TR200102436T2 - 5-HT1F agonistleri - Google Patents
5-HT1F agonistleriInfo
- Publication number
- TR200102436T2 TR200102436T2 TR2001/02436T TR200102436T TR200102436T2 TR 200102436 T2 TR200102436 T2 TR 200102436T2 TR 2001/02436 T TR2001/02436 T TR 2001/02436T TR 200102436 T TR200102436 T TR 200102436T TR 200102436 T2 TR200102436 T2 TR 200102436T2
- Authority
- TR
- Turkey
- Prior art keywords
- ht1f agonists
- ht1f
- agonists
- vascularization
- mammal
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Hospice & Palliative Care (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Anesthesiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Bu bulus, bir memelide 4-HT1F reseptörlerinin aktive edilmesinde ve nöron proteininin damar disina sizmasinin inhibe edilmesinde faydali olan, formül (i)'e sahip bir bilesige veya bunun farmasötik bir asit ilave iliskindir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12201699P | 1999-02-26 | 1999-02-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200102436T2 true TR200102436T2 (tr) | 2002-06-21 |
Family
ID=22400069
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2001/02436T TR200102436T2 (tr) | 1999-02-26 | 2000-02-11 | 5-HT1F agonistleri |
Country Status (21)
Country | Link |
---|---|
EP (1) | EP1155020B1 (tr) |
JP (1) | JP2002537398A (tr) |
KR (1) | KR20010102355A (tr) |
AR (1) | AR026856A1 (tr) |
AT (1) | ATE258935T1 (tr) |
AU (1) | AU3354000A (tr) |
BR (1) | BR0008479A (tr) |
CA (1) | CA2371784A1 (tr) |
CO (1) | CO5150234A1 (tr) |
DE (1) | DE60008073T2 (tr) |
EA (1) | EA200100918A1 (tr) |
ES (1) | ES2214256T3 (tr) |
HU (1) | HUP0200245A2 (tr) |
ID (1) | ID30056A (tr) |
IL (1) | IL144355A0 (tr) |
NO (1) | NO20014127D0 (tr) |
PE (1) | PE20001432A1 (tr) |
PL (1) | PL350864A1 (tr) |
TR (1) | TR200102436T2 (tr) |
WO (1) | WO2000050426A2 (tr) |
ZA (1) | ZA200106109B (tr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI263497B (en) | 2002-03-29 | 2006-10-11 | Lilly Co Eli | Pyridinoylpiperidines as 5-HT1F agonists |
WO2004094380A1 (en) | 2003-04-18 | 2004-11-04 | Eli Lilly And Company | (piperidinyloxy)phenyl, (piperidinyloxy)pyridinyl, (piperidinylsulfanyl)phenyl and (piperidinylsulfanyl)pyridinyl compounds as 5-ht1f agonists |
UA82711C2 (en) | 2003-09-12 | 2008-05-12 | Эли Лилли Энд Компани | Substituted 2-carbonylamino-6-piperidinaminopyridines and substituted 1-carbonylamino-3-piperidinaminobenzenes as 5-ht1f agonists |
JP2007516266A (ja) | 2003-12-17 | 2007-06-21 | イーライ リリー アンド カンパニー | 5−ht1fアゴニストとしての置換(4−アミノシクロヘキセン−1−イル)フェニルおよび(4−アミノシクロヘキセン−1−イル)ピリジニル化合物 |
WO2011123654A1 (en) | 2010-04-02 | 2011-10-06 | Colucid Pharmaceuticals, Inc. | Compositions and methods of synthesis of pyridinoylpiperidine 5-ht1f agonists |
EP2940022B1 (en) * | 2014-04-30 | 2020-09-02 | Masarykova Univerzita | Furopyridines as inhibitors of protein kinases |
