TW200934771A - New compounds - Google Patents
New compoundsInfo
- Publication number
- TW200934771A TW200934771A TW097139967A TW97139967A TW200934771A TW 200934771 A TW200934771 A TW 200934771A TW 097139967 A TW097139967 A TW 097139967A TW 97139967 A TW97139967 A TW 97139967A TW 200934771 A TW200934771 A TW 200934771A
- Authority
- TW
- Taiwan
- Prior art keywords
- disease
- pain
- methyl
- compound
- triazol
- Prior art date
Links
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- General Chemical & Material Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
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| US98129407P | 2007-10-19 | 2007-10-19 |
Publications (1)
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| TW200934771A true TW200934771A (en) | 2009-08-16 |
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| TW097139967A TW200934771A (en) | 2007-10-19 | 2008-10-17 | New compounds |
Country Status (21)
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| US (1) | US7960422B2 (OSRAM) |
| EP (1) | EP2231647A4 (OSRAM) |
| JP (1) | JP2011500673A (OSRAM) |
| KR (1) | KR20100090777A (OSRAM) |
| CN (1) | CN101896480A (OSRAM) |
| AR (1) | AR068921A1 (OSRAM) |
| AU (1) | AU2008312055A1 (OSRAM) |
| BR (1) | BRPI0818448A2 (OSRAM) |
| CA (1) | CA2703425A1 (OSRAM) |
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| CR (1) | CR11376A (OSRAM) |
| DO (1) | DOP2010000119A (OSRAM) |
| EA (1) | EA201000654A1 (OSRAM) |
| IL (1) | IL204958A0 (OSRAM) |
| MX (1) | MX2010004272A (OSRAM) |
| PE (1) | PE20090875A1 (OSRAM) |
| TW (1) | TW200934771A (OSRAM) |
| UY (1) | UY31403A1 (OSRAM) |
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| EP1847543A1 (de) | 2006-04-19 | 2007-10-24 | Boehringer Ingelheim Pharma GmbH & Co. KG | Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen |
| BRPI0817781A2 (pt) * | 2007-10-19 | 2019-09-24 | Boehringer Ingelheim Int | piperazino-diidroteinopirimidinas substituídas com heterociclo |
| CA2702518A1 (en) | 2007-10-19 | 2009-04-23 | Boehringer Ingelheim International Gmbh | New piperazino-dihydrothienopyrimidine derivatives |
| PT2215092E (pt) * | 2007-10-19 | 2012-04-10 | Boehringer Ingelheim Int | Piperidino-di-hidrotienopirimidinas substituídas |
| AP3272A (en) | 2008-09-22 | 2015-05-31 | Cayman Chem Co | Multiheteroaryl compounds as inhibitors of H-PGDS and their use for treating prosaglandin D2 mediated diseases |
| CN102256967A (zh) * | 2008-12-18 | 2011-11-23 | 阿斯利康(瑞典)有限公司 | 制备3-{4-甲基-5-[(1r)-1-(2-(3-甲基苯基-2h-四唑-5-基)-乙氧基]-4h-[1,2,4]三唑-3-基}-吡啶、4-甲基-3-甲基硫基-5-(吡啶-3-基)-1,2,4-三唑和(1r)-1-[2-(3-甲基苯基)-2h-四唑-5-基]乙醇的方法 |
| US8883827B2 (en) | 2009-06-05 | 2014-11-11 | Oslo University Hospital Hf | Azole derivatives as WTN pathway inhibitors |
| JP2013544874A (ja) | 2010-12-08 | 2013-12-19 | オスロ ユニヴァーシティー ホスピタル エイチエフ | Ｗｎｔシグナル伝達経路阻害薬としてのトリアゾール誘導体 |
| MX2013010698A (es) | 2011-03-18 | 2014-02-17 | Novartis Ag | Combinaciones de activadores del receptor de acetil-colina nicotinico alfa-7 y antagonistas del receptor de glutamato metabotropico 5 (mglur5) para usarse en la discinesia inducida por dopamina en la enfermedad de parkinson. |
| US9802954B2 (en) | 2011-08-24 | 2017-10-31 | Boehringer Ingelheim International Gmbh | Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma |
| US20130059866A1 (en) | 2011-08-24 | 2013-03-07 | Boehringer Ingelheim International Gmbh | Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma |
