-05-26 Octacyclodepsipeptide mit endoparasitizider Wirkung

Publications (1)

Publication Number Publication Date
TW348178B true TW348178B (en) 1998-12-21

Family

ID=6488906

Family Applications (1)

Application Number Title Priority Date Filing Date
TW083102609A TW348178B (en) 1993-05-26 1994-03-25 Octacyclodepsipeptides having an action for killing endoparasites in animals

Country Status (10)

Country Link
US (2) US6468966B1 (zh)
EP (1) EP0626376A1 (zh)
JP (1) JP3535217B2 (zh)
KR (1) KR100357448B1 (zh)
AU (1) AU679724B2 (zh)
CA (1) CA2124054A1 (zh)
DE (1) DE4317432A1 (zh)
NZ (1) NZ260570A (zh)
TW (1) TW348178B (zh)
ZA (1) ZA943639B (zh)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4341992A1 (de) * 1993-12-09 1995-06-14 Bayer Ag Endoparasitizide Mittel auf Basis von offenkettigen Tetradepsipeptiden
DE4341993A1 (de) * 1993-12-09 1995-06-14 Bayer Ag Endoparasitizide Mittel auf Basis von offenkettigen Octadepsipeptiden
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
DE4437198A1 (de) * 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
DE4440193A1 (de) * 1994-11-10 1996-05-15 Bayer Ag Verwendung von Dioxomorpholinen zur Bekämpfung von Endoparasiten, neue Dioxomorpholine und Verfahren zur ihrer Herstellung
CA2228632A1 (en) * 1995-09-07 1997-03-13 William W. Mcwhorter, Jr. Cycloanthelmintic inhibitors
DE69634961T2 (de) * 1995-09-22 2006-04-20 Bayer Ag Neue zyklische depsipeptid pf1022 derivate
CA2267376C (en) * 1996-10-07 2006-11-14 Fujisawa Pharmaceutical Co., Ltd. Process for producing depsipeptide derivatives and novel intermediates therefor
DE19713626A1 (de) * 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung
CN1076349C (zh) * 1997-06-04 2001-12-19 拜尔公司 去氧环缩肽及其防治体内寄生虫的用途
DE19926622A1 (de) 1999-06-11 2000-12-14 Bayer Ag Thermoplastische Formmassen
DE19926620A1 (de) * 1999-06-11 2000-12-14 Bayer Ag Neue Cycloiminodepsipeptide, Verfahren zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Endoparasiten
DE19962147A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel / PF 1022-221
DE19962145A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel/Depsipeptide
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
ATE419373T1 (de) * 2002-11-12 2009-01-15 Kitasato Inst Anthelmintische substanz fki-1033 und verfahren zur herstellung davon
DE10358525A1 (de) 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
TWI276915B (en) * 2004-06-30 2007-03-21 Innolux Display Corp Photo-resist stripping process and equipment
US20060008492A1 (en) * 2004-07-09 2006-01-12 Pablo Janowicz Composition and method for delivering chemical agent to insects
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102005011779A1 (de) * 2005-03-11 2006-09-14 Bayer Healthcare Ag Endoparasitizide Mittel
DE102008022520A1 (de) * 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
DE102008030764A1 (de) 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031283A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
DE102008031284A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
DE102009012423A1 (de) * 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
EP2509967B1 (en) * 2009-12-11 2016-02-17 Bayer Intellectual Property GmbH Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
KR20150037766A (ko) 2012-06-13 2015-04-08 메이지 세이카 파루마 가부시키가이샤 신규한 환상 뎁시펩티드 유도체 및 이를 포함하는 해충 방제제
JP7045191B2 (ja) 2015-05-20 2022-03-31 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性デプシペプチド化合物
JP6943859B2 (ja) 2015-12-28 2021-10-06 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性デプシペプチド化合物
JP2020504710A (ja) * 2016-11-16 2020-02-13 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性デプシペプチド化合物
WO2019091975A1 (en) * 2017-11-07 2019-05-16 Bayer Animal Health Gmbh Method for the synthesis of cyclic depsipeptides
US11331369B2 (en) 2017-11-29 2022-05-17 Zoetis Services Llc Endoparasitic depsipeptides
WO2019217449A1 (en) 2018-05-10 2019-11-14 Zoetis Services Llc Endoparasitic depsipeptides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
JPH0570366A (ja) * 1991-03-08 1993-03-23 Meiji Seika Kaisha Ltd 薬用組成物
DE4341993A1 (de) * 1993-12-09 1995-06-14 Bayer Ag Endoparasitizide Mittel auf Basis von offenkettigen Octadepsipeptiden

Also Published As

Publication number Publication date
ZA943639B (en) 1995-01-27
US6468966B1 (en) 2002-10-22
DE4317432A1 (de) 1994-12-01
JP3535217B2 (ja) 2004-06-07
AU679724B2 (en) 1997-07-10
EP0626376A1 (de) 1994-11-30
KR100357448B1 (ko) 2003-01-08
US5717063A (en) 1998-02-10
JPH06340694A (ja) 1994-12-13
CA2124054A1 (en) 1994-11-27
AU6064194A (en) 1994-12-01
NZ260570A (en) 1996-01-26

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Legal Events

Date Code Title Description
MM4A Annulment or lapse of patent due to non-payment of fees