TW202404983A - Mci-1拮抗劑之鹽形式及溶劑化物 - Google Patents
Mci-1拮抗劑之鹽形式及溶劑化物 Download PDFInfo
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- TW202404983A TW202404983A TW112112762A TW112112762A TW202404983A TW 202404983 A TW202404983 A TW 202404983A TW 112112762 A TW112112762 A TW 112112762A TW 112112762 A TW112112762 A TW 112112762A TW 202404983 A TW202404983 A TW 202404983A
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202263327659P | 2022-04-05 | 2022-04-05 | |
| US63/327,659 | 2022-04-05 |
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|---|---|
| TW202404983A true TW202404983A (zh) | 2024-02-01 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW112112762A TW202404983A (zh) | 2022-04-05 | 2023-04-06 | Mci-1拮抗劑之鹽形式及溶劑化物 |
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| Country | Link |
|---|---|
| US (1) | US12351588B2 (enExample) |
| EP (1) | EP4504737A1 (enExample) |
| JP (1) | JP2025513774A (enExample) |
| AU (1) | AU2023249146A1 (enExample) |
| CA (1) | CA3254998A1 (enExample) |
| MX (1) | MX2024012192A (enExample) |
| TW (1) | TW202404983A (enExample) |
| UY (1) | UY40217A (enExample) |
| WO (1) | WO2023196360A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4519271A1 (en) | 2022-05-04 | 2025-03-12 | Gilead Sciences, Inc. | Salts and polymorphs of certain mcl-1 inhibitors |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JO3474B1 (ar) | 2014-08-29 | 2020-07-05 | Amgen Inc | مشتقات تيتراهيدرونافثالين التي تثبط بروتين mcl-1 |
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2023
- 2023-04-05 JP JP2024558381A patent/JP2025513774A/ja active Pending
- 2023-04-05 EP EP23724438.9A patent/EP4504737A1/en active Pending
- 2023-04-05 WO PCT/US2023/017504 patent/WO2023196360A1/en not_active Ceased
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- 2023-04-05 US US18/296,215 patent/US12351588B2/en active Active
- 2023-04-05 AU AU2023249146A patent/AU2023249146A1/en active Pending
- 2023-04-06 TW TW112112762A patent/TW202404983A/zh unknown
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Also Published As
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|---|---|
| CA3254998A1 (en) | 2023-10-12 |
| MX2024012192A (es) | 2024-11-08 |
| US20230312602A1 (en) | 2023-10-05 |
| JP2025513774A (ja) | 2025-04-30 |
| US12351588B2 (en) | 2025-07-08 |
| AU2023249146A1 (en) | 2024-10-10 |
| WO2023196360A1 (en) | 2023-10-12 |
| EP4504737A1 (en) | 2025-02-12 |
| UY40217A (es) | 2023-10-31 |
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