| CN106032377A (zh) * | 2015-03-12 | 2016-10-19 | 天津药物研究院有限公司 | 四氮唑类urat1抑制剂、制备方法及其在高尿酸血症和痛风治疗上的用途 |
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| US4663332A (en) | 1985-10-10 | 1987-05-05 | Hoffman-La Roche Inc. | 5-substituted N-alkylated tetrazoles |
| AU2363492A (en) | 1991-08-03 | 1993-03-02 | Smithkline Beecham Plc | 5-ht4 receptor antagonists |
| DE10023430A1 (de) | 2000-05-12 | 2001-11-15 | Bayer Ag | Substituierte N-Benzoyl-N'-(tetrazolylphenyl)-harnstoffe |
| GB0115862D0 (en) | 2001-06-28 | 2001-08-22 | Smithkline Beecham Plc | Compounds |
| GB0121033D0 (en) | 2001-08-30 | 2001-10-24 | Novartis Ag | Organic compounds |
| ATE396186T1 (de) | 2001-10-04 | 2008-06-15 | Merck & Co Inc | Heteroarylsubstituierte tetrazolmodulatoren des metabotropischen glutamatrezeptors-5 |
| US7592337B2 (en) | 2002-03-12 | 2009-09-22 | Merck & Co., Inc. | Di-aryl substituted tetrazole modulators of metabotropic glutamate receptor-5 |
| PL375256A1 (en) * | 2002-08-09 | 2005-11-28 | Astra Zeneca Ab | 1,2,4-oxadiazoles as modulators of metabotropic glutamate receptor-5 |
| WO2005077345A1 (en) | 2004-02-03 | 2005-08-25 | Astrazeneca Ab | Compounds for the treatment of gastro-esophageal reflux disease |
| UA85576C2 (ru) * | 2004-02-18 | 2009-02-10 | Астразенека Аб | Тетразольные соединения и их применение в качестве метаботропических антагонистов рецепторов глутамата |
| RU2006127575A (ru) * | 2004-02-18 | 2008-03-27 | Астразенека Аб (Se) | Соединение триазола и их применение в качестве антагонистов метаботропного рецептора глутамата |
| NZ548693A (en) | 2004-02-18 | 2010-05-28 | Astrazeneca Ab | Polyheterocyclic compounds and their use as metabotropic glutamate receptor antagonists |
| US7585881B2 (en) | 2004-02-18 | 2009-09-08 | Astrazeneca Ab | Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
| UY29796A1 (es) | 2005-09-29 | 2007-04-30 | Astrazeneca Ab | Nuevos compuestos para el tratamiento de trastornos neurológicos, psiquiátricos o del dolor |
| TW200811156A (en) | 2006-05-05 | 2008-03-01 | Astrazeneca Ab | mGluR5 modulators IV |
| TW200811157A (en) | 2006-05-05 | 2008-03-01 | Astrazeneca Ab | mGluR5 modulators I |
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2008
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2010
- 2010-04-08 IL IL204958A patent/IL204958A0/en unknown
- 2010-04-16 ZA ZA2010/02694A patent/ZA201002694B/en unknown
- 2010-04-19 DO DO2010000119A patent/DOP2010000119A/es unknown
- 2010-04-19 CR CR11376A patent/CR11376A/es not_active Application Discontinuation
- 2010-04-28 CO CO10050285A patent/CO6321281A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AR068921A1 (es) | 2009-12-16 |
| ZA201002694B (en) | 2011-03-30 |
| EP2231647A1 (en) | 2010-09-29 |
| US7960422B2 (en) | 2011-06-14 |
| CO6321281A2 (es) | 2011-09-20 |
| EA201000654A1 (ru) | 2010-12-30 |
| UY31403A1 (es) | 2009-05-29 |
| MX2010004272A (es) | 2010-04-30 |
| CL2008003085A1 (es) | 2009-10-09 |
| AU2008312055A1 (en) | 2009-04-23 |
| CA2703425A1 (en) | 2009-04-23 |
| EP2231647A4 (en) | 2011-08-31 |
| BRPI0818448A2 (pt) | 2015-05-12 |
| WO2009051556A1 (en) | 2009-04-23 |
| JP2011500673A (ja) | 2011-01-06 |
| CR11376A (es) | 2010-07-19 |
| PE20090875A1 (es) | 2009-08-08 |
| DOP2010000119A (es) | 2010-05-31 |
| CN101896480A (zh) | 2010-11-24 |
| IL204958A0 (en) | 2010-11-30 |
| US20090131454A1 (en) | 2009-05-21 |
| KR20100090777A (ko) | 2010-08-17 |
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