TW200420561A - Antimicrobial 1-aryl dihydropyridone compounds - Google Patents

Antimicrobial 1-aryl dihydropyridone compounds

Info

Publication number
TW200420561A
TW200420561A TW092127838A TW92127838A TW200420561A TW 200420561 A TW200420561 A TW 200420561A TW 092127838 A TW092127838 A TW 092127838A TW 92127838 A TW92127838 A TW 92127838A TW 200420561 A TW200420561 A TW 200420561A
Authority
TW
Taiwan
Prior art keywords
antimicrobial
aryl
dihydropyridone compounds
dihydropyridone
compounds
Prior art date
Application number
TW092127838A
Other languages
English (en)
Inventor
Mikhail Fedor Gordeev
Upinder Singh
Dinesh Vinoobhai Patel
Paul Dennis May
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of TW200420561A publication Critical patent/TW200420561A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
TW092127838A 2002-10-10 2003-10-07 Antimicrobial 1-aryl dihydropyridone compounds TW200420561A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41749202P 2002-10-10 2002-10-10

Publications (1)

Publication Number Publication Date
TW200420561A true TW200420561A (en) 2004-10-16

Family

ID=32094028

Family Applications (1)

Application Number Title Priority Date Filing Date
TW092127838A TW200420561A (en) 2002-10-10 2003-10-07 Antimicrobial 1-aryl dihydropyridone compounds

Country Status (10)

Country Link
US (1) US7105547B2 (zh)
EP (1) EP1554273A1 (zh)
JP (1) JP2006504726A (zh)
AR (1) AR041556A1 (zh)
AU (1) AU2003265090A1 (zh)
BR (1) BR0315206A (zh)
CA (1) CA2499105A1 (zh)
MX (1) MXPA05003774A (zh)
TW (1) TW200420561A (zh)
WO (1) WO2004033449A1 (zh)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7208490B2 (en) 2002-10-07 2007-04-24 Pharmacia & Upjohn Company Llc Tricyclic tetrahydroquinoline antibacterial agents
CN101720325B (zh) * 2007-08-06 2013-04-24 上海盟科药业有限公司 用于治疗细菌感染的抗菌邻-氟苯基噁唑烷酮
CN101798302B (zh) 2009-02-06 2014-11-05 上海盟科药业有限公司 抗生素类药物1-(邻-氟苯基)二氢吡啶酮的合成及生产的方法和工艺
CN102206213A (zh) * 2010-03-31 2011-10-05 盟科医药技术(上海)有限公司 (5s)-5-[(异噁唑-3-基氨基)甲基]-3-[2,3,5-三氟-4-(4-氧代-2,3-二氢吡啶-1-基)苯基]噁唑烷-2-酮的药物晶型
WO2015127316A1 (en) 2014-02-21 2015-08-27 Micurx Pharmaceuticals, Inc. Water-soluble o-carbonyl phosphoramidate prodrugs for therapeutic administration
CN108727406B (zh) * 2017-03-28 2021-12-07 北京协和制药二厂 含氮杂环取代的苯并噁嗪噁唑烷酮类化合物及其制备方法和用途

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK283420B6 (sk) 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
US5668286A (en) 1994-03-15 1997-09-16 Pharmacia & Upjohn Company Oxazolidinone derivatives and pharmaceutical compositions containing them
ATE293609T1 (de) * 1997-05-30 2005-05-15 Upjohn Co Antibakteriell wirksam oxazolidinone mit einer thiocarbonylfunktionalität
ATE222894T1 (de) 1998-02-13 2002-09-15 Upjohn Co Substituierte aminophenylisoxazolinderivate verwendbar als antimikrobielle agenzien
TW572757B (en) * 1998-08-24 2004-01-21 Bristol Myers Squibb Co Novel isoxazolinone antibacterial agents
EP1472247A1 (en) * 2002-02-05 2004-11-03 PHARMACIA & UPJOHN COMPANY Antimicrobial thiadiazinone derivatives useful in treatment of bacterial infections
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados

Also Published As

Publication number Publication date
AU2003265090A1 (en) 2004-05-04
US20050070580A1 (en) 2005-03-31
EP1554273A1 (en) 2005-07-20
CA2499105A1 (en) 2004-04-22
JP2006504726A (ja) 2006-02-09
WO2004033449A1 (en) 2004-04-22
MXPA05003774A (es) 2005-06-08
US7105547B2 (en) 2006-09-12
BR0315206A (pt) 2005-08-16
AR041556A1 (es) 2005-05-18

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