AR119319A1 (es) | 2019-07-09 | 2021-12-09 | Lilly Co Eli | Procesos e intermediario para la preparación a gran escala de hemisuccinato de 2,4,6-trifluoro-n-[6-(1-metil-piperidina-4-carbonil)-piridin-2-il]-benzamida y preparación de acetato de 2,4,6-trifluoro-n-[6-(1-metil-piperidina-4-carbonil)-piridin-2-il]-benzamida |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX9706969A (es) * | 1995-03-20 | 1997-11-29 | Lilly Co Eli | 3-(1,2,3,6-tetrahidropiridin-4-il)-1h-indoles y 3-(piperidin-4-il)-1h-indoles sustituidos en la posicion 5: agonistas del 5-ht1f novedosos. |
FR2732969B1 (fr) * | 1995-04-14 | 1997-05-16 | Adir | Nouveaux composes pyridiniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
AU4074897A (en) * | 1996-09-18 | 1998-04-14 | Eli Lilly And Company | A method for the prevention of migraine |
-
2000
- 2000-02-11 CA CA002371784A patent/CA2371784A1/en not_active Abandoned
- 2000-02-11 TR TR2001/02436T patent/TR200102436T2/tr unknown
- 2000-02-11 KR KR1020017010743A patent/KR20010102355A/ko not_active Application Discontinuation
- 2000-02-11 BR BR0008479-4A patent/BR0008479A/pt not_active Application Discontinuation
- 2000-02-11 EP EP00911678A patent/EP1155020B1/en not_active Expired - Lifetime
- 2000-02-11 ID IDW00200101739D patent/ID30056A/id unknown
- 2000-02-11 DE DE60008073T patent/DE60008073T2/de not_active Expired - Fee Related
- 2000-02-11 PL PL00350864A patent/PL350864A1/xx not_active Application Discontinuation
- 2000-02-11 HU HU0200245A patent/HUP0200245A2/hu unknown
- 2000-02-11 IL IL14435500A patent/IL144355A0/xx unknown
- 2000-02-11 WO PCT/US2000/002505 patent/WO2000050426A2/en not_active Application Discontinuation
- 2000-02-11 AU AU33540/00A patent/AU3354000A/en not_active Abandoned
- 2000-02-11 AT AT00911678T patent/ATE258935T1/de not_active IP Right Cessation
- 2000-02-11 EA EA200100918A patent/EA200100918A1/ru unknown
- 2000-02-11 ES ES00911678T patent/ES2214256T3/es not_active Expired - Lifetime
- 2000-02-11 JP JP2000601006A patent/JP2002537398A/ja not_active Withdrawn
- 2000-02-24 AR ARP000100791A patent/AR026856A1/es unknown
- 2000-02-24 CO CO00013084A patent/CO5150234A1/es unknown
- 2000-02-24 PE PE2000000153A patent/PE20001432A1/es not_active Application Discontinuation
-
2001
- 2001-07-25 ZA ZA200106109A patent/ZA200106109B/en unknown
- 2001-08-24 NO NO20014127A patent/NO20014127D0/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL144355A0 (en) | 2002-05-23 |
CA2371784A1 (en) | 2000-08-31 |
CO5150234A1 (es) | 2002-04-29 |
KR20010102355A (ko) | 2001-11-15 |
DE60008073T2 (de) | 2004-08-05 |
NO20014127L (no) | 2001-08-24 |
WO2000050426A3 (en) | 2000-12-21 |
ES2214256T3 (es) | 2004-09-16 |
HUP0200245A2 (en) | 2002-06-29 |
ZA200106109B (en) | 2002-07-25 |
EP1155020A2 (en) | 2001-11-21 |
AU3354000A (en) | 2000-09-14 |
PL350864A1 (en) | 2003-02-10 |
EA200100918A1 (ru) | 2002-02-28 |
NO20014127D0 (no) | 2001-08-24 |
ID30056A (id) | 2001-11-01 |
JP2002537398A (ja) | 2002-11-05 |
EP1155020B1 (en) | 2004-02-04 |
ATE258935T1 (de) | 2004-02-15 |
PE20001432A1 (es) | 2000-12-18 |
AR026856A1 (es) | 2003-03-05 |
DE60008073D1 (de) | 2004-03-11 |
BR0008479A (pt) | 2002-01-29 |
WO2000050426A2 (en) | 2000-08-31 |
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