UY40217A - Formas de sal y solvatos de antagonistas de mci-1 - Google Patents

Formas de sal y solvatos de antagonistas de mci-1

Info

Publication number
UY40217A
UY40217A UY0001040217A UY40217A UY40217A UY 40217 A UY40217 A UY 40217A UY 0001040217 A UY0001040217 A UY 0001040217A UY 40217 A UY40217 A UY 40217A UY 40217 A UY40217 A UY 40217A
Authority
UY
Uruguay
Prior art keywords
salt
mci
solvates
antagonists
solvate forms
Prior art date
Application number
UY0001040217A
Other languages
English (en)
Spanish (es)
Inventor
D Parent Stephan
Travis Houston
Henry Morrison
S Tedrow Jason
Courtney Johnson
Melanie Bevill
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of UY40217A publication Critical patent/UY40217A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
UY0001040217A 2022-04-05 2023-04-10 Formas de sal y solvatos de antagonistas de mci-1 UY40217A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US202263327659P 2022-04-05 2022-04-05

Publications (1)

Publication Number Publication Date
UY40217A true UY40217A (es) 2023-10-31

Family

ID=86386785

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001040217A UY40217A (es) 2022-04-05 2023-04-10 Formas de sal y solvatos de antagonistas de mci-1

Country Status (9)

Country Link
US (1) US12351588B2 (enExample)
EP (1) EP4504737A1 (enExample)
JP (1) JP2025513774A (enExample)
AU (1) AU2023249146A1 (enExample)
CA (1) CA3254998A1 (enExample)
MX (1) MX2024012192A (enExample)
TW (1) TW202404983A (enExample)
UY (1) UY40217A (enExample)
WO (1) WO2023196360A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4519271A1 (en) 2022-05-04 2025-03-12 Gilead Sciences, Inc. Salts and polymorphs of certain mcl-1 inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3474B1 (ar) 2014-08-29 2020-07-05 Amgen Inc مشتقات تيتراهيدرونافثالين التي تثبط بروتين mcl-1

Also Published As

Publication number Publication date
CA3254998A1 (en) 2023-10-12
MX2024012192A (es) 2024-11-08
US20230312602A1 (en) 2023-10-05
TW202404983A (zh) 2024-02-01
JP2025513774A (ja) 2025-04-30
US12351588B2 (en) 2025-07-08
AU2023249146A1 (en) 2024-10-10
WO2023196360A1 (en) 2023-10-12
EP4504737A1 (en) 2025-02-12

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